BR0111800A - Combinações de inibidores de depeptidil peptidase iv e outros agentes antidiabéticos para o tratamento de diabete mellitus - Google Patents

Combinações de inibidores de depeptidil peptidase iv e outros agentes antidiabéticos para o tratamento de diabete mellitus

Info

Publication number
BR0111800A
BR0111800A BR0111800-5A BR0111800A BR0111800A BR 0111800 A BR0111800 A BR 0111800A BR 0111800 A BR0111800 A BR 0111800A BR 0111800 A BR0111800 A BR 0111800A
Authority
BR
Brazil
Prior art keywords
diabetes mellitus
treatment
antidiabetic agents
inhibitor combinations
peptidase
Prior art date
Application number
BR0111800-5A
Other languages
English (en)
Inventor
Jonathan Roberts Sanders Arch
James Martin Lenhard
Original Assignee
Smithkline Beecham Plc
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc, Smithkline Beecham Corp filed Critical Smithkline Beecham Plc
Publication of BR0111800A publication Critical patent/BR0111800A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/427Thiazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Abstract

"COMBINAçõES DE INIBIDORES DE DEPEPTIDIL PEPTIDASE IV E OUTROS AGENTES ANTIDIABéTICOS PARA O TRATAMENTO DE DIABETE MELLITUS". Trata-se de um método para o tratamento de diabetes mellitus, especialmente diabetes tipo 2 e condições associadas a diabetes mellitus em um mamífero como um ser humano, cujo método compreende administrar uma quantidade eficaz, não tóxica e farmaceuticamente aceitável de um inibidor de dipeptidil peptidase IV e outro agente antidiabético, a um mamífero necessitando do mesmo.
BR0111800-5A 2000-06-19 2001-06-19 Combinações de inibidores de depeptidil peptidase iv e outros agentes antidiabéticos para o tratamento de diabete mellitus BR0111800A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0014969.0A GB0014969D0 (en) 2000-06-19 2000-06-19 Novel method of treatment
PCT/GB2001/002696 WO2001097808A1 (en) 2000-06-19 2001-06-19 Combinations of depeptidyl peptidase iv inhibitors and other antidiabetic agents for the treatment of diabete mellitus

Publications (1)

Publication Number Publication Date
BR0111800A true BR0111800A (pt) 2003-05-27

Family

ID=9893956

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0111800-5A BR0111800A (pt) 2000-06-19 2001-06-19 Combinações de inibidores de depeptidil peptidase iv e outros agentes antidiabéticos para o tratamento de diabete mellitus

Country Status (29)

Country Link
US (2) US7241756B2 (pt)
EP (2) EP1292300B1 (pt)
JP (1) JP2003535898A (pt)
KR (1) KR20030019440A (pt)
CN (1) CN1443068A (pt)
AP (1) AP2002002703A0 (pt)
AT (1) ATE419850T1 (pt)
AU (3) AU2001264148A1 (pt)
BG (1) BG107385A (pt)
BR (1) BR0111800A (pt)
CA (1) CA2413299A1 (pt)
CZ (1) CZ20024069A3 (pt)
DE (1) DE60137329D1 (pt)
DZ (1) DZ3390A1 (pt)
EA (1) EA200300036A1 (pt)
EC (1) ECSP024397A (pt)
GB (1) GB0014969D0 (pt)
HR (1) HRP20020994A2 (pt)
HU (1) HUP0301194A3 (pt)
IL (2) IL153529A0 (pt)
MA (1) MA25820A1 (pt)
MX (1) MXPA02012763A (pt)
NO (1) NO20026038L (pt)
OA (1) OA12295A (pt)
PL (1) PL360493A1 (pt)
SK (1) SK17832002A3 (pt)
WO (1) WO2001097808A1 (pt)
YU (1) YU1703A (pt)
ZA (1) ZA200300203B (pt)

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OA12295A (en) 2003-11-10
CZ20024069A3 (cs) 2004-02-18
MA25820A1 (fr) 2003-07-01
EP2036554A1 (en) 2009-03-18
AU2005232303A1 (en) 2005-12-01
AU2001264148A1 (en) 2002-01-02
AP2002002703A0 (en) 2002-12-31
GB0014969D0 (en) 2000-08-09
NO20026038L (no) 2003-02-03
PL360493A1 (en) 2004-09-06
EP1292300A1 (en) 2003-03-19
ZA200300203B (en) 2004-03-26
EA200300036A1 (ru) 2003-04-24
HUP0301194A3 (en) 2007-09-28
DE60137329D1 (de) 2009-02-26
DZ3390A1 (fr) 2001-12-27
JP2003535898A (ja) 2003-12-02
US20070238756A1 (en) 2007-10-11
ECSP024397A (es) 2003-02-06
US20060205675A1 (en) 2006-09-14
CA2413299A1 (en) 2001-12-27
CN1443068A (zh) 2003-09-17
IL153529A0 (en) 2003-07-06
HUP0301194A2 (hu) 2003-08-28
US7241756B2 (en) 2007-07-10
SK17832002A3 (en) 2004-10-05
MXPA02012763A (es) 2003-04-25
YU1703A (sh) 2006-03-03
IL188471A0 (en) 2008-03-20
ATE419850T1 (de) 2009-01-15
HRP20020994A2 (en) 2005-02-28
NO20026038D0 (no) 2002-12-16
AU2008212061A1 (en) 2008-10-02
BG107385A (bg) 2003-09-30
WO2001097808A1 (en) 2001-12-27
KR20030019440A (ko) 2003-03-06

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