PT1099694E - Processo para a preparacao de um derivado de quinolina e um intermediario para esse fim - Google Patents

Processo para a preparacao de um derivado de quinolina e um intermediario para esse fim

Info

Publication number
PT1099694E
PT1099694E PT99931484T PT99931484T PT1099694E PT 1099694 E PT1099694 E PT 1099694E PT 99931484 T PT99931484 T PT 99931484T PT 99931484 T PT99931484 T PT 99931484T PT 1099694 E PT1099694 E PT 1099694E
Authority
PT
Portugal
Prior art keywords
preparation
intermediary
quinoline derivative
quinoline
derivative
Prior art date
Application number
PT99931484T
Other languages
English (en)
Inventor
Mikio Suzuki
Yoshio Ohara
Yoshinobu Yanagawa
Yasutaka Takada
Original Assignee
Nissan Chemical Ind Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nissan Chemical Ind Ltd filed Critical Nissan Chemical Ind Ltd
Publication of PT1099694E publication Critical patent/PT1099694E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D215/14Radicals substituted by oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
PT99931484T 1998-07-23 1999-07-22 Processo para a preparacao de um derivado de quinolina e um intermediario para esse fim PT1099694E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP20791198 1998-07-23

Publications (1)

Publication Number Publication Date
PT1099694E true PT1099694E (pt) 2005-10-31

Family

ID=16547618

Family Applications (1)

Application Number Title Priority Date Filing Date
PT99931484T PT1099694E (pt) 1998-07-23 1999-07-22 Processo para a preparacao de um derivado de quinolina e um intermediario para esse fim

Country Status (21)

Country Link
US (1) US6335449B1 (pt)
EP (1) EP1099694B1 (pt)
JP (1) JP4281248B2 (pt)
KR (1) KR100529201B1 (pt)
CN (1) CN1107670C (pt)
AT (1) ATE302190T1 (pt)
AU (1) AU746722C (pt)
CA (1) CA2338334C (pt)
CZ (1) CZ299881B6 (pt)
DE (1) DE69926760T2 (pt)
DK (1) DK1099694T3 (pt)
ES (1) ES2247813T3 (pt)
IL (2) IL140924A0 (pt)
MX (1) MXPA01000890A (pt)
NO (1) NO317787B1 (pt)
NZ (1) NZ509401A (pt)
PT (1) PT1099694E (pt)
RU (1) RU2214402C2 (pt)
SK (1) SK285675B6 (pt)
WO (1) WO2000005213A1 (pt)
ZA (1) ZA200100525B (pt)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1222512C (zh) * 2000-01-24 2005-10-12 日产化学工业株式会社 喹啉基丙烯醛的制备方法
JP4496586B2 (ja) * 2000-01-24 2010-07-07 日産化学工業株式会社 キノリルアクリロニトリルの製造法及びその中間体
JP4496585B2 (ja) * 2000-01-24 2010-07-07 日産化学工業株式会社 キノリルプロペナールの製造方法
JP4496584B2 (ja) * 2000-01-24 2010-07-07 日産化学工業株式会社 キノリルプロペナールの製造法
JP4867071B2 (ja) * 2000-02-21 2012-02-01 日産化学工業株式会社 キノリン誘導体の製造方法
AU2001232342A1 (en) * 2000-02-21 2001-08-27 Kuraray Co. Ltd. Processes for preparing quinoline derivatives and intermediates thereof
CN1230173C (zh) * 2000-10-12 2005-12-07 日产化学工业株式会社 糖尿病合并症预防及治疗剂
US6777552B2 (en) * 2001-08-16 2004-08-17 Teva Pharmaceutical Industries, Ltd. Processes for preparing calcium salt forms of statins
JP2002155056A (ja) * 2000-11-17 2002-05-28 Ube Ind Ltd キノリルアクリロニトリル誘導体の製法
TWI309644B (pt) 2001-02-14 2009-05-11 Nissan Chemical Ind Ltd
JP4590749B2 (ja) * 2001-02-14 2010-12-01 宇部興産株式会社 キノリンカルボキシアルデヒド誘導体の製法
JP5192147B2 (ja) * 2003-02-12 2013-05-08 日産化学工業株式会社 ピタバスタチンカルシウムの結晶質形態
US8455640B2 (en) 2006-05-03 2013-06-04 Msn Laboratories Limited Process for statins and its pharmaceutically acceptable salts thereof
ES2567171T3 (es) 2006-10-09 2016-04-20 Msn Laboratories Private Limited Nuevo procedimiento para la preparación de estatinas y sus sales farmacéuticamente aceptables
US8487105B2 (en) 2009-01-19 2013-07-16 Msn Laboratories Limited Process for preparing pitavastatin, intermediates and pharmaceuctically acceptable salts thereof
US8987444B2 (en) 2010-01-18 2015-03-24 Msn Laboratories Private Limited Process for the preparation of amide intermediates and their use thereof
US20120022102A1 (en) 2010-01-20 2012-01-26 Cadila Healthcare Limited Method for preparation of pitavastatin and its pharmaceutical acceptable salts thereof
JP2013536219A (ja) 2010-08-25 2013-09-19 カディラ・ヘルスケア・リミテッド ピタバスタチンカルシウムおよびその調製方法
CN103508949B (zh) * 2013-10-22 2015-12-09 黄河三角洲京博化工研究院有限公司 一种(e)-3-[2-环丙基-4-(4-氟-苯基)-3-喹啉基]丙烯醛的合成方法
WO2016005919A1 (en) 2014-07-09 2016-01-14 Lupin Limited Polymorphic forms of pitavastatin sodium

