SK281403B6 - N4-alkoxykarbonyl-5'-deoxy-5-fluórcytidínové deriváty, spôsob ich výroby, farmaceutické prostriedky s ich obsahom a ich použitie - Google Patents

N4-alkoxykarbonyl-5'-deoxy-5-fluórcytidínové deriváty, spôsob ich výroby, farmaceutické prostriedky s ich obsahom a ich použitie Download PDF

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Publication number
SK281403B6
SK281403B6 SK1444-93A SK144493A SK281403B6 SK 281403 B6 SK281403 B6 SK 281403B6 SK 144493 A SK144493 A SK 144493A SK 281403 B6 SK281403 B6 SK 281403B6
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SK
Slovakia
Prior art keywords
deoxy
fluorocytidine
fluoro
cytidine
acetyl
Prior art date
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SK1444-93A
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English (en)
Slovak (sk)
Other versions
SK144493A3 (en
Inventor
Motohiro Arasaki
Hideo Ishitsuka
Isami Kuruma
Masanori Miwa
Chikako Murasaki
Nobuo Shimma
Isao Umeda
Original Assignee
F. Hoffmann-La Roche Ag
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8210304&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK281403(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by F. Hoffmann-La Roche Ag filed Critical F. Hoffmann-La Roche Ag
Publication of SK144493A3 publication Critical patent/SK144493A3/sk
Publication of SK281403B6 publication Critical patent/SK281403B6/sk

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
SK1444-93A 1992-12-18 1993-12-17 N4-alkoxykarbonyl-5'-deoxy-5-fluórcytidínové deriváty, spôsob ich výroby, farmaceutické prostriedky s ich obsahom a ich použitie SK281403B6 (sk)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP92121538 1992-12-18

Publications (2)

Publication Number Publication Date
SK144493A3 SK144493A3 (en) 1994-10-05
SK281403B6 true SK281403B6 (sk) 2001-03-12

Family

ID=8210304

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1444-93A SK281403B6 (sk) 1992-12-18 1993-12-17 N4-alkoxykarbonyl-5'-deoxy-5-fluórcytidínové deriváty, spôsob ich výroby, farmaceutické prostriedky s ich obsahom a ich použitie

Country Status (41)

Country Link
US (1) US5472949A (lv)
EP (1) EP0602454B1 (lv)
JP (1) JP2501297B2 (lv)
KR (1) KR100347218B1 (lv)
CN (1) CN1035617C (lv)
AT (1) ATE137244T1 (lv)
AU (1) AU671491B2 (lv)
BG (1) BG61485B1 (lv)
BR (1) BR9305089A (lv)
CA (1) CA2103324C (lv)
CZ (1) CZ284788B6 (lv)
DE (1) DE69302360T2 (lv)
DK (1) DK0602454T3 (lv)
EE (1) EE03086B1 (lv)
ES (1) ES2086856T3 (lv)
FI (1) FI112365B (lv)
GE (1) GEP20074251B (lv)
GR (1) GR3020286T3 (lv)
HK (1) HK1005875A1 (lv)
HR (1) HRP931430B1 (lv)
HU (2) HU218291B (lv)
IL (1) IL108000A0 (lv)
IS (1) IS4108A (lv)
LT (1) LT3115B (lv)
LV (1) LV10625B (lv)
MY (1) MY109282A (lv)
NO (1) NO300066B1 (lv)
NZ (1) NZ250414A (lv)
PH (1) PH30168A (lv)
PL (1) PL174100B1 (lv)
RO (1) RO112619B1 (lv)
RU (2) RU2458932C2 (lv)
SA (1) SA93140409B1 (lv)
SI (1) SI9300648B (lv)
SK (1) SK281403B6 (lv)
SV (1) SV1993000080A (lv)
TW (1) TW372239B (lv)
UA (1) UA39158C2 (lv)
UY (1) UY23697A1 (lv)
YU (1) YU49411B (lv)
ZA (1) ZA939293B (lv)

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Publication number Publication date
HUT65757A (en) 1994-07-28
ATE137244T1 (de) 1996-05-15
HRP931430A2 (en) 1998-06-30
CA2103324C (en) 1997-12-23
PH30168A (en) 1997-01-21
CN1094056A (zh) 1994-10-26
YU49411B (sh) 2006-01-16
NO300066B1 (no) 1997-04-01
LV10625B (en) 1996-04-20
IS4108A (is) 1994-06-19
NZ250414A (en) 1995-12-21
UY23697A1 (es) 1994-06-08
CA2103324A1 (en) 1994-06-19
ES2086856T3 (es) 1996-07-01
SI9300648A (en) 1994-09-30
CZ284788B6 (cs) 1999-03-17
RU2493162C1 (ru) 2013-09-20
FI935616A0 (fi) 1993-12-14
GEP20074251B (en) 2007-12-10
PL301541A1 (en) 1994-06-27
IL108000A0 (en) 1994-04-12
BG98304A (bg) 1994-01-03
NO934671L (no) 1994-06-20
UA39158C2 (uk) 2001-06-15
HK1005875A1 (en) 1999-01-29
HU211965A9 (en) 1996-01-29
RO112619B1 (ro) 1997-11-28
US5472949A (en) 1995-12-05
SA93140409B1 (ar) 2004-07-24
CN1035617C (zh) 1997-08-13
DK0602454T3 (da) 1996-07-29
RU2458932C2 (ru) 2012-08-20
TW372239B (en) 1999-10-21
JP2501297B2 (ja) 1996-05-29
KR100347218B1 (ko) 2003-01-24
HU9303525D0 (en) 1994-04-28
CZ273193A3 (en) 1994-07-13
NO934671D0 (no) 1993-12-17
SV1993000080A (es) 1996-01-26
EP0602454B1 (en) 1996-04-24
FI935616A (fi) 1994-06-19
JPH06211891A (ja) 1994-08-02
LT3115B (en) 1994-12-27
GR3020286T3 (en) 1996-09-30
ZA939293B (en) 1994-06-18
BG61485B1 (bg) 1997-09-30
LTIP1627A (en) 1994-07-15
FI112365B (fi) 2003-11-28
SI9300648B (sl) 2000-06-30
EE03086B1 (et) 1998-04-15
SK144493A3 (en) 1994-10-05
DE69302360T2 (de) 1996-10-31
LV10625A (lv) 1995-04-20
PL174100B1 (pl) 1998-06-30
BR9305089A (pt) 1994-07-05
HU218291B (en) 2000-07-28
DE69302360D1 (de) 1996-05-30
KR940014428A (ko) 1994-07-18
YU77993A (sh) 1996-10-18
MY109282A (en) 1996-12-31
AU5069093A (en) 1994-06-30
EP0602454A1 (en) 1994-06-22
RU2135511C1 (ru) 1999-08-27
AU671491B2 (en) 1996-08-29
HRP931430B1 (en) 1999-08-31

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Expiry date: 20131217