OA12295A - Combinations of depeptidyl peptidase IV inhibitorsand other antidabetic agents for the treatment of diabetes mellitus. - Google Patents

Combinations of depeptidyl peptidase IV inhibitorsand other antidabetic agents for the treatment of diabetes mellitus. Download PDF

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Publication number
OA12295A
OA12295A OA1200200388A OA1200200388A OA12295A OA 12295 A OA12295 A OA 12295A OA 1200200388 A OA1200200388 A OA 1200200388A OA 1200200388 A OA1200200388 A OA 1200200388A OA 12295 A OA12295 A OA 12295A
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OA
OAPI
Prior art keywords
inhibitor
use according
diabètes
dipeptidyl peptidase
insulin
Prior art date
Application number
OA1200200388A
Other languages
English (en)
Inventor
Jonathan Robert Sanders Arch
James Martin Lenhard
Original Assignee
Smithkline Beecham Plc
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc, Smithkline Beecham Corp filed Critical Smithkline Beecham Plc
Publication of OA12295A publication Critical patent/OA12295A/en

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/427Thiazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

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  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Obesity (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
OA1200200388A 2000-06-19 2001-06-19 Combinations of depeptidyl peptidase IV inhibitorsand other antidabetic agents for the treatment of diabetes mellitus. OA12295A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0014969.0A GB0014969D0 (en) 2000-06-19 2000-06-19 Novel method of treatment

Publications (1)

Publication Number Publication Date
OA12295A true OA12295A (en) 2003-11-10

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Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200200388A OA12295A (en) 2000-06-19 2001-06-19 Combinations of depeptidyl peptidase IV inhibitorsand other antidabetic agents for the treatment of diabetes mellitus.

Country Status (29)

Country Link
US (2) US7241756B2 (ru)
EP (2) EP2036554A1 (ru)
JP (1) JP2003535898A (ru)
KR (1) KR20030019440A (ru)
CN (1) CN1443068A (ru)
AP (1) AP2002002703A0 (ru)
AT (1) ATE419850T1 (ru)
AU (3) AU2001264148A1 (ru)
BG (1) BG107385A (ru)
BR (1) BR0111800A (ru)
CA (1) CA2413299A1 (ru)
CZ (1) CZ20024069A3 (ru)
DE (1) DE60137329D1 (ru)
DZ (1) DZ3390A1 (ru)
EA (1) EA200300036A1 (ru)
EC (1) ECSP024397A (ru)
GB (1) GB0014969D0 (ru)
HR (1) HRP20020994A2 (ru)
HU (1) HUP0301194A3 (ru)
IL (2) IL153529A0 (ru)
MA (1) MA25820A1 (ru)
MX (1) MXPA02012763A (ru)
NO (1) NO20026038L (ru)
OA (1) OA12295A (ru)
PL (1) PL360493A1 (ru)
SK (1) SK17832002A3 (ru)
WO (1) WO2001097808A1 (ru)
YU (1) YU1703A (ru)
ZA (1) ZA200300203B (ru)

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IL188471A0 (en) 2008-03-20
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GB0014969D0 (en) 2000-08-09
US7241756B2 (en) 2007-07-10
HUP0301194A2 (hu) 2003-08-28
MXPA02012763A (es) 2003-04-25
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SK17832002A3 (en) 2004-10-05
AU2008212061A1 (en) 2008-10-02
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