NO951594D0 - N-(2-amino-4,6-diklorpyrimidin-5-yl) formamid, samt fremgangsmåte ved fremstilling derav - Google Patents

N-(2-amino-4,6-diklorpyrimidin-5-yl) formamid, samt fremgangsmåte ved fremstilling derav

Info

Publication number
NO951594D0
NO951594D0 NO951594A NO951594A NO951594D0 NO 951594 D0 NO951594 D0 NO 951594D0 NO 951594 A NO951594 A NO 951594A NO 951594 A NO951594 A NO 951594A NO 951594 D0 NO951594 D0 NO 951594D0
Authority
NO
Norway
Prior art keywords
formula
amino
alkyl
dichloropyrimidin
formamide
Prior art date
Application number
NO951594A
Other languages
English (en)
Other versions
NO306461B1 (no
NO951594L (no
Inventor
Gerhard Stucky
Rene Imwinkelried
Original Assignee
Lonza Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=4207186&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO951594(D0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lonza Ag filed Critical Lonza Ag
Publication of NO951594D0 publication Critical patent/NO951594D0/no
Publication of NO951594L publication Critical patent/NO951594L/no
Publication of NO306461B1 publication Critical patent/NO306461B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Virology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
NO951594A 1994-04-27 1995-04-26 N-(2-amino-4,6-diklorpyrimidin-5-yl) formamid samt fremgangsmÕte ved fremstilling derav NO306461B1 (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH129994 1994-04-27

Publications (3)

Publication Number Publication Date
NO951594D0 true NO951594D0 (no) 1995-04-26
NO951594L NO951594L (no) 1995-10-30
NO306461B1 NO306461B1 (no) 1999-11-08

Family

ID=4207186

Family Applications (2)

Application Number Title Priority Date Filing Date
NO951594A NO306461B1 (no) 1994-04-27 1995-04-26 N-(2-amino-4,6-diklorpyrimidin-5-yl) formamid samt fremgangsmÕte ved fremstilling derav
NO984588A NO306859B1 (no) 1994-04-27 1998-10-01 Fremgangsmåte for fremstilling av 2,5-di-amino-4,6-diklorpyrimidin

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO984588A NO306859B1 (no) 1994-04-27 1998-10-01 Fremgangsmåte for fremstilling av 2,5-di-amino-4,6-diklorpyrimidin

Country Status (18)

Country Link
US (4) US5583226A (no)
EP (2) EP0684236B2 (no)
JP (2) JP3811966B2 (no)
KR (1) KR100327996B1 (no)
CN (2) CN1065862C (no)
AT (2) ATE167672T1 (no)
CA (1) CA2145928C (no)
CZ (1) CZ287261B6 (no)
DE (2) DE59502637D1 (no)
DK (2) DK0684236T4 (no)
ES (2) ES2201229T3 (no)
FI (2) FI109119B (no)
HU (3) HU219986B (no)
NO (2) NO306461B1 (no)
PL (1) PL190855B1 (no)
PT (1) PT816344E (no)
SK (1) SK282208B6 (no)
TW (1) TW442474B (no)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9402161D0 (en) * 1994-02-04 1994-03-30 Wellcome Found Chloropyrimidine intermediates
CA2145928C (en) * 1994-04-27 2007-10-09 Gerhard Stucky N-(2-amino-4,6-dichloropyrimidin-5-yl)formamide, and a process for its preparation
AU1158000A (en) * 1998-10-30 2000-05-22 Lonza A.G. Method for producing 4- ((2',5'- diamino-6'- halopyrimidine- 4'-YL)amino)- cyclopent- 2-enylmethanols
DE59905679D1 (de) 1998-10-30 2003-06-26 Lonza Ag Verfahren zur herstellung von 4-[(2',5'-diamino-6'-halogenpyrimidin-4'-yl)amino]-cyclopent-2-enylmethanolen
EP1188750B1 (de) * 1998-12-21 2003-10-15 Lonza AG Verfahren zur Herstellung von 2,5-Diamino-4,6-dihalogenpyrimidinen
US6608199B2 (en) 2000-07-07 2003-08-19 Syngenta Limited Synthesis of chlorinated pyrimidines
JP2002223094A (ja) * 2001-01-25 2002-08-09 Yokohama Rubber Co Ltd:The 電波吸収体の構造
US6982331B2 (en) * 2001-06-08 2006-01-03 Syngenta Crop Protection, Inc. Synthesis of chlorinated pyrimidines
FR2849030A1 (fr) * 2002-12-20 2004-06-25 Isochem Sa Procede de preparation des n-(2-amino-4, 6-dihalogenopyrimidin-5-yl) formamides
JPWO2004103979A1 (ja) * 2003-05-26 2006-07-20 住友化学株式会社 Ｎ−（２−アミノ−４，６−ジクロロピリミジン−５−イル）ホルムアミドの製造方法
DE102004002055A1 (de) * 2004-01-15 2005-08-11 Degussa Ag Verfahren zur Herstellung von 2-Amino-4,6-dichlor-5-formamidopyrimidin
CN101003511B (zh) * 2007-01-19 2010-06-09 中国科学院上海有机化学研究所 制备2-氨基-4,6-二氯-5-甲酰氨基嘧啶的方法
CN102127022A (zh) * 2010-12-30 2011-07-20 苏州开元民生科技股份有限公司 2-氨基-4,6-二氯-5-甲酰胺基嘧啶的合成方法
CZ305457B6 (cs) * 2011-02-28 2015-09-30 Ústav organické chemie a biochemie, Akademie věd ČR v. v. i. Pyrimidinové sloučeniny inhibující tvorbu oxidu dusnatého a prostaglandinu E2, způsob výroby a použití
CZ305750B6 (cs) * 2012-01-26 2016-03-02 Ústav Organické Chemie A Biochemie Akademie Věd Čr, V.V.I. Způsob výroby N-9 substituovaných analogů purinu
CN102702110A (zh) * 2012-05-24 2012-10-03 盛世泰科生物医药技术(苏州)有限公司 一种4-氨基-5,6-二氯嘧啶的制备方法
WO2014023681A1 (en) * 2012-08-06 2014-02-13 Enantia, S.L. A process for the preparation of an intermediate for a triazolopyrimidine carbonucleoside

