FR2784993B1 - Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme fongicides - Google Patents
Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme fongicidesInfo
- Publication number
- FR2784993B1 FR2784993B1 FR9813361A FR9813361A FR2784993B1 FR 2784993 B1 FR2784993 B1 FR 2784993B1 FR 9813361 A FR9813361 A FR 9813361A FR 9813361 A FR9813361 A FR 9813361A FR 2784993 B1 FR2784993 B1 FR 2784993B1
- Authority
- FR
- France
- Prior art keywords
- fungicides
- application
- preparation process
- echinocandin derivatives
- novel
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Peptides Or Proteins (AREA)
Priority Applications (52)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
UA2000074030A UA72200C2 (uk) | 1997-12-10 | 1998-09-12 | Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція |
FR9813361A FR2784993B1 (fr) | 1998-10-26 | 1998-10-26 | Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme fongicides |
TNTNSN98222A TNSN98222A1 (fr) | 1997-12-10 | 1998-12-08 | Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongicides |
AU15659/99A AU755033B2 (en) | 1997-12-10 | 1998-12-09 | Echinocandin derivatives, preparation method and application as anti-fungal agents |
IL13664798A IL136647A0 (en) | 1997-12-10 | 1998-12-09 | Echinocandin derivatives, preparation method and application as anti-fungal agents |
MA25378A MA26575A1 (fr) | 1997-12-10 | 1998-12-09 | Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongicides. |
CN98813413A CN1284084A (zh) | 1997-12-10 | 1998-12-09 | 棘白菌素衍生物、其制备方法及其作为抗真菌剂的用途 |
ES98959935T ES2259462T3 (es) | 1997-12-10 | 1998-12-09 | Derivados de la equinocandina, procedimiento de preparacion y su aplicacion como agentes antifungicos. |
CZ20002113A CZ301919B6 (cs) | 1997-12-10 | 1998-12-09 | Deriváty echinokandinu, zpusob jejich prípravy, nové chemické produkty, použití derivátu echinokandinu a farmaceutické prostredky obsahující tyto deriváty echinokandinu |
EP98959935A EP1036090B1 (fr) | 1997-12-10 | 1998-12-09 | Derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques |
YUP-339/00A RS49905B (sr) | 1997-12-10 | 1998-12-09 | Derivati ehinokandina, postupak za njihovo dobijanje i njihova primena kao antifungicida |
JP2000524307A JP4361679B2 (ja) | 1997-12-10 | 1998-12-09 | エキノカンジン誘導体、それらの製造方法及びそれらの抗真菌剤としての使用 |
DZ980280A DZ2670A1 (fr) | 1997-12-10 | 1998-12-09 | Nouveaux dérivés de l'échinocandine leur procédé de préparation et leur application comme anti-fongiques. |
EEP200000336A EE04837B1 (et) | 1997-12-10 | 1998-12-09 | Ehhinokandiini derivaadid, nende valmistamismeetod ja kasutamine antimükootikumidena |
APAP/P/2000/001826A AP1260A (en) | 1997-12-10 | 1998-12-09 | Echinocandin derivatives, preparation method and application as anti-fungal agents. |
EA200000625A EA002706B1 (ru) | 1997-12-10 | 1998-12-09 | Производные эхинокандина, способ их получения и их применение в качестве противогрибковых средств |
SK839-2000A SK286916B6 (sk) | 1997-12-10 | 1998-12-09 | Deriváty echinokandínu, spôsob ich prípravy a ich aplikácia ako antifungálnych činidiel |
SI9830834T SI1036090T1 (sl) | 1997-12-10 | 1998-12-09 | Derivati ehinokandina, postopek za njihovo pripravo in njihova uporaba kot protiglivicna sredstva |
DE69834057T DE69834057T2 (de) | 1997-12-10 | 1998-12-09 | Echinocandinderivate, deren herstellung und deren verwendung zur bekämpfung von pilzen |
