ECSP024397A - Combinaciones de inihibidores de dipeptildil peptidasa iv y otros agentes antidiabeticos para el tratamiento de diabetes mellitus - Google Patents
Combinaciones de inihibidores de dipeptildil peptidasa iv y otros agentes antidiabeticos para el tratamiento de diabetes mellitusInfo
- Publication number
- ECSP024397A ECSP024397A EC2002004397A ECSP024397A ECSP024397A EC SP024397 A ECSP024397 A EC SP024397A EC 2002004397 A EC2002004397 A EC 2002004397A EC SP024397 A ECSP024397 A EC SP024397A EC SP024397 A ECSP024397 A EC SP024397A
- Authority
- EC
- Ecuador
- Prior art keywords
- treatment
- dipeptildil
- peptidasa
- inihibitors
- combinations
- Prior art date
Links
- 206010012601 diabetes mellitus Diseases 0.000 title abstract 3
- 239000003472 antidiabetic agent Substances 0.000 title abstract 2
- 229940125708 antidiabetic agent Drugs 0.000 title abstract 2
- 241000124008 Mammalia Species 0.000 abstract 2
- 229940124213 Dipeptidyl peptidase 4 (DPP IV) inhibitor Drugs 0.000 abstract 1
- 239000003603 dipeptidyl peptidase IV inhibitor Substances 0.000 abstract 1
- 231100000252 nontoxic Toxicity 0.000 abstract 1
- 230000003000 nontoxic effect Effects 0.000 abstract 1
- 208000001072 type 2 diabetes mellitus Diseases 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- General Chemical & Material Sciences (AREA)
- Obesity (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Un método para el tratamiento de diabetes mellitus, especialmente diabetes de tipo 2, y condiciones asociadas con diabetes mellitus, en un mamífero como un humano; dicho método comprende administrar una cantidad efectiva, no tóxica y farmacéuticamente aceptable de un inhibidor de dipeptidil peptidasa IV y otro agente antidiabético, a un mamífero en necesidad del mismo.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0014969.0A GB0014969D0 (en) | 2000-06-19 | 2000-06-19 | Novel method of treatment |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP024397A true ECSP024397A (es) | 2003-02-06 |
Family
ID=9893956
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2002004397A ECSP024397A (es) | 2000-06-19 | 2002-12-19 | Combinaciones de inihibidores de dipeptildil peptidasa iv y otros agentes antidiabeticos para el tratamiento de diabetes mellitus |
Country Status (29)
| Country | Link |
|---|---|
| US (2) | US7241756B2 (es) |
| EP (2) | EP2036554A1 (es) |
| JP (1) | JP2003535898A (es) |
| KR (1) | KR20030019440A (es) |
| CN (1) | CN1443068A (es) |
| AP (1) | AP2002002703A0 (es) |
| AT (1) | ATE419850T1 (es) |
| AU (3) | AU2001264148A1 (es) |
| BG (1) | BG107385A (es) |
| BR (1) | BR0111800A (es) |
| CA (1) | CA2413299A1 (es) |
| CZ (1) | CZ20024069A3 (es) |
| DE (1) | DE60137329D1 (es) |
| DZ (1) | DZ3390A1 (es) |
| EA (1) | EA200300036A1 (es) |
| EC (1) | ECSP024397A (es) |
| GB (1) | GB0014969D0 (es) |
| HR (1) | HRP20020994A2 (es) |
| HU (1) | HUP0301194A3 (es) |
| IL (2) | IL153529A0 (es) |
| MA (1) | MA25820A1 (es) |
| MX (1) | MXPA02012763A (es) |
| NO (1) | NO20026038L (es) |
| OA (1) | OA12295A (es) |
| PL (1) | PL360493A1 (es) |
| SK (1) | SK17832002A3 (es) |
| WO (1) | WO2001097808A1 (es) |
| YU (1) | YU1703A (es) |
| ZA (1) | ZA200300203B (es) |
Families Citing this family (111)
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|---|---|---|---|---|
| DE19828113A1 (de) | 1998-06-24 | 2000-01-05 | Probiodrug Ges Fuer Arzneim | Prodrugs von Inhibitoren der Dipeptidyl Peptidase IV |
| DE19940130A1 (de) | 1999-08-24 | 2001-03-01 | Probiodrug Ges Fuer Arzneim | Neue Effektoren der Dipeptidyl Peptidase IV zur topischen Anwendung |
| GB0014969D0 (en) * | 2000-06-19 | 2000-08-09 | Smithkline Beecham Plc | Novel method of treatment |
| US6890905B2 (en) | 2001-04-02 | 2005-05-10 | Prosidion Limited | Methods for improving islet signaling in diabetes mellitus and for its prevention |
| GB0109146D0 (en) * | 2001-04-11 | 2001-05-30 | Ferring Bv | Treatment of type 2 diabetes |
| US7368421B2 (en) | 2001-06-27 | 2008-05-06 | Probiodrug Ag | Use of dipeptidyl peptidase IV inhibitors in the treatment of multiple sclerosis |
| US20030130199A1 (en) | 2001-06-27 | 2003-07-10 | Von Hoersten Stephan | Dipeptidyl peptidase IV inhibitors and their uses as anti-cancer agents |
| JP2004521149A (ja) * | 2001-06-27 | 2004-07-15 | プロバイオドラッグ アーゲー | 新規なジペプチジルぺプチダ−ゼiv阻害剤およびそれらの抗癌剤としての使用 |
