GB1153994A - Hydroxyphenyl Anthranilic Acid Derivatives Capable of Absorbing 'Ultra-Violet Light and Compositions containing them - Google Patents

Hydroxyphenyl Anthranilic Acid Derivatives Capable of Absorbing 'Ultra-Violet Light and Compositions containing them

Info

Publication number
GB1153994A
GB1153994A GB898966A GB898966A GB1153994A GB 1153994 A GB1153994 A GB 1153994A GB 898966 A GB898966 A GB 898966A GB 898966 A GB898966 A GB 898966A GB 1153994 A GB1153994 A GB 1153994A
Authority
GB
United Kingdom
Prior art keywords
group
ultra
hydrogen
violet light
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB898966A
Inventor
Maurice Ward Gittos
John William James
Leslie Frederick Wiggins
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aspro Nicholas Ltd
Original Assignee
Aspro Nicholas Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aspro Nicholas Ltd filed Critical Aspro Nicholas Ltd
Priority to GB898966A priority Critical patent/GB1153994A/en
Priority to BE684403D priority patent/BE684403A/xx
Priority to FR70260A priority patent/FR1513274A/en
Publication of GB1153994A publication Critical patent/GB1153994A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
    • C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D265/20—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in position 4
    • C07D265/22—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/40—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing nitrogen
    • A61K8/41—Amines
    • A61K8/411—Aromatic amines, i.e. where the amino group is directly linked to the aromatic nucleus
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q17/00—Barrier preparations; Preparations brought into direct contact with the skin for affording protection against external influences, e.g. sunlight, X-rays or other harmful rays, corrosive materials, bacteria or insect stings
    • A61Q17/04—Topical preparations for affording protection against sunlight or other radiation; Topical sun tanning preparations
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08K—Use of inorganic or non-macromolecular organic substances as compounding ingredients
    • C08K5/00—Use of organic ingredients
    • C08K5/16—Nitrogen-containing compounds
    • C08K5/20—Carboxylic acid amides
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08K—Use of inorganic or non-macromolecular organic substances as compounding ingredients
    • C08K5/00—Use of organic ingredients
    • C08K5/16—Nitrogen-containing compounds
    • C08K5/34—Heterocyclic compounds having nitrogen in the ring
    • C08K5/3412—Heterocyclic compounds having nitrogen in the ring having one nitrogen atom in the ring
    • C08K5/3432—Six-membered rings
    • C08K5/3437—Six-membered rings condensed with carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08K—Use of inorganic or non-macromolecular organic substances as compounding ingredients
    • C08K5/00—Use of organic ingredients
    • C08K5/16—Nitrogen-containing compounds
    • C08K5/34—Heterocyclic compounds having nitrogen in the ring
    • C08K5/35—Heterocyclic compounds having nitrogen in the ring having also oxygen in the ring

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Polymers & Plastics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Birds (AREA)
  • Dermatology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

1,153,994. U/V light-absorbing preparations. ASPRO-NICHOLAS Ltd. 15 July, 1966 [21 July, 1965; 1 March, 1966], Nos. 30924/65 and 8989/66. Heading A5B [Also in Divisions C2 and C3] Compounds of formula I or II in which X is an oxygen atom or an imino group; R and R 1 , which may be the same or different, are each hydrogen, a C 1 - C 12 alkyl or alkoxy group, a halogen atom, a hydroxy group, a nitro group, a sulphonic acid group, or an amino group of formula in which R 4 is hydrogen or a C 1 - C 4 alkyl group and R 5 is hydrogen, a C 1 - C 4 alkyl group, a 2 - hydroxy benzoyl group or a 2,4 - dichlorotriazine group linked in the 6 - position, R 2 is halogen, C 1 - C 12 alkyl or alkoxy, a sulphonic acid radical, a nitro group or carboxyl; R 3 is hydrogen, a C 1 - C 12 alkyl group optionally substituted by a sulphonic acid radical or an amino group and n is an integer from 0 to 4 (R 2 being the same or different when n is 2, 3 or 4), are used as sun-screening agents in cosmetics and to prevent degradation of perfumes due to the action of ultra violet light. They may be incorporated in a liquid or semi-liquid carrier to give a dermatologically acceptable composition to give a composition which diminishes burning of the skin caused by ultra-violet light. Examples are given of the preparation of creams containing (a) n - hexyl N - (2 - hydroxy - benzoyl) anthranilate (Ex. 23) and (b) isobutyl N - (2 - hydroxybenzoyl) antbranilate (Ex. 24) which protect the skin from ultra-violet light and the protection of a perfume for deterioration of colour by the addition of ethyl N - (2 - hydroxybenzoyl) anthraniliate (Ex. 25).
GB898966A 1965-07-21 1965-07-21 Hydroxyphenyl Anthranilic Acid Derivatives Capable of Absorbing 'Ultra-Violet Light and Compositions containing them Expired GB1153994A (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
GB898966A GB1153994A (en) 1965-07-21 1965-07-21 Hydroxyphenyl Anthranilic Acid Derivatives Capable of Absorbing 'Ultra-Violet Light and Compositions containing them
BE684403D BE684403A (en) 1965-07-21 1966-07-20
FR70260A FR1513274A (en) 1965-07-21 1966-07-21 Compounds capable of absorbing ultraviolet light and compositions containing them