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5815836A (ja) * 1981-07-17 1983-01-29 オリンパス光学工業株式会社 内視鏡管路の洗浄装置
US5854259A (en) 1987-08-20 1998-12-29 Nissan Chemical Industries Ltd. Quinoline type mevalonolactones
JP2569746B2 (ja) 1987-08-20 1997-01-08 日産化学工業株式会社 キノリン系メバロノラクトン類
US5185328A (en) 1987-08-20 1993-02-09 Nissan Chemical Industries Ltd. Quinoline type mevalonolactones useful for treating hyperlipidemia, hyperlipoproteinemia or atherosclerosis
DE3905908A1 (de) * 1989-02-25 1990-09-06 Bayer Ag Substituierte chinoline, verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln
JP3528186B2 (ja) 1991-06-24 2004-05-17 日産化学工業株式会社 光学活性キノリンメバロン酸のジアステレオマー塩
JP3130342B2 (ja) 1991-10-04 2001-01-31 日産化学工業株式会社 動脈硬化性血管内膜肥厚抑制薬
CN1136183C (zh) 1994-02-25 2004-01-28 代科化学工业株式会社 光学活性甲羟戊酸内酯类化合物的制造方法

Also Published As

Publication number Publication date
EP1099694A4 (en) 2002-08-14
US6335449B1 (en) 2002-01-01
CA2338334C (en) 2008-07-15
WO2000005213A1 (fr) 2000-02-03
MXPA01000890A (es) 2002-06-04
CA2338334A1 (en) 2000-02-03
AU4799299A (en) 2000-02-14
NZ509401A (en) 2002-08-28
DE69926760T2 (de) 2006-01-19
JP4281248B2 (ja) 2009-06-17
CN1310711A (zh) 2001-08-29
NO20010357L (no) 2001-01-22
ZA200100525B (en) 2001-08-01
AU746722C (en) 2003-03-27
EP1099694B1 (en) 2005-08-17
EP1099694A1 (en) 2001-05-16
NO20010357D0 (no) 2001-01-22
DE69926760D1 (de) 2005-09-22
SK285675B6 (sk) 2007-06-07
SK622001A3 (en) 2001-08-06
NO317787B1 (no) 2004-12-13
CZ200162A3 (en) 2001-06-13
CZ299881B6 (cs) 2008-12-17
IL140924A (en) 2006-06-11
IL140924A0 (en) 2002-02-10
KR20010070987A (ko) 2001-07-28
ATE302190T1 (de) 2005-09-15
AU746722B2 (en) 2002-05-02
DK1099694T3 (da) 2005-09-19
CN1107670C (zh) 2003-05-07
RU2214402C2 (ru) 2003-10-20
ES2247813T3 (es) 2006-03-01
KR100529201B1 (ko) 2005-11-17

Similar Documents

Publication Publication Date Title
PT1099694E (pt) Processo para a preparacao de um derivado de quinolina e um intermediario para esse fim
ATE384857T1 (de) Blechklammer für kipphebel
DK1249281T3 (da) Selvrensende overflade med hydrofob overfladestruktur og fremgangsmåde til fremstilling af denne
ATE255110T1 (de) Fungizide 7-alkyl-triazolopyrimidine
ES8101732A1 (es) Acoplamiento realizado a partir de una plancha de chapa o deun trozo de tubo
DE69920923D1 (de) Anthranilsäurederivate
RU2001105200A (ru) Способ получения производного хинолина и промежуточного соединения
BR9915254A (pt) Processo de preparação da metionina
BR0311577A (pt) Trocador de calor para veìculo motorizado, veìculo motorizado, método para aplicar e para a fabricação de um trocador de calor
ATE390736T1 (de) Elektrische verbindung
AR028571A1 (es) Proceso para preparar compuestos de acido iminodiacético a partir de sustratos de monoetanolamina
BR9912016A (pt) Processo de hidrólise do 2-hidróxi 4-metiltiobutironitrilo com ácido sulfúrico
PT1347984E (pt) Processo para a preparacao de derivados de taxano
NO20014885D0 (no) Fremgangsmåte til fremstilling av en amidforbindelse
HK1027574A1 (en) Process for producing 3-alkenylcephem compounds
DK0957078T3 (da) Fremgangsmåde til fremstilling af shikimisyre og derivater deraf
DE60107044D1 (de) Kontaktstreifen mit gebogenen Projektionen und Herstellungsverfahren
PT924195E (pt) Processo para a preparacao de aminocianacetamida
ATE374840T1 (de) Vorrichtung zum induktiven härten
BR9913401A (pt) Processo para a preparação de 2hidróxi-6-trifluorometilpiridina
DK1206453T3 (da) Fremgangsmåde til fremstilling af 3,5-dichlorpyridin
PT1234817E (pt) Processo para a preparacao de midodrina
BR0113856A (pt) Processo de fixação de pelo menos um inserto de guia entre dois tubos coaxiais
ATE410640T1 (de) Lichtblendenbefestigung für fahrzeugleuchte
EA200301225A1 (ru) Способ получения аморфного циластатин-натрия