PL2854859T3 - Krystaliczne postacie inhibitora kinazy tyrozynowej brutona - Google Patents

Krystaliczne postacie inhibitora kinazy tyrozynowej brutona

Info

Publication number
PL2854859T3
PL2854859T3 PL13799982.7T PL13799982T PL2854859T3 PL 2854859 T3 PL2854859 T3 PL 2854859T3 PL 13799982 T PL13799982 T PL 13799982T PL 2854859 T3 PL2854859 T3 PL 2854859T3
Authority
PL
Poland
Prior art keywords
bruton
tyrosine kinase
kinase inhibitor
crystalline forms
crystalline
Prior art date
Application number
PL13799982.7T
Other languages
English (en)
Inventor
Norbert Purro
Mark Smyth
Erick Goldman
David D. Wirth
Original Assignee
Pharmacyclics Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49712527&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL2854859(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacyclics Llc filed Critical Pharmacyclics Llc
Publication of PL2854859T3 publication Critical patent/PL2854859T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B65—CONVEYING; PACKING; STORING; HANDLING THIN OR FILAMENTARY MATERIAL
    • B65D—CONTAINERS FOR STORAGE OR TRANSPORT OF ARTICLES OR MATERIALS, e.g. BAGS, BARRELS, BOTTLES, BOXES, CANS, CARTONS, CRATES, DRUMS, JARS, TANKS, HOPPERS, FORWARDING CONTAINERS; ACCESSORIES, CLOSURES, OR FITTINGS THEREFOR; PACKAGING ELEMENTS; PACKAGES
    • B65D75/00—Packages comprising articles or materials partially or wholly enclosed in strips, sheets, blanks, tubes or webs of flexible sheet material, e.g. in folded wrappers
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Otolaryngology (AREA)
  • Reproductive Health (AREA)
  • Dermatology (AREA)
  • Composite Materials (AREA)
  • Mechanical Engineering (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Toxicology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Cardiology (AREA)
PL13799982.7T 2012-06-04 2013-06-03 Krystaliczne postacie inhibitora kinazy tyrozynowej brutona PL2854859T3 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261655381P 2012-06-04 2012-06-04
PCT/US2013/043888 WO2013184572A1 (en) 2012-06-04 2013-06-03 Crystalline forms of a bruton's tyrosine kinase inhibitor

Publications (1)

Publication Number Publication Date
PL2854859T3 true PL2854859T3 (pl) 2026-06-22

Family

ID=49712527

Family Applications (1)

Application Number Title Priority Date Filing Date
PL13799982.7T PL2854859T3 (pl) 2012-06-04 2013-06-03 Krystaliczne postacie inhibitora kinazy tyrozynowej brutona

Country Status (41)

Country Link
US (27) US9296753B2 (pl)
EP (2) EP4729054A1 (pl)
JP (10) JP6236071B2 (pl)
KR (8) KR20150015021A (pl)
CN (2) CN110354132A (pl)
AR (2) AR092844A1 (pl)
AU (7) AU2013271918C1 (pl)
BR (1) BR112014030424A8 (pl)
CA (4) CA3015208C (pl)
CL (3) CL2014003306A1 (pl)
CO (1) CO7240408A2 (pl)
CR (1) CR20140558A (pl)
DK (1) DK2854859T3 (pl)
DO (3) DOP2014000274A (pl)
EA (1) EA201492082A1 (pl)
EC (2) ECSP14033163A (pl)
ES (1) ES3069541T3 (pl)
FI (1) FI2854859T3 (pl)
GT (1) GT201400281A (pl)
HK (1) HK1208803A1 (pl)
HR (1) HRP20260603T1 (pl)
IL (4) IL315394A (pl)
JO (2) JO3754B1 (pl)
LT (1) LT2854859T (pl)
MA (2) MA37711A1 (pl)
MX (3) MX348290B (pl)
MY (2) MY194911A (pl)
NZ (4) NZ731932A (pl)
PE (3) PE20241581A1 (pl)
PH (3) PH12021552282A1 (pl)
PL (1) PL2854859T3 (pl)
PT (1) PT2854859T (pl)
RS (1) RS68001B1 (pl)
SG (2) SG10202101389TA (pl)
SI (1) SI2854859T1 (pl)
TN (1) TN2014000492A1 (pl)
TW (3) TWI662963B (pl)
UA (2) UA126959C2 (pl)
UY (2) UY39740A (pl)
WO (1) WO2013184572A1 (pl)
ZA (4) ZA202105175B (pl)

Families Citing this family (137)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2529621B1 (en) 2006-09-22 2016-10-05 Pharmacyclics LLC Inhibitors of bruton's tyrosine kinase
US8809273B2 (en) 2007-03-28 2014-08-19 Pharmacyclics, Inc. Inhibitors of Bruton's tyrosine kinase
CN102159214A (zh) 2008-07-16 2011-08-17 药品循环公司 用于实体肿瘤的治疗的布鲁顿酪氨酸激酶的抑制剂
US8491927B2 (en) * 2009-12-02 2013-07-23 Nimble Epitech, Llc Pharmaceutical composition containing a hypomethylating agent and a histone deacetylase inhibitor
MX380504B (es) 2010-06-03 2025-03-12 Pharmacyclics Llc El uso de inhibidores de la tirosina quinasa de bruton (btk).
BR112013017722A2 (pt) 2011-01-11 2016-07-12 Glaxosmithkline Llc combinação
KR20140048968A (ko) 2011-07-13 2014-04-24 파마시클릭스, 인코포레이티드 브루톤형 티로신 키나제의 억제제
DK2734205T3 (en) 2011-07-21 2018-06-14 Tolero Pharmaceuticals Inc Heterocyclic Protein Kinase Inhibitors
RS57248B1 (sr) 2011-12-11 2018-07-31 Viamet Pharmaceuticals Nc Inc Jedinjenja inhibitori metaloenzima
US8377946B1 (en) 2011-12-30 2013-02-19 Pharmacyclics, Inc. Pyrazolo[3,4-d]pyrimidine and pyrrolo[2,3-d]pyrimidine compounds as kinase inhibitors
MA37711A1 (fr) 2012-06-04 2017-05-31 Pharmacyclics Inc Formes cristallines d'un inhibiteur de tyrosine kinase de bruton
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