PT1631295E - Uso de compostos heterocíclicos condensados como inibidores de scce para o tratamento de doenças da pele - Google Patents

Uso de compostos heterocíclicos condensados como inibidores de scce para o tratamento de doenças da pele Download PDF

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Publication number
PT1631295E
PT1631295E PT04736195T PT04736195T PT1631295E PT 1631295 E PT1631295 E PT 1631295E PT 04736195 T PT04736195 T PT 04736195T PT 04736195 T PT04736195 T PT 04736195T PT 1631295 E PT1631295 E PT 1631295E
Authority
PT
Portugal
Prior art keywords
phenyl
thia
oxa
aza
oxazin
Prior art date
Application number
PT04736195T
Other languages
English (en)
Portuguese (pt)
Inventor
Marcel Linschoten
Original Assignee
Arexis Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arexis Ab filed Critical Arexis Ab
Publication of PT1631295E publication Critical patent/PT1631295E/pt

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5365Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/536Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/04Antipruritics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/10Anti-acne agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/12Keratolytics, e.g. wart or anti-corn preparations
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Cosmetics (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PT04736195T 2003-06-06 2004-06-07 Uso de compostos heterocíclicos condensados como inibidores de scce para o tratamento de doenças da pele PT1631295E (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DKPA200300844 2003-06-06
DKPA200300842 2003-06-06
DKPA200300840 2003-06-06
DKPA200300843 2003-06-06

Publications (1)

Publication Number Publication Date
PT1631295E true PT1631295E (pt) 2010-05-24

Family

ID=33514772

Family Applications (1)

Application Number Title Priority Date Filing Date
PT04736195T PT1631295E (pt) 2003-06-06 2004-06-07 Uso de compostos heterocíclicos condensados como inibidores de scce para o tratamento de doenças da pele

Country Status (17)

Country Link
US (1) US7872052B2 (https=)
EP (1) EP1631295B1 (https=)
JP (1) JP5044214B2 (https=)
KR (2) KR101205257B1 (https=)
CN (1) CN101152185B (https=)
AT (1) ATE459359T1 (https=)
CA (1) CA2525383C (https=)
CY (1) CY1110084T1 (https=)
DE (1) DE602004025803D1 (https=)
DK (1) DK1631295T3 (https=)
ES (1) ES2341545T3 (https=)
NO (1) NO20060091L (https=)
NZ (1) NZ543636A (https=)
PL (1) PL1631295T3 (https=)
PT (1) PT1631295E (https=)
SI (1) SI1631295T1 (https=)
WO (1) WO2004108139A2 (https=)

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Also Published As

Publication number Publication date
WO2004108139A2 (en) 2004-12-16
WO2004108139A8 (en) 2005-04-28
HK1091731A1 (zh) 2007-01-26
WO2004108139A3 (en) 2005-03-10
DK1631295T3 (da) 2010-06-21
CN101152185A (zh) 2008-04-02
CY1110084T1 (el) 2015-01-14
ES2341545T3 (es) 2010-06-22
JP2006526581A (ja) 2006-11-24
AU2004244704A1 (en) 2004-12-16
CA2525383A1 (en) 2004-12-16
CA2525383C (en) 2012-03-06
KR20110120960A (ko) 2011-11-04
CN101152185B (zh) 2010-12-08
EP1631295B1 (en) 2010-03-03
KR101099409B1 (ko) 2011-12-27
SI1631295T1 (sl) 2010-06-30
EP1631295A2 (en) 2006-03-08
JP5044214B2 (ja) 2012-10-10
PL1631295T3 (pl) 2010-09-30
NZ543636A (en) 2009-07-31
ATE459359T1 (de) 2010-03-15
KR20060008331A (ko) 2006-01-26
US20060258651A1 (en) 2006-11-16
KR101205257B1 (ko) 2012-11-27
DE602004025803D1 (de) 2010-04-15
NO20060091L (no) 2006-03-06
US7872052B2 (en) 2011-01-18
HK1120209A1 (en) 2009-03-27

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