HU0100263A HUP0100263A3 (en) | 1997-12-10 | 1998-12-09 | Echinocandin derivatives, preparation method and application as anti-fungal agents |
PT98959935T PT1036090E (pt) | 1997-12-10 | 1998-12-09 | Derivados da equinocandina, seu processo de preparacao e sua aplicacao como antifungicos |
NZ504614A NZ504614A (en) | 1997-12-10 | 1998-12-09 | Echinocandin derivatives and application as anti-fungal agents |
PL341012A PL196889B1 (pl) | 1997-12-10 | 1998-12-09 | Pochodne echinokandyny, sposób wytwarzania pochodnej echinokandyny, jej zastosowanie jako substancji przeciwgrzybicznej oraz zawierająca ją kompozycja farmaceutyczna |
BR9813531-7A BR9813531A (pt) | 1997-12-10 | 1998-12-09 | "derivados da equinocandina, seu processo de preparo e sua aplicação como antifúngicos" |
OA00000164A OA11899A (fr) | 1997-12-10 | 1998-12-09 | Dérivés de l'échinocandine, leur procédé de préparation et leur application comme anti-fongiques. |
KR1020007006268A KR100564872B1 (ko) | 1997-12-10 | 1998-12-09 | 에키노칸딘 유도체, 그의 제조 방법 및 항진균제로서의 응용 |
AT98959935T ATE321772T1 (de) | 1997-12-10 | 1998-12-09 | Echinocandinderivate, deren herstellung und deren verwendung zur bekämpfung von pilzen |
APAP/P/2003/002874A AP1567A (en) | 1997-12-10 | 1998-12-09 | Echinocandin derivatives, preparation method and application as anti-fungal agents. |
US09/581,451 US6677429B1 (en) | 1997-12-10 | 1998-12-09 | Echinocandin derivatives, preparation method and application as anti-fungal agents |
CA002311295A CA2311295A1 (fr) | 1997-12-10 | 1998-12-09 | Derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques |
GEAP19985441A GEP20032975B (en) | 1997-12-10 | 1998-12-09 | Echinocandin Derivatives, Preparation Method and Pharmaceutical Composition |
PA19988464201A PA8464201A1 (es) | 1997-12-10 | 1998-12-09 | Nuevos derivados de la equinocandina, su procedimiento de preparacion y su aplicacion como fungicidas |
DK98959935T DK1036090T3 (da) | 1997-12-10 | 1998-12-09 | Echinocandinderivater, fremgangsmåde til deres fremstilling samt deres anvendelse som antifungale midler |
PCT/FR1998/002671 WO1999029716A1 (fr) | 1997-12-10 | 1998-12-09 | Derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques |
TR2000/01655T TR200001655T2 (tr) | 1997-12-10 | 1998-12-09 | Ekinokandin türevleri, hazırlama yöntemi ve anti-fungal maddeler |
UY25292A UY25292A1 (es) | 1997-12-10 | 1998-12-09 | Nuevos derivados de la equinocandina, su procedimiento de preparación y su aplicación como fungicidas. |
PE1998001202A PE130099A1 (es) | 1997-12-10 | 1998-12-10 | Nuevos derivados de la equinocandina, su procedimiento de preparacion y su aplicacion como fungicidas |
ARP980106281A AR016432A1 (es) | 1997-12-10 | 1998-12-10 | Derivados de la equinocandina, su procedimiento de preparacion, compuestos intermediarios y composiciones farmaceuticas. |
CO98073452A CO4980875A1 (es) | 1997-12-10 | 1998-12-10 | Nuevos derivados de la equinocandina, su procedimiento de preparacion y su aplicacion como fungicidas |
TW087121185A TW446541B (en) | 1997-12-10 | 1999-01-22 | New derivatives of echinocandine, their preparation process and their use as fungicides |
GT199900026A GT199900026A (es) | 1998-10-26 | 1999-02-26 | Nuevos derivados de la equinocandina, su procedimiento de preparacion y su aplicacion como fungicidas. |
SA99191248A SA99191248B1 (ar) | 1997-12-10 | 1999-04-05 | مشتقات اكينوكاندين echinocandin وطريقة تحضيرها واستخدامها كمضادات للفطريات anti-fungal |
