UY39740A - Formas cristalinas de un inhibidor de tirosina quinasa de bruton - Google Patents

Formas cristalinas de un inhibidor de tirosina quinasa de bruton

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Publication number
UY39740A
UY39740A UY0001039740A UY39740A UY39740A UY 39740 A UY39740 A UY 39740A UY 0001039740 A UY0001039740 A UY 0001039740A UY 39740 A UY39740 A UY 39740A UY 39740 A UY39740 A UY 39740A
Authority
UY
Uruguay
Prior art keywords
bruton
tyrosine kinase
crystalline forms
inhibitor
kinase inhibitor
Prior art date
Application number
UY0001039740A
Other languages
English (en)
Inventor
Mark Smyth
Erick Goldman
D Wirth David
Norbert Purro
Original Assignee
Pharmacyclics Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49712527&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY39740(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacyclics Llc filed Critical Pharmacyclics Llc
Publication of UY39740A publication Critical patent/UY39740A/es

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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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Abstract

Se describe aquí al inhibidor de tirosina quinasa (Btk) de Bruton 1-((R)-3-(4-amino-3-(4-fenoxifenil)-1H-pirazolo[3,4-d] pirimidin-1-il)piperidin-1-il)prop-2-en-1-ona, incluyendo las formas cristalinas, solvatos y sus sales aceptables en el campo farmacéutico. Se describe también composiciones farmacéuticas que incluyen al inhibidor Btk, así como métodos para usar a dicho inhibidor solo o en combinación con otros agentes terapéuticos, para el tratamiento de enfermedades o condiciones autoinmunes, enfermedades o condiciones heteroinmunes, cáncer, incluyendo linfoma, así como enfermedades o condiciones inflamatorias.
UY0001039740A 2012-06-04 2013-06-04 Formas cristalinas de un inhibidor de tirosina quinasa de bruton UY39740A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261655381P 2012-06-04 2012-06-04
UY0001034848A UY34848A (es) 2012-06-04 2013-06-04 Formas cristalinas de un inhibidor de tirosina quinasa de bruton

Publications (1)

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UY39740A true UY39740A (es) 2022-06-30

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UY0001039740A UY39740A (es) 2012-06-04 2013-06-04 Formas cristalinas de un inhibidor de tirosina quinasa de bruton
UY0001034848A UY34848A (es) 2012-06-04 2013-06-04 Formas cristalinas de un inhibidor de tirosina quinasa de bruton

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US (25) US9540382B2 (es)
EP (1) EP2854859A4 (es)
JP (8) JP6236071B2 (es)
KR (7) KR20190040370A (es)
CN (2) CN104736178A (es)
AR (2) AR092844A1 (es)
AU (6) AU2013271918C1 (es)
BR (1) BR112014030424A8 (es)
CA (4) CA3218491A1 (es)
CL (3) CL2014003306A1 (es)
CO (1) CO7240408A2 (es)
CR (1) CR20140558A (es)
DO (3) DOP2014000274A (es)
EA (1) EA201492082A1 (es)
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GT (1) GT201400281A (es)
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UA (2) UA126959C2 (es)
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EP3311818A3 (en) 2008-07-16 2018-07-18 Pharmacyclics, LLC Inhibitors of bruton's tyrosine kinase for the treatment of solid tumors
US8491927B2 (en) * 2009-12-02 2013-07-23 Nimble Epitech, Llc Pharmaceutical composition containing a hypomethylating agent and a histone deacetylase inhibitor
WO2011153514A2 (en) 2010-06-03 2011-12-08 Pharmacyclics, Inc. The use of inhibitors of bruton's tyrosine kinase (btk)
BR112013017722A2 (pt) 2011-01-11 2016-07-12 Glaxosmithkline Llc combinação
WO2013010136A2 (en) 2011-07-13 2013-01-17 Pharmacyclics, Inc. Inhibitors of bruton's tyrosine kinase
ES2671748T3 (es) 2011-07-21 2018-06-08 Tolero Pharmaceuticals, Inc. Inhibidores heterocíclicos de proteína quinasas
PT2788343T (pt) 2011-12-11 2018-06-01 Viamet Pharmaceuticals Nc Inc Compostos inibidores de metaloenzimas
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US9713617B2 (en) 2017-07-25
CL2014003306A1 (es) 2015-04-17
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