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB898966A GB1153994A (en) 1965-07-21 1965-07-21 Hydroxyphenyl Anthranilic Acid Derivatives Capable of Absorbing 'Ultra-Violet Light and Compositions containing them
GB3092465 1965-07-21

Publications (1)

Publication Number Publication Date
GB1153994A true GB1153994A (en) 1969-06-04

Family

ID=26242558

Family Applications (1)

Application Number Title Priority Date Filing Date
GB898966A Expired GB1153994A (en) 1965-07-21 1965-07-21 Hydroxyphenyl Anthranilic Acid Derivatives Capable of Absorbing 'Ultra-Violet Light and Compositions containing them

Country Status (3)

Country Link
BE (1) BE684403A (en)
FR (1) FR1513274A (en)
GB (1) GB1153994A (en)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0032242B1 (en) * 1980-01-05 1983-12-14 BASF Aktiengesellschaft 4h-3,1-benzoxazine derivatives, process for their preparation and their use in inhibiting the growth of unwanted plants
US5560852A (en) * 1994-03-26 1996-10-01 Sandoz Ltd. Use of 4H-3,1-benzoxazin-4-one compounds to improve the light fastness of textile materials
WO2004108139A3 (en) * 2003-06-06 2005-03-10 Arexis Ab Use of fused heterocyclic compounds as scce inhibitors for the treatment of skin conditions or cancer
WO2005049604A2 (en) * 2003-09-30 2005-06-02 Eli Lilly And Company Antithrombotic aromatic ethers
CN100518740C (en) * 2003-06-06 2009-07-29 阿里克斯股份公司 Use of heterocyclic compounds as SCCE inhibitors
WO2015112081A1 (en) * 2014-01-23 2015-07-30 Sixera Pharma Ab Benzoxazinone derivatives for treatment of skin diseases

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3938526A1 (en) * 1989-11-21 1991-05-23 Basf Ag USE OF HETEROCYCLIC COMPOUNDS AS BLEACH ACTIVATORS OR OPTICAL BRIGHTENERS IN DETERGENT AND CLEANING AGENTS
CA2545023A1 (en) * 2003-11-25 2005-06-09 Novo Nordisk A/S Novel salicylic anilides

Cited By (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0032242B1 (en) * 1980-01-05 1983-12-14 BASF Aktiengesellschaft 4h-3,1-benzoxazine derivatives, process for their preparation and their use in inhibiting the growth of unwanted plants
US5560852A (en) * 1994-03-26 1996-10-01 Sandoz Ltd. Use of 4H-3,1-benzoxazin-4-one compounds to improve the light fastness of textile materials
WO2004108139A3 (en) * 2003-06-06 2005-03-10 Arexis Ab Use of fused heterocyclic compounds as scce inhibitors for the treatment of skin conditions or cancer
CN100518740C (en) * 2003-06-06 2009-07-29 阿里克斯股份公司 Use of heterocyclic compounds as SCCE inhibitors
WO2005049604A2 (en) * 2003-09-30 2005-06-02 Eli Lilly And Company Antithrombotic aromatic ethers
WO2005049604A3 (en) * 2003-09-30 2005-09-15 Lilly Co Eli Antithrombotic aromatic ethers
US7511066B2 (en) 2003-09-30 2009-03-31 Eli Lilly And Company Antithrombotic aromatic ethers
WO2015112081A1 (en) * 2014-01-23 2015-07-30 Sixera Pharma Ab Benzoxazinone derivatives for treatment of skin diseases
US9695194B2 (en) 2014-01-23 2017-07-04 Sixera Pharma Ab Benzoxazinone derivatives for treatment of skin diseases
US10072024B2 (en) 2014-01-23 2018-09-11 Sixera Pharma Ab Benzoxazinone derivatives for treatment of skin diseases

Also Published As

Publication number Publication date
BE684403A (en) 1967-01-20
FR1513274A (en) 1968-02-16

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