PL1675573T3 - Sterylny preparat do wstrzykiwań arypiprazolu o kontrolowanym uwalnianiu i sposób - Google Patents

Sterylny preparat do wstrzykiwań arypiprazolu o kontrolowanym uwalnianiu i sposób

Info

Publication number
PL1675573T3
PL1675573T3 PL04795514T PL04795514T PL1675573T3 PL 1675573 T3 PL1675573 T3 PL 1675573T3 PL 04795514 T PL04795514 T PL 04795514T PL 04795514 T PL04795514 T PL 04795514T PL 1675573 T3 PL1675573 T3 PL 1675573T3
Authority
PL
Poland
Prior art keywords
controlled release
sterile injectable
aripiprazole formulation
release sterile
injectable aripiprazole
Prior art date
Application number
PL04795514T
Other languages
English (en)
Other versions
PL1675573T5 (pl
PL1675573T4 (pl
Inventor
Janusz W Kostanski
Takakuni Corpo Faburesu B-201 MATSUDA
Manoj Nerurkar
Vijay H Naringrekar
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34549292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL1675573(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of PL1675573T3 publication Critical patent/PL1675573T3/pl
Publication of PL1675573T5 publication Critical patent/PL1675573T5/pl
Publication of PL1675573T4 publication Critical patent/PL1675573T4/pl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965Non-condensed pyrazines
    • A61K31/497Non-condensed pyrazines containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Dermatology (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
PL04795514T 2003-10-23 2004-10-18 Sterylny preparat do wstrzykiwań arypiprazolu o kontrolowanym uwalnianiu i sposób PL1675573T4 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US51361803P 2003-10-23 2003-10-23
EP04795514A EP1675573B2 (en) 2003-10-23 2004-10-18 Controlled release sterile injectable aripiprazole formulation and method
PCT/US2004/034367 WO2005041937A2 (en) 2003-10-23 2004-10-18 Controlled release sterile injectable aripiprazole formulation and method

Publications (3)

Publication Number Publication Date
PL1675573T3 true PL1675573T3 (pl) 2009-04-30
PL1675573T5 PL1675573T5 (pl) 2012-10-31
PL1675573T4 PL1675573T4 (pl) 2016-04-29

Family

ID=34549292

Family Applications (1)

Application Number Title Priority Date Filing Date
PL04795514T PL1675573T4 (pl) 2003-10-23 2004-10-18 Sterylny preparat do wstrzykiwań arypiprazolu o kontrolowanym uwalnianiu i sposób

Country Status (32)

Country Link
US (12) US7807680B2 (pl)
EP (1) EP1675573B2 (pl)
JP (2) JP4836797B2 (pl)
KR (1) KR100931784B1 (pl)
CN (1) CN1870980B (pl)
AR (2) AR046141A1 (pl)
AT (1) ATE411797T2 (pl)
AU (1) AU2004285448C1 (pl)
BR (1) BRPI0415531B8 (pl)
CA (1) CA2543242C (pl)
CO (1) CO5690539A2 (pl)
CY (2) CY1109040T1 (pl)
DE (1) DE602004017342D1 (pl)
DK (1) DK1675573T4 (pl)
EC (2) ECSP066512A (pl)
ES (1) ES2315721T5 (pl)
FR (1) FR14C0039I1 (pl)
GE (1) GEP20115205B (pl)
IL (1) IL175072A (pl)
LU (1) LU92427I2 (pl)
MX (1) MXPA06004489A (pl)
MY (1) MY146093A (pl)
NO (2) NO334919B1 (pl)
NZ (1) NZ546063A (pl)
PE (1) PE20050811A1 (pl)
PL (1) PL1675573T4 (pl)
PT (1) PT1675573E (pl)
SI (1) SI1675573T2 (pl)
TW (2) TWI421101B (pl)
UA (1) UA82561C2 (pl)
WO (1) WO2005041937A2 (pl)
ZA (1) ZA200602347B (pl)

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DK1808164T3 (da) 2006-01-05 2009-04-20 Teva Pharma Vådgranuleringsmetode til fremstilling af farmaceutiske sammensætninger af aripiprazol
CN101351193A (zh) * 2006-01-05 2009-01-21 特瓦制药工业有限公司 阿立哌唑的干法制剂
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CN115768407A (zh) * 2020-05-21 2023-03-07 江苏先声药业有限公司 一种含依匹哌唑药物组合物及其制备方法
KR102785446B1 (ko) * 2020-09-09 2025-03-25 주식회사 대웅테라퓨틱스 니클로사마이드를 포함하는 항인플루엔자 바이러스용 조성물
CN112656761B (zh) * 2020-12-30 2023-09-08 河南合智医药科技有限公司 一种低刺激性阿立哌唑前药的油溶缓释注射制剂及其制备方法
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