RS20050306A - Purine compounds and uses thereof as cannabinoid receptor ligands - Google Patents

Purine compounds and uses thereof as cannabinoid receptor ligands

Info

Publication number
RS20050306A
RS20050306A YUP-2005/0306A YUP20050306A RS20050306A RS 20050306 A RS20050306 A RS 20050306A YU P20050306 A YUP20050306 A YU P20050306A RS 20050306 A RS20050306 A RS 20050306A
Authority
RS
Serbia
Prior art keywords
receptor ligands
cannabinoid receptor
purine compounds
compounds
cannabinoid
Prior art date
Application number
YUP-2005/0306A
Other languages
English (en)
Inventor
David Andrew Griffith
Original Assignee
Pfizer Products Inc.,
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc., filed Critical Pfizer Products Inc.,
Publication of RS20050306A publication Critical patent/RS20050306A/sr

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/28—Oxygen atom
    • C07D473/30—Oxygen atom attached in position 6, e.g. hypoxanthine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/40—Heterocyclic compounds containing purine ring systems with halogen atoms or perhalogeno-alkyl radicals directly attached in position 2 or 6

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  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
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  • Veterinary Medicine (AREA)
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  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
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  • Biomedical Technology (AREA)
  • Diabetes (AREA)
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  • Hematology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
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  • Psychology (AREA)
  • Reproductive Health (AREA)
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Abstract

Opisna su jedinjenja Formule (I) koja deluju kao ligandi kanabinoidnog receptora i njihova upotreba u tretmanu bolesti povezanih sa posredovanjem kanabinoidnih receptora kod animalnih bića.
YUP-2005/0306A 2002-10-28 2003-10-21 Purine compounds and uses thereof as cannabinoid receptor ligands RS20050306A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US42187402P 2002-10-28 2002-10-28
PCT/IB2003/004619 WO2004037823A1 (en) 2002-10-28 2003-10-21 Purine compounds and uses thereof as cannabinoid receptor ligands

Publications (1)

Publication Number Publication Date
RS20050306A true RS20050306A (en) 2007-04-10

Family

ID=32176739

Family Applications (2)

Application Number Title Priority Date Filing Date
YUP-2005/0306A RS20050306A (en) 2002-10-28 2003-10-21 Purine compounds and uses thereof as cannabinoid receptor ligands
YUP-2005/0395A RS20050395A (en) 2002-10-28 2003-11-14 Ppar activators

Family Applications After (1)

Application Number Title Priority Date Filing Date
YUP-2005/0395A RS20050395A (en) 2002-10-28 2003-11-14 Ppar activators

Country Status (45)

Country Link
US (2) US7129239B2 (sr)
EP (1) EP1558615B8 (sr)
JP (2) JP3954618B2 (sr)
KR (1) KR100674560B1 (sr)
CN (3) CN100439369C (sr)
AP (1) AP1916A (sr)
AR (1) AR041835A1 (sr)
AT (1) ATE371658T1 (sr)
AU (1) AU2003269368B2 (sr)
BR (1) BR0314918A (sr)
CA (1) CA2503900C (sr)
CO (1) CO5560546A2 (sr)
CR (1) CR7812A (sr)
CU (1) CU23535A3 (sr)
CY (1) CY1107505T1 (sr)
DE (1) DE60316012T2 (sr)
DK (1) DK1558615T3 (sr)
DO (1) DOP2003000742A (sr)
EA (1) EA008176B1 (sr)
EC (1) ECSP055767A (sr)
EG (1) EG24662A (sr)
ES (1) ES2291669T3 (sr)
GE (1) GEP20084325B (sr)
GT (1) GT200300232A (sr)
HK (2) HK1081189A1 (sr)
HR (1) HRP20050378A2 (sr)
IS (1) IS2602B (sr)
MA (1) MA27479A1 (sr)
MX (1) MXPA05003882A (sr)
MY (1) MY140010A (sr)
NL (1) NL1024643C2 (sr)
NO (1) NO332195B1 (sr)
NZ (1) NZ539589A (sr)
OA (1) OA13080A (sr)
PE (1) PE20040781A1 (sr)
PL (1) PL376311A1 (sr)
PT (1) PT1558615E (sr)
RS (2) RS20050306A (sr)
SG (1) SG148071A1 (sr)
TN (1) TNSN05121A1 (sr)
TW (1) TWI327567B (sr)
UA (1) UA79507C2 (sr)
UY (1) UY28044A1 (sr)
WO (1) WO2004037823A1 (sr)
ZA (1) ZA200503378B (sr)

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