OA13080A - Purine compounds and uses thereof as cannabinoid receptor ligands. - Google Patents

Purine compounds and uses thereof as cannabinoid receptor ligands. Download PDF

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Publication number
OA13080A
OA13080A OA1200500128A OA1200500128A OA13080A OA 13080 A OA13080 A OA 13080A OA 1200500128 A OA1200500128 A OA 1200500128A OA 1200500128 A OA1200500128 A OA 1200500128A OA 13080 A OA13080 A OA 13080A
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OA
OAPI
Prior art keywords
alkyl
alkylamino
aryl
partially
membered
Prior art date
Application number
OA1200500128A
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English (en)
Inventor
David Andrew Griffith
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Pfizer Prod Inc
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Publication of OA13080A publication Critical patent/OA13080A/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • A—HUMAN NECESSITIES
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    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/28—Oxygen atom
    • C07D473/30—Oxygen atom attached in position 6, e.g. hypoxanthine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/40—Heterocyclic compounds containing purine ring systems with halogen atoms or perhalogeno-alkyl radicals directly attached in position 2 or 6

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  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Biomedical Technology (AREA)
  • Diabetes (AREA)
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  • Hematology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
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  • Cardiology (AREA)
  • Psychology (AREA)
  • Reproductive Health (AREA)
  • Child & Adolescent Psychology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Communicable Diseases (AREA)
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  • Gastroenterology & Hepatology (AREA)
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OA1200500128A 2002-10-28 2003-10-21 Purine compounds and uses thereof as cannabinoid receptor ligands. OA13080A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US42187402P 2002-10-28 2002-10-28

Publications (1)

Publication Number Publication Date
OA13080A true OA13080A (en) 2006-11-10

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ID=32176739

Family Applications (1)

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OA1200500128A OA13080A (en) 2002-10-28 2003-10-21 Purine compounds and uses thereof as cannabinoid receptor ligands.

Country Status (45)

Country Link
US (2) US7129239B2 (fr)
EP (1) EP1558615B8 (fr)
JP (2) JP3954618B2 (fr)
KR (1) KR100674560B1 (fr)
CN (3) CN100478343C (fr)
AP (1) AP1916A (fr)
AR (1) AR041835A1 (fr)
AT (1) ATE371658T1 (fr)
AU (1) AU2003269368B2 (fr)
BR (1) BR0314918A (fr)
CA (1) CA2503900C (fr)
CO (1) CO5560546A2 (fr)
CR (1) CR7812A (fr)
CU (1) CU23535A3 (fr)
CY (1) CY1107505T1 (fr)
DE (1) DE60316012T2 (fr)
DK (1) DK1558615T3 (fr)
DO (1) DOP2003000742A (fr)
EA (1) EA008176B1 (fr)
EC (1) ECSP055767A (fr)
EG (1) EG24662A (fr)
ES (1) ES2291669T3 (fr)
GE (1) GEP20084325B (fr)
GT (1) GT200300232A (fr)
HK (2) HK1081189A1 (fr)
HR (1) HRP20050378A2 (fr)
IS (1) IS2602B (fr)
MA (1) MA27479A1 (fr)
MX (1) MXPA05003882A (fr)
MY (1) MY140010A (fr)
NL (1) NL1024643C2 (fr)
NO (1) NO332195B1 (fr)
NZ (1) NZ539589A (fr)
OA (1) OA13080A (fr)
PE (1) PE20040781A1 (fr)
PL (1) PL376311A1 (fr)
PT (1) PT1558615E (fr)
RS (2) RS20050306A (fr)
SG (1) SG148071A1 (fr)
TN (1) TNSN05121A1 (fr)
TW (1) TWI327567B (fr)
UA (1) UA79507C2 (fr)
UY (1) UY28044A1 (fr)
WO (1) WO2004037823A1 (fr)
ZA (1) ZA200503378B (fr)

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