SG11201908569QA - Substituted dihydroindene-4-carboxamides and analogs thereof, and methods using same - Google Patents
Substituted dihydroindene-4-carboxamides and analogs thereof, and methods using sameInfo
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- SG11201908569QA SG11201908569QA SG11201908569QA SG11201908569QA SG 11201908569Q A SG11201908569Q A SG 11201908569QA SG 11201908569Q A SG11201908569Q A SG 11201908569QA SG 11201908569Q A SG11201908569Q A SG 11201908569QA
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- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/24—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a ring other than a six-membered aromatic ring
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- A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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- A61K31/27—Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
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- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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US11267825B2 (en) | 2017-11-02 | 2022-03-08 | Aicuris Gmbh & Co. Kg | Highly active amino-thiazole substituted indole-2-carboxamides active against the hepatitis B virus (HBV) |
WO2020046941A1 (en) * | 2018-08-28 | 2020-03-05 | Arbutus Biopharma Corporation | Crystalline forms of substituted dihydroindene-4-carboxamide compounds and methods of preparing and using same |
UY38436A (es) | 2018-11-02 | 2020-05-29 | Aicuris Gmbh & Co Kg | Nuevas 6,7-dihidro-4h-pirazolo[1,5-a] pirazinindol-2-carboxamidas activas contra el virus de la hepatitis b (vhb) |
AR116946A1 (es) | 2018-11-02 | 2021-06-30 | Aicuris Gmbh & Co Kg | Derivados de urea 6,7-dihidro-4h-pirazolo[4,3-c]piridinas activas contra el virus de la hepatitis b (vhb) |
AR117189A1 (es) | 2018-11-02 | 2021-07-21 | Aicuris Gmbh & Co Kg | Derivados de 6,7-dihidro-4h-pirazolo[1,5-a]pirazin indol-2-carboxamidas activos contra el virus de la hepatitis b (vhb) |
WO2020089460A1 (en) | 2018-11-02 | 2020-05-07 | Aicuris Gmbh & Co. Kg | Novel urea 6,7-dihydro-4h-thiazolo[5,4-c]pyridines active against the hepatitis b virus (hbv) |
UY38435A (es) | 2018-11-02 | 2020-05-29 | Aicuris Gmbh & Co Kg | Nuevas urea 6,7-dihidro-4h-pirazol[1,5-a] pirazinas activas contra el virus de la hepatitis b (vhb) |
AR117188A1 (es) | 2018-11-02 | 2021-07-21 | Aicuris Gmbh & Co Kg | Derivados de urea 6,7-dihidro-4h-pirazolo[1,5-a]pirazinas activas contra el virus de la hepatitis b (vhb) |
US20220227789A1 (en) | 2019-04-30 | 2022-07-21 | Aicuris Gmbh & Co. Kg | Novel indolizine-2-carboxamides active against the hepatitis b virus (hbv) |
SG11202111493WA (en) | 2019-04-30 | 2021-11-29 | Aicuris Gmbh & Co Kg | Novel oxalyl piperazines active against the hepatitis b virus (hbv) |
JP2022531199A (ja) | 2019-04-30 | 2022-07-06 | アイクリス ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディトゲゼルシャフト | B型肝炎ウイルス(hbv)に対し活性な新規のフェニル及びピリジル尿素 |
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-
2018
- 2018-03-20 CA CA3056886A patent/CA3056886A1/en not_active Abandoned
- 2018-03-20 SG SG11201908569Q patent/SG11201908569QA/en unknown
- 2018-03-20 EP EP18771245.0A patent/EP3601216B1/de active Active
- 2018-03-20 US US16/495,794 patent/US11098010B2/en active Active
- 2018-03-20 MA MA049014A patent/MA49014A/fr unknown
- 2018-03-20 WO PCT/IB2018/000387 patent/WO2018172852A1/en unknown
- 2018-03-20 AU AU2018238138A patent/AU2018238138A1/en not_active Abandoned
- 2018-03-21 TW TW107109698A patent/TW201838966A/zh unknown
Also Published As
Publication number | Publication date |
---|---|
AU2018238138A1 (en) | 2019-10-17 |
EP3601216B1 (de) | 2023-10-25 |
US11098010B2 (en) | 2021-08-24 |
TW201838966A (zh) | 2018-11-01 |
US20200024226A1 (en) | 2020-01-23 |
CA3056886A1 (en) | 2018-09-27 |
MA49014A (fr) | 2020-02-05 |
EP3601216A4 (de) | 2021-01-06 |
WO2018172852A1 (en) | 2018-09-27 |
EP3601216A1 (de) | 2020-02-05 |
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