| DE10150203A1 (de) | 2001-10-12 | 2003-04-17 | Probiodrug Ag | Peptidylketone als Inhibitoren der DPIV |
| WO2003002531A2 (en) | 2001-06-27 | 2003-01-09 | Smithkline Beecham Corporation | Fluoropyrrolidines as dipeptidyl peptidase inhibitors |
| US6844316B2 (en) | 2001-09-06 | 2005-01-18 | Probiodrug Ag | Inhibitors of dipeptidyl peptidase I |
| DK1480961T3 (da) | 2002-02-28 | 2007-05-07 | Prosidion Ltd | Glutaminylbaserede DPIV-inhibitorer |
| AU2007203210B2 (en) * | 2002-05-29 | 2009-10-01 | Novartis Ag | Combination of a DPP IV inhibitor and a cardiovascular compound |
| GB0212412D0 (en) * | 2002-05-29 | 2002-07-10 | Novartis Ag | Combination of organic compounds |
| US6710040B1 (en) | 2002-06-04 | 2004-03-23 | Pfizer Inc. | Fluorinated cyclic amides as dipeptidyl peptidase IV inhibitors |
| BRPI0313648B8 (pt) * | 2002-08-21 | 2021-05-25 | Boehringer Ingelheim Pharma | 8-[3-amino-piperidin-1-il]-xantinas, seus sais fisiologicamente compatíveis, seus usos e seus processos de preparação, bem como medicamentos que as contêm e seus processos de preparação |
| US7407955B2 (en) | 2002-08-21 | 2008-08-05 | Boehringer Ingelheim Pharma Gmbh & Co., Kg | 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions |
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| RU2328280C2 (ru) * | 2002-09-26 | 2008-07-10 | Эйсай Ар Энд Ди Менеджмент Ко., Лтд. | Комбинационное лекарство |
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| KR20120035203A (ko) | 2003-05-05 | 2012-04-13 | 프로비오드룩 아게 | 글루타미닐 및 글루타메이트 사이클라제의 이펙터의 용도 |
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| US20050070531A1 (en) | 2003-08-13 | 2005-03-31 | Syrrx, Inc. | Dipeptidyl peptidase inhibitors |
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2000
- 2000-06-19 GB GBGB0014969.0A patent/GB0014969D0/en not_active Ceased
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2001
- 2001-06-19 HR HR20020994A patent/HRP20020994A2/hr not_active Application Discontinuation
- 2001-06-19 AP APAP/P/2002/002703A patent/AP2002002703A0/en unknown
- 2001-06-19 MX MXPA02012763A patent/MXPA02012763A/es active IP Right Grant
- 2001-06-19 WO PCT/GB2001/002696 patent/WO2001097808A1/en active Application Filing
- 2001-06-19 DZ DZ013390A patent/DZ3390A1/xx active
- 2001-06-19 YU YU1703A patent/YU1703A/sh unknown
- 2001-06-19 CA CA002413299A patent/CA2413299A1/en not_active Abandoned
- 2001-06-19 KR KR1020027017279A patent/KR20030019440A/ko not_active Ceased
- 2001-06-19 JP JP2002503292A patent/JP2003535898A/ja not_active Withdrawn
- 2001-06-19 AT AT01938472T patent/ATE419850T1/de not_active IP Right Cessation
- 2001-06-19 CZ CZ20024069A patent/CZ20024069A3/cs unknown
- 2001-06-19 SK SK17832002A patent/SK17832002A3/sk not_active Application Discontinuation
- 2001-06-19 CN CN01813126A patent/CN1443068A/zh active Pending
- 2001-06-19 AU AU2001264148A patent/AU2001264148A1/en not_active Abandoned
- 2001-06-19 EA EA200300036A patent/EA200300036A1/ru unknown
- 2001-06-19 HU HU0301194A patent/HUP0301194A3/hu unknown
- 2001-06-19 EP EP08168689A patent/EP2036554A1/en not_active Withdrawn
- 2001-06-19 EP EP01938472A patent/EP1292300B1/en not_active Expired - Lifetime
- 2001-06-19 IL IL15352901A patent/IL153529A0/xx unknown
- 2001-06-19 OA OA1200200388A patent/OA12295A/en unknown
- 2001-06-19 PL PL36049301A patent/PL360493A1/xx unknown
- 2001-06-19 DE DE60137329T patent/DE60137329D1/de not_active Expired - Fee Related
- 2001-06-19 BR BR0111800-5A patent/BR0111800A/pt not_active Application Discontinuation
-
2002
- 2002-12-12 BG BG107385A patent/BG107385A/bg unknown
- 2002-12-16 NO NO20026038A patent/NO20026038L/no not_active Application Discontinuation
- 2002-12-18 MA MA26965A patent/MA25820A1/fr unknown
- 2002-12-19 EC EC2002004397A patent/ECSP024397A/es unknown
-
2003
- 2003-01-08 ZA ZA200300203A patent/ZA200300203B/en unknown
-
2005
- 2005-11-11 AU AU2005232303A patent/AU2005232303A1/en not_active Abandoned
-
2006
- 2006-06-01 US US11/421,548 patent/US7241756B2/en not_active Expired - Fee Related
-
2007
- 2007-06-05 US US11/758,259 patent/US20070238756A1/en not_active Abandoned
- 2007-12-27 IL IL188471A patent/IL188471A0/en unknown
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2008
- 2008-09-08 AU AU2008212061A patent/AU2008212061A1/en not_active Abandoned
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