RS49905B - Derivati ehinokandina, postupak za njihovo dobijanje i njihova primena kao antifungicida - Google Patents

Derivati ehinokandina, postupak za njihovo dobijanje i njihova primena kao antifungicida

Info

Publication number
RS49905B
RS49905B YUP-339/00A YU33900A RS49905B RS 49905 B RS49905 B RS 49905B YU 33900 A YU33900 A YU 33900A RS 49905 B RS49905 B RS 49905B
Authority
RS
Serbia
Prior art keywords
radical
formula
hydrogen atom
compounds
carbon atoms
Prior art date
Application number
YUP-339/00A
Other languages
English (en)
Serbian (sr)
Inventor
Olivier COURTIN
Patrick FAUVEAU
Astrid Markus
Dominique MELON MANGUER
Jean-Marc MICHEL
Laurent SCHIO
Original Assignee
Aventis Pharma,
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9715628A external-priority patent/FR2772028B1/fr
Priority claimed from FR9813361A external-priority patent/FR2784993B1/fr
Application filed by Aventis Pharma, filed Critical Aventis Pharma,
Publication of YU33900A publication Critical patent/YU33900A/sh
Publication of RS49905B publication Critical patent/RS49905B/sr

Links

Classifications

    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/18Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Veterinary Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Detergent Compositions (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
YUP-339/00A 1997-12-10 1998-12-09 Derivati ehinokandina, postupak za njihovo dobijanje i njihova primena kao antifungicida RS49905B (sr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9715628A FR2772028B1 (fr) 1997-12-10 1997-12-10 Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme fongicides
FR9813361A FR2784993B1 (fr) 1998-10-26 1998-10-26 Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme fongicides

Publications (2)

Publication Number Publication Date
YU33900A YU33900A (sh) 2002-08-12
RS49905B true RS49905B (sr) 2008-08-07

Family

ID=26233984

Family Applications (1)

Application Number Title Priority Date Filing Date
YUP-339/00A RS49905B (sr) 1997-12-10 1998-12-09 Derivati ehinokandina, postupak za njihovo dobijanje i njihova primena kao antifungicida

Country Status (43)

Country Link
US (3) US6677429B1 (enExample)
EP (1) EP1036090B1 (enExample)
JP (1) JP4361679B2 (enExample)
KR (1) KR100564872B1 (enExample)
CN (1) CN1284084A (enExample)
AP (2) AP1567A (enExample)
AR (1) AR016432A1 (enExample)
AT (1) ATE321772T1 (enExample)
AU (1) AU755033B2 (enExample)
BG (1) BG65033B1 (enExample)
BR (1) BR9813531A (enExample)
CA (1) CA2311295A1 (enExample)
CO (1) CO4980875A1 (enExample)
CU (1) CU22962A3 (enExample)
CY (1) CY1105695T1 (enExample)
CZ (1) CZ301919B6 (enExample)
DE (1) DE69834057T2 (enExample)
DK (1) DK1036090T3 (enExample)
DZ (1) DZ2670A1 (enExample)
EA (1) EA002706B1 (enExample)
EE (1) EE04837B1 (enExample)
ES (1) ES2259462T3 (enExample)
GE (1) GEP20032975B (enExample)
HR (1) HRP20000384B1 (enExample)
HU (1) HUP0100263A3 (enExample)
IL (4) IL136647A0 (enExample)
MA (1) MA26575A1 (enExample)
NO (1) NO327498B1 (enExample)
NZ (1) NZ504614A (enExample)
OA (1) OA11899A (enExample)
PA (1) PA8464201A1 (enExample)
PE (1) PE130099A1 (enExample)
PL (1) PL196889B1 (enExample)
PT (1) PT1036090E (enExample)
RS (1) RS49905B (enExample)
SA (1) SA99191248B1 (enExample)
SK (1) SK286916B6 (enExample)
TN (1) TNSN98222A1 (enExample)
TR (1) TR200001655T2 (enExample)
TW (1) TW446541B (enExample)
UA (1) UA72200C2 (enExample)
UY (1) UY25292A1 (enExample)
WO (1) WO1999029716A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA72200C2 (uk) * 1997-12-10 2005-02-15 Авентіс Фарма С.А. Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція
AU1517900A (en) * 1998-10-28 2000-05-15 Eli Lilly And Company Photochemical process for making 1-deoxy-2-keto derivatives
FR2794746B1 (fr) * 1999-06-09 2002-12-06 Hoechst Marion Roussel Inc Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques
FR2794747B1 (fr) 1999-06-09 2004-04-16 Hoechst Marion Roussel Inc Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques
FR2833596B1 (fr) * 2001-12-14 2005-02-18 Aventis Pharma Sa Procede de preparation de derives d'echinocandine
CN101659693B (zh) * 2008-08-27 2012-11-21 上海医药工业研究院 制备纽莫康定b0的方法
CN101659692B (zh) * 2008-08-27 2012-07-04 上海医药工业研究院 制备棘球康定b的方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2241955A (en) * 1990-03-16 1991-09-18 Merck & Co Inc Cyclohexapeptide compounds
IL105048A (en) * 1992-03-19 2001-06-14 Eli Lilly And Company U S Cyclic peptide antifungal agents and process for preparation thereof
US5516757A (en) * 1994-09-16 1996-05-14 Merck & Co., Inc. Semi-synthetic lipopeptides, compositions containing said lipopeptides, and methods of use
US5516756A (en) * 1994-10-31 1996-05-14 Merck & Co., Inc. Aza cyclohexapeptide compounds
DE69615535T2 (de) * 1995-01-26 2002-05-02 Merck & Co., Inc. Neue fungizide cyclohexapeptide
US5646111A (en) * 1995-04-07 1997-07-08 Eli Lilly And Company Cyclic peptide antifungal Agents
UA72200C2 (uk) * 1997-12-10 2005-02-15 Авентіс Фарма С.А. Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція
FR2794747B1 (fr) * 1999-06-09 2004-04-16 Hoechst Marion Roussel Inc Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques