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8916698D0 (en) * 1989-07-21 1989-09-06 Beecham Group Plc Novel process
SK279618B6 (sk) * 1992-01-22 1999-01-11 Lonza A.G. (Dir.:Basel) N-5-chránené 2,5-diamino-4,6-dichlórpyrimidíny a s
GB9402161D0 (en) * 1994-02-04 1994-03-30 Wellcome Found Chloropyrimidine intermediates
CA2145928C (en) * 1994-04-27 2007-10-09 Gerhard Stucky N-(2-amino-4,6-dichloropyrimidin-5-yl)formamide, and a process for its preparation

Also Published As

Publication number Publication date
NO306461B1 (no) 1999-11-08
NO306859B1 (no) 2000-01-03
HU0003724D0 (no) 2000-11-28
KR100327996B1 (ko) 2002-07-27
CN1113237A (zh) 1995-12-13
ATE167672T1 (de) 1998-07-15
CN1193991C (zh) 2005-03-23
ES2120099T3 (es) 1998-10-16
HU219716B (hu) 2001-06-28
EP0684236B2 (de) 2007-12-26
PT816344E (pt) 2003-10-31
ES2201229T3 (es) 2004-03-16
US5583226A (en) 1996-12-10
FI952009A0 (fi) 1995-04-27
ES2120099T5 (es) 2008-05-16
PL190855B1 (pl) 2006-02-28
NO984588D0 (no) 1998-10-01
TW442474B (en) 2001-06-23
ATE243200T1 (de) 2003-07-15
CZ287261B6 (en) 2000-10-11
CZ106795A3 (en) 1995-11-15
HU219712B (hu) 2001-06-28
KR950032143A (ko) 1995-12-20
DE59502637D1 (de) 1998-07-30
DK0816344T3 (da) 2003-10-06
CA2145928A1 (en) 1995-10-28
US5744601A (en) 1998-04-28
PL308394A1 (en) 1995-10-30
EP0816344A1 (de) 1998-01-07
JP2006199707A (ja) 2006-08-03
HU0003725D0 (no) 1995-04-26
EP0684236A3 (de) 1996-07-17
EP0684236A2 (de) 1995-11-29
EP0816344B1 (de) 2003-06-18
US5693800A (en) 1997-12-02
CN1259517A (zh) 2000-07-12
FI109693B (fi) 2002-09-30
NO984588L (no) 1995-10-30
HU9501194D0 (en) 1995-06-28
FI109119B (fi) 2002-05-31
CN1065862C (zh) 2001-05-16
SK54195A3 (en) 1995-11-08
NO951594L (no) 1995-10-30
JP4525625B2 (ja) 2010-08-18
HUT70700A (en) 1995-10-30
HU219986B (hu) 2001-10-28
DK0684236T4 (da) 2008-05-05
EP0684236B1 (de) 1998-06-24
FI20011433A (fi) 2001-07-02
JP3811966B2 (ja) 2006-08-23
FI952009A (fi) 1995-10-28
DE59510726D1 (de) 2003-07-24
CA2145928C (en) 2007-10-09
DK0684236T3 (da) 1998-11-02
US5663340A (en) 1997-09-02
SK282208B6 (sk) 2001-12-03
JPH07300466A (ja) 1995-11-14

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