SK286446B6 - Amidové deriváty, spôsob ich prípravy, farmaceutický prostriedok, ktorý ich obsahuje, a ich použitie - Google Patents

Amidové deriváty, spôsob ich prípravy, farmaceutický prostriedok, ktorý ich obsahuje, a ich použitie Download PDF

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SK286446B6
SK286446B6 SK172-2001A SK1722001A SK286446B6 SK 286446 B6 SK286446 B6 SK 286446B6 SK 1722001 A SK1722001 A SK 1722001A SK 286446 B6 SK286446 B6 SK 286446B6
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Slovakia
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carbon atoms
alkyl
moiety
alkyl moiety
alkoxy
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SK172-2001A
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Slovak (sk)
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SK1722001A3 (en
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Dearg Sutherland Brown
George Robert Brown
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Astrazeneca Ab
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    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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    • C07C237/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having nitrogen atoms of amino groups bound to the carbon skeleton of the acid part, further acylated
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    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
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    • C07D223/06—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Quinoline Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
SK172-2001A 1998-08-04 1999-07-29 Amidové deriváty, spôsob ich prípravy, farmaceutický prostriedok, ktorý ich obsahuje, a ich použitie SK286446B6 (sk)

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GBGB9816837.0A GB9816837D0 (en) 1998-08-04 1998-08-04 Amide derivatives
PCT/GB1999/002494 WO2000007980A1 (en) 1998-08-04 1999-07-29 Amide derivatives which are useful as cytokine inhibitors

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CZ2001384A3 (cs) 2001-07-11
ATE221047T1 (de) 2002-08-15
PT1102743E (pt) 2002-12-31
HU230343B1 (hu) 2016-02-29
HUP0103366A3 (en) 2002-12-28
PL345809A1 (en) 2002-01-02
NO20010533L (no) 2001-03-30
CA2337770A1 (en) 2000-02-17
ZA200100617B (en) 2002-01-22
DE69902277T2 (de) 2003-06-18
GB9816837D0 (en) 1998-09-30
DE69902277D1 (de) 2002-08-29
AU756292B2 (en) 2003-01-09
AU5179199A (en) 2000-02-28
BRPI9912726B1 (pt) 2011-05-31
CN1330631A (zh) 2002-01-09
NZ509162A (en) 2004-01-30
CN1243724C (zh) 2006-03-01
IL141184A0 (en) 2002-02-10
BRPI9912726A (pt) 2001-05-02
CZ301971B6 (cs) 2010-08-18
US6821965B1 (en) 2004-11-23
HUP0103366A2 (hu) 2002-01-28
JP2002522414A (ja) 2002-07-23
NO20010533D0 (no) 2001-01-31
ES2178895T3 (es) 2003-01-01
DK1102743T3 (da) 2002-09-30
SK1722001A3 (en) 2001-08-06
HK1037608A1 (en) 2002-02-15
NO321017B1 (no) 2006-02-27
KR100628285B1 (ko) 2006-09-27
PL195722B1 (pl) 2007-10-31
CA2337770C (en) 2009-01-20
KR20010099608A (ko) 2001-11-09
IL141184A (en) 2009-11-18
BRPI9912726B8 (pt) 2021-07-06
JP4502509B2 (ja) 2010-07-14
EP1102743B1 (en) 2002-07-24
WO2000007980A1 (en) 2000-02-17
RU2220951C2 (ru) 2004-01-10
EP1102743A1 (en) 2001-05-30

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