NO331925B1 - Substituerte pyrimidiner som proteinkinase-inhibitorer - Google Patents
Substituerte pyrimidiner som proteinkinase-inhibitorer Download PDFInfo
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- NO331925B1 NO331925B1 NO20050144A NO20050144A NO331925B1 NO 331925 B1 NO331925 B1 NO 331925B1 NO 20050144 A NO20050144 A NO 20050144A NO 20050144 A NO20050144 A NO 20050144A NO 331925 B1 NO331925 B1 NO 331925B1
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- Prior art keywords
- aurora
- kinase
- cancer
- pharmaceutically acceptable
- agents
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Classifications
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- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/34—One oxygen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
Landscapes
- Health & Medical Sciences (AREA)
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- Organic Chemistry (AREA)
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- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
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- Engineering & Computer Science (AREA)
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- Immunology (AREA)
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- Biomedical Technology (AREA)
- Neurology (AREA)
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- Hematology (AREA)
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- Oncology (AREA)
- Urology & Nephrology (AREA)
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- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
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- Obesity (AREA)
- Endocrinology (AREA)
- Cardiology (AREA)
- Gastroenterology & Hepatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US39065802P | 2002-06-20 | 2002-06-20 | |
| US41160902P | 2002-09-18 | 2002-09-18 | |
| PCT/US2003/019266 WO2004000833A1 (en) | 2002-06-20 | 2003-06-19 | Processes for preparing substituted pyrimidines and pyrimidine derivatives as inhibitors of protein kinase |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20050144D0 NO20050144D0 (no) | 2005-01-11 |
| NO20050144L NO20050144L (no) | 2005-03-21 |
| NO331925B1 true NO331925B1 (no) | 2012-05-07 |
Family
ID=30003168
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20050144A NO331925B1 (no) | 2002-06-20 | 2005-01-11 | Substituerte pyrimidiner som proteinkinase-inhibitorer |
| NO20110523A NO20110523L (no) | 2002-06-20 | 2011-04-05 | Fremgangsmate for a fremstille substituerte pyrimidiner |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20110523A NO20110523L (no) | 2002-06-20 | 2011-04-05 | Fremgangsmate for a fremstille substituerte pyrimidiner |
Country Status (27)
| Country | Link |
|---|---|
| US (4) | US20040049032A1 (ru) |
| EP (4) | EP1517905B1 (ru) |
| JP (5) | JP4237701B2 (ru) |
| KR (2) | KR101141959B1 (ru) |
| CN (1) | CN100484934C (ru) |
| AR (1) | AR040286A1 (ru) |
| AT (2) | ATE556068T1 (ru) |
| AU (1) | AU2003245568B2 (ru) |
| BR (1) | BR0312443A (ru) |
| CA (1) | CA2489824C (ru) |
| CO (1) | CO5680433A2 (ru) |
| DE (1) | DE60336092D1 (ru) |
| EA (2) | EA015990B1 (ru) |
| EC (1) | ECSP055561A (ru) |
| ES (1) | ES2386781T3 (ru) |
| HK (3) | HK1077057A1 (ru) |
| HR (1) | HRP20050064A2 (ru) |
| IL (1) | IL165849A0 (ru) |
| IS (2) | IS7606A (ru) |
| MX (1) | MXPA05000068A (ru) |
| MY (1) | MY141867A (ru) |
| NO (2) | NO331925B1 (ru) |
| NZ (4) | NZ537720A (ru) |
| PL (1) | PL374953A1 (ru) |
| SG (1) | SG170614A1 (ru) |
| TW (2) | TWI297684B (ru) |
| WO (1) | WO2004000833A1 (ru) |
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