AP813A - Urea derivatives as inhibitors of IMPDH enzyme. - Google Patents
Urea derivatives as inhibitors of IMPDH enzyme. Download PDFInfo
- Publication number
- AP813A AP813A APAP/P/1997/000973A AP9700973A AP813A AP 813 A AP813 A AP 813A AP 9700973 A AP9700973 A AP 9700973A AP 813 A AP813 A AP 813A
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
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- C—CHEMISTRY; METALLURGY
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/28—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C275/42—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by carboxyl groups
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/636,361 US5807876A (en) | 1996-04-23 | 1996-04-23 | Inhibitors of IMPDH enzyme |
| US08/801,780 US6344465B1 (en) | 1996-04-23 | 1997-02-14 | Inhibitors of IMPDH enzyme |
| US08/832,165 US6054472A (en) | 1996-04-23 | 1997-04-02 | Inhibitors of IMPDH enzyme |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AP9700973A0 AP9700973A0 (en) | 1997-07-31 |
| AP813A true AP813A (en) | 2000-02-28 |
Family
ID=27417590
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| APAP/P/1997/000973A AP813A (en) | 1996-04-23 | 1997-04-23 | Urea derivatives as inhibitors of IMPDH enzyme. |
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| EP (1) | EP0902782A1 (show.php) |
| CN (2) | CN1515248A (show.php) |
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| BR (1) | BR9708735A (show.php) |
| CA (1) | CA2252465C (show.php) |
| CZ (1) | CZ298463B6 (show.php) |
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| HU (1) | HUP0004421A3 (show.php) |
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| US5380879A (en) * | 1994-02-18 | 1995-01-10 | Syntex (U.S.A.) Inc. | Derivatives of mycophenolic acid |
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| DE2928485A1 (de) * | 1979-07-14 | 1981-01-29 | Bayer Ag | Verwendung von harnstoffderivaten als arzneimittel bei der behandlung von fettstoffwechselstoerungen |
| US5283257A (en) | 1992-07-10 | 1994-02-01 | The Board Of Trustees Of The Leland Stanford Junior University | Method of treating hyperproliferative vascular disease |
| WO1994012184A1 (en) | 1992-11-24 | 1994-06-09 | Syntex (U.S.A.) Inc. | Use of mycophenolic acid, mycophenolate mofetil or derivate thereof to inhibit stenosis |
| US5444072A (en) | 1994-02-18 | 1995-08-22 | Syntex (U.S.A.) Inc. | 6-substituted mycophenolic acid and derivatives |
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1997
- 1997-04-21 HU HU0004421A patent/HUP0004421A3/hu not_active Application Discontinuation
- 1997-04-21 TR TR1998/02136T patent/TR199802136T2/xx unknown
- 1997-04-21 EP EP97918759A patent/EP0902782A1/en not_active Withdrawn
- 1997-04-21 PL PL329639A patent/PL192628B1/pl not_active IP Right Cessation
- 1997-04-21 CN CNA031002366A patent/CN1515248A/zh active Pending
- 1997-04-21 EA EA199800943A patent/EA004771B1/ru not_active IP Right Cessation
- 1997-04-21 AU AU26785/97A patent/AU723730B2/en not_active Ceased
- 1997-04-21 CA CA002252465A patent/CA2252465C/en not_active Expired - Fee Related
- 1997-04-21 WO PCT/US1997/006623 patent/WO1997040028A1/en not_active Ceased
- 1997-04-21 BR BR9708735A patent/BR9708735A/pt not_active IP Right Cessation
- 1997-04-21 CZ CZ0338098A patent/CZ298463B6/cs not_active IP Right Cessation
- 1997-04-21 NZ NZ332405A patent/NZ332405A/en not_active IP Right Cessation
- 1997-04-21 CN CN97194856A patent/CN1116288C/zh not_active Expired - Fee Related
- 1997-04-21 SK SK1461-98A patent/SK286662B6/sk not_active IP Right Cessation
- 1997-04-21 IL IL12667497A patent/IL126674A/xx not_active IP Right Cessation
- 1997-04-22 IN IN702CA1997 patent/IN190508B/en unknown
- 1997-04-23 ID IDP971349A patent/ID16664A/id unknown
- 1997-04-23 AP APAP/P/1997/000973A patent/AP813A/en active
-
1998
- 1998-10-21 OA OA9800199A patent/OA10902A/en unknown
- 1998-10-22 NO NO19984917A patent/NO312963B1/no not_active IP Right Cessation
- 1998-11-23 BG BG102945A patent/BG64507B1/bg unknown
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2000
- 2000-04-24 US US09/556,253 patent/US6541496B1/en not_active Expired - Fee Related
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2003
- 2003-01-23 US US10/351,731 patent/US6967214B2/en not_active Expired - Fee Related
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2005
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5380879A (en) * | 1994-02-18 | 1995-01-10 | Syntex (U.S.A.) Inc. | Derivatives of mycophenolic acid |
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