Also Published As

Publication number Publication date
AR016432A1 (es) 2001-07-04
CY1105695T1 (el) 2010-12-22
EA002706B1 (ru) 2002-08-29
SK286916B6 (sk) 2009-07-06
AP1567A (en) 2006-02-08
TR200001655T2 (tr) 2000-11-21
US6677429B1 (en) 2004-01-13
NO20002959D0 (no) 2000-06-09
HRP20000384A2 (en) 2000-10-31
IL172412A (en) 2008-11-26
BG65033B1 (bg) 2006-12-29
EP1036090A1 (fr) 2000-09-20
NO20002959L (no) 2000-08-09
DZ2670A1 (fr) 2003-03-22
ATE321772T1 (de) 2006-04-15
SA99191248B1 (ar) 2006-08-12
AP2003002874A0 (en) 2003-09-30
IL136647A0 (en) 2001-06-14
EA200000625A1 (ru) 2000-12-25
CZ301919B6 (cs) 2010-07-28
WO1999029716A1 (fr) 1999-06-17
MA26575A1 (fr) 2004-12-20
GEP20032975B (en) 2003-05-27
BG104494A (en) 2001-01-31
UA72200C2 (uk) 2005-02-15
CA2311295A1 (fr) 1999-06-17
CU22962A3 (es) 2004-06-21
KR20010032924A (ko) 2001-04-25
OA11899A (fr) 2006-04-10
CN1284084A (zh) 2001-02-14
HRP20000384B1 (en) 2010-02-28
TNSN98222A1 (fr) 2005-03-15
SK8392000A3 (en) 2001-10-08
IL184171A0 (en) 2007-10-31
JP4361679B2 (ja) 2009-11-11
NO327498B1 (no) 2009-07-20
AU755033B2 (en) 2002-11-28
BR9813531A (pt) 2000-10-10
ES2259462T3 (es) 2006-10-01
EE200000336A (et) 2001-08-15
US20050267019A1 (en) 2005-12-01
US7160983B2 (en) 2007-01-09
JP2001525421A (ja) 2001-12-11
PA8464201A1 (es) 2000-09-29
AU1565999A (en) 1999-06-28
CZ20002113A3 (cs) 2000-11-15
PT1036090E (pt) 2006-06-30
US7285619B2 (en) 2007-10-23
EP1036090B1 (fr) 2006-03-29
PL341012A1 (en) 2001-03-12
HUP0100263A1 (hu) 2001-08-28
CO4980875A1 (es) 2000-11-27
DE69834057D1 (de) 2006-05-18
AP2000001826A0 (en) 2000-06-30
PE130099A1 (es) 1999-12-16
US20040072737A1 (en) 2004-04-15
NZ504614A (en) 2002-12-20
IL136647A (en) 2007-06-03
KR100564872B1 (ko) 2006-03-30
AP1260A (en) 2004-03-16
PL196889B1 (pl) 2008-02-29
YU33900A (sh) 2002-08-12
DK1036090T3 (da) 2006-07-24
TW446541B (en) 2001-07-21
UY25292A1 (es) 2000-12-29
HUP0100263A3 (en) 2002-11-28
DE69834057T2 (de) 2006-12-14
EE04837B1 (et) 2007-06-15

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