BG104494A BG65033B1 (bg) | 1997-12-10 | 2000-05-31 | Производни на ехинокандин, метод за тяхното получаване и използването им като противогъбично средство |
CU20000136A CU22962A3 (es) | 1997-12-10 | 2000-06-07 | Derivados de la equinocandia, su procedimiento de preparación y su aplicación como antifúngicos |
IL136647A IL136647A (en) | 1997-12-10 | 2000-06-08 | History of Echinocandin, method of preparation and use as antifungal preparations |
NO20002959A NO327498B1 (no) | 1997-12-10 | 2000-06-09 | Echinocandinderivater, fremgangsmate for fremstilling av slike, antifungale forbindelser og farmasoytiske preparater inneholdende disse forbindelser. |
HR20000384A HRP20000384B1 (en) | 1997-12-10 | 2000-06-09 | Echinocandin derivatives, preparation method and application as anti-fungla agents |
US10/666,072 US7160983B2 (en) | 1997-12-10 | 2003-09-19 | Echinocandin derivatives, their method of preparation and their application as anti-fungal agents |
US11/165,458 US7285619B2 (en) | 1997-12-10 | 2005-06-23 | Echinocandin derivatives, their method of preparation and their application as anti-fungal agents |
IL172412A IL172412A (en) | 1997-12-10 | 2005-12-06 | History of Echinocandin, method of preparation and use as antifungal preparations |
CY20061100686T CY1105695T1 (el) | 1997-12-10 | 2006-05-30 | Παραγωγα της εχινοκανδινης, μεθοδος παρασκευης τους και εφαρμογη τους σαν αντι-μυκητιασικα |
IL184171A IL184171A0 (en) | 1997-12-10 | 2007-06-24 | Echinocandin derivatives, preparation method and application as anti-fungal agents |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9813361A FR2784993B1 (fr) | 1998-10-26 | 1998-10-26 | Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme fongicides |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2784993A1 FR2784993A1 (fr) | 2000-04-28 |
FR2784993B1 true FR2784993B1 (fr) | 2002-10-31 |
Family
ID=9531958
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR9813361A Expired - Fee Related FR2784993B1 (fr) | 1997-12-10 | 1998-10-26 | Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme fongicides |
Country Status (2)
Country | Link |
---|---|
FR (1) | FR2784993B1 (fr) |
GT (1) | GT199900026A (fr) |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB2241955A (en) * | 1990-03-16 | 1991-09-18 | Merck & Co Inc | Cyclohexapeptide compounds |
TW264477B (fr) * | 1992-03-19 | 1995-12-01 | Lilly Co Eli | |
US5516757A (en) * | 1994-09-16 | 1996-05-14 | Merck & Co., Inc. | Semi-synthetic lipopeptides, compositions containing said lipopeptides, and methods of use |
US5516756A (en) * | 1994-10-31 | 1996-05-14 | Merck & Co., Inc. | Aza cyclohexapeptide compounds |
ES2162039T3 (es) * | 1995-01-26 | 2001-12-16 | Merck & Co Inc | Nuevos ciclohexapeptidos antifungicos. |
US5646111A (en) * | 1995-04-07 | 1997-07-08 | Eli Lilly And Company | Cyclic peptide antifungal Agents |
-
1998
- 1998-10-26 FR FR9813361A patent/FR2784993B1/fr not_active Expired - Fee Related
-
1999
- 1999-02-26 GT GT199900026A patent/GT199900026A/es unknown
Also Published As
Publication number | Publication date |
---|---|
FR2784993A1 (fr) | 2000-04-28 |
GT199900026A (es) | 2000-08-19 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
TP | Transmission of property | ||
CA | Change of address | ||
TP | Transmission of property | ||
ST | Notification of lapse |
Effective date: 20130628 |