UY36272A - Difluoropirrolidinas como moduladores de los receptores de orexinas - Google Patents

Difluoropirrolidinas como moduladores de los receptores de orexinas

Info

Publication number
UY36272A
UY36272A UY0001036272A UY36272A UY36272A UY 36272 A UY36272 A UY 36272A UY 0001036272 A UY0001036272 A UY 0001036272A UY 36272 A UY36272 A UY 36272A UY 36272 A UY36272 A UY 36272A
Authority
UY
Uruguay
Prior art keywords
disorder
difluoropirrolidins
modulators
orexin receptors
methods
Prior art date
Application number
UY0001036272A
Other languages
English (en)
Inventor
Kamenecka Theodore
He Yuanjun
Original Assignee
Eolas Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eolas Therapeutics Inc filed Critical Eolas Therapeutics Inc
Publication of UY36272A publication Critical patent/UY36272A/es

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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Psychology (AREA)
  • Anesthesiology (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Nutrition Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Reproductive Health (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)

Abstract

La presente especificación se refiere a ciertos compuestos de difluoropirrolidina, composiciones farmacéuticas que los contienen, y métodos para su utilización, incluyendo métodos para tratar adicción a una sustancia, trastorno de pánico, ansiedad, trastorno de estrés post-traumático, dolor, depresión, trastorno afectivo estacional, un trastorno de la alimentación, o hipertensión.
UY0001036272A 2014-08-13 2015-08-13 Difluoropirrolidinas como moduladores de los receptores de orexinas UY36272A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201462037024P 2014-08-13 2014-08-13

Publications (1)

Publication Number Publication Date
UY36272A true UY36272A (es) 2016-02-29

Family

ID=55304607

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001036272A UY36272A (es) 2014-08-13 2015-08-13 Difluoropirrolidinas como moduladores de los receptores de orexinas

Country Status (8)

Country Link
US (1) US10221170B2 (es)
EP (1) EP3180332B1 (es)
JP (1) JP6663909B2 (es)
AR (1) AR101558A1 (es)
ES (1) ES2901418T3 (es)
TW (1) TW201613902A (es)
UY (1) UY36272A (es)
WO (1) WO2016025669A1 (es)

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