UY25292A1 - Nuevos derivados de la equinocandina, su procedimiento de preparación y su aplicación como fungicidas. - Google Patents

Nuevos derivados de la equinocandina, su procedimiento de preparación y su aplicación como fungicidas.

Info

Publication number
UY25292A1
UY25292A1 UY25292A UY25292A UY25292A1 UY 25292 A1 UY25292 A1 UY 25292A1 UY 25292 A UY25292 A UY 25292A UY 25292 A UY25292 A UY 25292A UY 25292 A1 UY25292 A1 UY 25292A1
Authority
UY
Uruguay
Prior art keywords
echinocandine
fungicides
application
preparation procedure
new derivatives
Prior art date
Application number
UY25292A
Other languages
English (en)
Inventor
Olivier Courtin
Manguer Dominique Melon
Patrick Faveau
Jean Marc Michel
Astrid Markus
Laurent Schio Laurent Schio
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9715628A external-priority patent/FR2772028B1/fr
Priority claimed from FR9813361A external-priority patent/FR2784993B1/fr
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of UY25292A1 publication Critical patent/UY25292A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/18—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50—Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Detergent Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Compuestos de fórmula (i), así como sus sales que presentan propiedades antifúngicas especialmente útiles en candidiasis, criptococosis y aspergillosis.
UY25292A 1997-12-10 1998-12-09 Nuevos derivados de la equinocandina, su procedimiento de preparación y su aplicación como fungicidas. UY25292A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9715628A FR2772028B1 (fr) 1997-12-10 1997-12-10 Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme fongicides
FR9813361A FR2784993B1 (fr) 1998-10-26 1998-10-26 Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme fongicides

Publications (1)

Publication Number Publication Date
UY25292A1 true UY25292A1 (es) 2000-12-29

Family

ID=26233984

Family Applications (1)

Application Number Title Priority Date Filing Date
UY25292A UY25292A1 (es) 1997-12-10 1998-12-09 Nuevos derivados de la equinocandina, su procedimiento de preparación y su aplicación como fungicidas.

Country Status (43)

Country Link
US (3) US6677429B1 (es)
EP (1) EP1036090B1 (es)
JP (1) JP4361679B2 (es)
KR (1) KR100564872B1 (es)
CN (1) CN1284084A (es)
AP (2) AP1260A (es)
AR (1) AR016432A1 (es)
AT (1) ATE321772T1 (es)
AU (1) AU755033B2 (es)
BG (1) BG65033B1 (es)
BR (1) BR9813531A (es)
CA (1) CA2311295A1 (es)
CO (1) CO4980875A1 (es)
CU (1) CU22962A3 (es)
CY (1) CY1105695T1 (es)
CZ (1) CZ301919B6 (es)
DE (1) DE69834057T2 (es)
DK (1) DK1036090T3 (es)
DZ (1) DZ2670A1 (es)
EA (1) EA002706B1 (es)
EE (1) EE04837B1 (es)
ES (1) ES2259462T3 (es)
GE (1) GEP20032975B (es)
HR (1) HRP20000384B1 (es)
HU (1) HUP0100263A3 (es)
IL (4) IL136647A0 (es)
MA (1) MA26575A1 (es)
NO (1) NO327498B1 (es)
NZ (1) NZ504614A (es)
OA (1) OA11899A (es)
PA (1) PA8464201A1 (es)
PE (1) PE130099A1 (es)
PL (1) PL196889B1 (es)
PT (1) PT1036090E (es)
RS (1) RS49905B (es)
SA (1) SA99191248B1 (es)
SK (1) SK286916B6 (es)
TN (1) TNSN98222A1 (es)
TR (1) TR200001655T2 (es)
TW (1) TW446541B (es)
UA (1) UA72200C2 (es)
UY (1) UY25292A1 (es)
WO (1) WO1999029716A1 (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA72200C2 (uk) * 1997-12-10 2005-02-15 Авентіс Фарма С.А. Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція
WO2000024694A1 (en) * 1998-10-28 2000-05-04 Eli Lilly And Company Photochemical process for making 1-deoxy-2-keto derivatives
FR2794746B1 (fr) * 1999-06-09 2002-12-06 Hoechst Marion Roussel Inc Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques
FR2794747B1 (fr) * 1999-06-09 2004-04-16 Hoechst Marion Roussel Inc Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques
FR2833596B1 (fr) * 2001-12-14 2005-02-18 Aventis Pharma Sa Procede de preparation de derives d'echinocandine
CN101659693B (zh) * 2008-08-27 2012-11-21 上海医药工业研究院 制备纽莫康定b0的方法
CN101659692B (zh) * 2008-08-27 2012-07-04 上海医药工业研究院 制备棘球康定b的方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2241955A (en) * 1990-03-16 1991-09-18 Merck & Co Inc Cyclohexapeptide compounds
IL105048A (en) * 1992-03-19 2001-06-14 Eli Lilly And Company U S Antifungal substances of the cyclic peptide type and a process for their preparation
US5516757A (en) 1994-09-16 1996-05-14 Merck & Co., Inc. Semi-synthetic lipopeptides, compositions containing said lipopeptides, and methods of use
US5516756A (en) 1994-10-31 1996-05-14 Merck & Co., Inc. Aza cyclohexapeptide compounds
ATE206054T1 (de) 1995-01-26 2001-10-15 Merck & Co Inc Neue fungizide cyclohexapeptide
US5646111A (en) * 1995-04-07 1997-07-08 Eli Lilly And Company Cyclic peptide antifungal Agents
UA72200C2 (uk) * 1997-12-10 2005-02-15 Авентіс Фарма С.А. Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція
FR2794747B1 (fr) * 1999-06-09 2004-04-16 Hoechst Marion Roussel Inc Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques

Also Published As

Publication number Publication date
OA11899A (fr) 2006-04-10
HRP20000384A2 (en) 2000-10-31
US20050267019A1 (en) 2005-12-01
MA26575A1 (fr) 2004-12-20
GEP20032975B (en) 2003-05-27
EA002706B1 (ru) 2002-08-29
AP2000001826A0 (en) 2000-06-30
HUP0100263A3 (en) 2002-11-28
CN1284084A (zh) 2001-02-14
ES2259462T3 (es) 2006-10-01
SK286916B6 (sk) 2009-07-06
NO327498B1 (no) 2009-07-20
NO20002959L (no) 2000-08-09
EA200000625A1 (ru) 2000-12-25
ATE321772T1 (de) 2006-04-15
IL136647A (en) 2007-06-03
US7285619B2 (en) 2007-10-23
HRP20000384B1 (en) 2010-02-28
AR016432A1 (es) 2001-07-04
CU22962A3 (es) 2004-06-21
CY1105695T1 (el) 2010-12-22
UA72200C2 (uk) 2005-02-15
SA99191248B1 (ar) 2006-08-12
AU755033B2 (en) 2002-11-28
EP1036090A1 (fr) 2000-09-20
EE04837B1 (et) 2007-06-15
PL196889B1 (pl) 2008-02-29
RS49905B (sr) 2008-08-07
TNSN98222A1 (fr) 2005-03-15
AP1260A (en) 2004-03-16
CO4980875A1 (es) 2000-11-27
BR9813531A (pt) 2000-10-10
BG104494A (en) 2001-01-31
NZ504614A (en) 2002-12-20
EE200000336A (et) 2001-08-15
JP4361679B2 (ja) 2009-11-11
PT1036090E (pt) 2006-06-30
DE69834057T2 (de) 2006-12-14
IL184171A0 (en) 2007-10-31
DZ2670A1 (fr) 2003-03-22
DE69834057D1 (de) 2006-05-18
KR100564872B1 (ko) 2006-03-30
HUP0100263A1 (hu) 2001-08-28
WO1999029716A1 (fr) 1999-06-17
US6677429B1 (en) 2004-01-13
BG65033B1 (bg) 2006-12-29
JP2001525421A (ja) 2001-12-11
IL172412A (en) 2008-11-26
US7160983B2 (en) 2007-01-09
PL341012A1 (en) 2001-03-12
PE130099A1 (es) 1999-12-16
TW446541B (en) 2001-07-21
IL136647A0 (en) 2001-06-14
YU33900A (sh) 2002-08-12
CA2311295A1 (fr) 1999-06-17
AU1565999A (en) 1999-06-28
SK8392000A3 (en) 2001-10-08
AP2003002874A0 (en) 2003-09-30
AP1567A (en) 2006-02-08
CZ301919B6 (cs) 2010-07-28
NO20002959D0 (no) 2000-06-09
DK1036090T3 (da) 2006-07-24
US20040072737A1 (en) 2004-04-15
CZ20002113A3 (cs) 2000-11-15
TR200001655T2 (tr) 2000-11-21
PA8464201A1 (es) 2000-09-29
EP1036090B1 (fr) 2006-03-29
KR20010032924A (ko) 2001-04-25

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Legal Events

Date Code Title Description
VENC Patent expired

Effective date: 20181209