NO323143B1 - Fremgangsmate for fremstilling av en legemiddelbaerer - Google Patents
Fremgangsmate for fremstilling av en legemiddelbaerer Download PDFInfo
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- NO323143B1 NO323143B1 NO19972142A NO972142A NO323143B1 NO 323143 B1 NO323143 B1 NO 323143B1 NO 19972142 A NO19972142 A NO 19972142A NO 972142 A NO972142 A NO 972142A NO 323143 B1 NO323143 B1 NO 323143B1
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- particles
- drug carrier
- drug
- active ingredient
- dispersed
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B82—NANOTECHNOLOGY
- B82Y—SPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
- B82Y5/00—Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dispersion Chemistry (AREA)
- Dermatology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Emulsifying, Dispersing, Foam-Producing Or Wetting Agents (AREA)
- Colloid Chemistry (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4440337A DE4440337A1 (de) | 1994-11-11 | 1994-11-11 | Pharmazeutische Nanosuspensionen zur Arzneistoffapplikation als Systeme mit erhöhter Sättigungslöslichkeit und Lösungsgeschwindigkeit |
| PCT/EP1995/004401 WO1996014830A1 (de) | 1994-11-11 | 1995-11-09 | Pharmazeutische nanosuspensionen zur arzneistoffapplikation als systeme mit erhöhter sättigungslöslichkeit und lösungsgeschwindigkeit |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO972142D0 NO972142D0 (no) | 1997-05-09 |
| NO972142L NO972142L (no) | 1997-06-26 |
| NO323143B1 true NO323143B1 (no) | 2007-01-08 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO19972142A NO323143B1 (no) | 1994-11-11 | 1997-05-09 | Fremgangsmate for fremstilling av en legemiddelbaerer |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US5858410A (hu) |
| EP (1) | EP0790821B1 (hu) |
| JP (1) | JP3977418B2 (hu) |
| KR (1) | KR100480447B1 (hu) |
| CN (1) | CN1210018C (hu) |
| AT (1) | ATE278387T1 (hu) |
| AU (1) | AU714978B2 (hu) |
| CA (1) | CA2205046C (hu) |
| CZ (1) | CZ293253B6 (hu) |
| DE (3) | DE4440337A1 (hu) |
| EE (1) | EE9700217A (hu) |
| ES (1) | ES2229242T3 (hu) |
| FI (1) | FI119465B (hu) |
| HU (1) | HU228097B1 (hu) |
| MX (1) | MX9703399A (hu) |
| NO (1) | NO323143B1 (hu) |
| PL (1) | PL320085A1 (hu) |
| SK (1) | SK284541B6 (hu) |
| WO (1) | WO1996014830A1 (hu) |
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| JP4484247B2 (ja) * | 1995-02-24 | 2010-06-16 | エラン ファーマ インターナショナル，リミティド | ナノ粒子分散体を含有するエアロゾル |
| US6465016B2 (en) | 1996-08-22 | 2002-10-15 | Research Triangle Pharmaceuticals | Cyclosporiine particles |
| US7255877B2 (en) * | 1996-08-22 | 2007-08-14 | Jagotec Ag | Fenofibrate microparticles |
| GB9625589D0 (en) * | 1996-12-10 | 1997-01-29 | Boots Co Plc | Therapeutic agents |
| JP3821407B2 (ja) * | 1997-06-26 | 2006-09-13 | 富士写真フイルム株式会社 | 感光性画像形成媒体塗布液の製造方法および熱現像感光材料 |
| US7799337B2 (en) | 1997-07-21 | 2010-09-21 | Levin Bruce H | Method for directed intranasal administration of a composition |
| US6432986B2 (en) | 1997-07-21 | 2002-08-13 | Bruce H. Levin | Compositions, kits, and methods for inhibiting cerebral neurovascular disorders and muscular headaches |
| US6045815A (en) * | 1997-08-15 | 2000-04-04 | Board Of Regents, The University Of Texas System | Parenteral pimaricin as treatment of systemic infections |
| US6844004B2 (en) * | 1997-08-15 | 2005-01-18 | Board Of Regents, The University Of Texas System | Topical formulations of natamycin/pimaricin |
| GB9718568D0 (en) | 1997-09-03 | 1997-11-05 | Chauvin Pharmaceuticals Limite | Compositions |
| EP1010435B1 (en) * | 1997-09-05 | 2010-11-03 | Maruho K.K. | Nanocapsule preparations for treating intraarticular diseases |
| PT1033132E (pt) * | 1997-10-20 | 2005-09-30 | Dainippon Pharmaceutical Co | Composicao de farmaco rapidamente soluvel |
| JP2001526194A (ja) * | 1997-12-19 | 2001-12-18 | ターロ ファーマシューティカルズ ユーエスエイ インコーポレイテッド | 局所的カルバマゼピン製剤及び使用方法 |
| US6287693B1 (en) | 1998-02-25 | 2001-09-11 | John Claude Savoir | Stable shaped particles of crystalline organic compounds |
| US6337092B1 (en) | 1998-03-30 | 2002-01-08 | Rtp Pharma Inc. | Composition and method of preparing microparticles of water-insoluble substances |
| JP4709378B2 (ja) | 1998-03-30 | 2011-06-22 | オバン・エナジー・リミテッド | 水不溶性物質のマイクロ粒子を製造するための組成物及び方法 |
| US7381423B2 (en) * | 1998-05-11 | 2008-06-03 | Ciba Specialty Chemicals Corp. | Use of nanodispersions in cosmetic end formulations |
| ATE259220T1 (de) | 1998-05-29 | 2004-02-15 | Skyepharma Canada Inc | Gegen hitzeeinwirkung geschützte mikropartikel und verfahren zur terminalen dampfsterilisation derselben |
| CN1221249C (zh) * | 1998-08-19 | 2005-10-05 | 斯凯伊药品加拿大公司 | 普鲁泊福的可注射水分散体 |
| US20040013613A1 (en) * | 2001-05-18 | 2004-01-22 | Jain Rajeev A | Rapidly disintegrating solid oral dosage form |
| JP2002527367A (ja) * | 1998-10-14 | 2002-08-27 | コグニス・ドイチュラント・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング | ナノスケールのステロールおよびステロールエステルの使用 |
| US20090297602A1 (en) * | 1998-11-02 | 2009-12-03 | Devane John G | Modified Release Loxoprofen Compositions |
| ID29270A (id) | 1998-11-20 | 2001-08-16 | Rtp Pharma Inc | Partikel-partikel mikro yang distabilkan oleh fosfolipid yang dapat menyebar |
| DE19856432A1 (de) | 1998-12-08 | 2000-06-15 | Basf Ag | Nanopartikuläre Kern-Schale Systeme sowie deren Verwendung in pharmazeutischen und kosmetischen Zubereitungen |
| NZ512599A (en) | 1998-12-30 | 2003-10-31 | Dexcel Ltd | Formulation for cyclosporin administration featuring a hydrophilic solvent and a surfactant with a HLB of less than 5 |
| WO2000067800A2 (de) * | 1999-05-07 | 2000-11-16 | Pharmasol Gmbh | Arzneistoffträger zur kontrollierten wirkstoffapplikation hergestellt aus lipidmatrix-arzneistoff-konjugaten (lak-partikel) |
| DE19932157A1 (de) * | 1999-07-13 | 2001-01-18 | Pharmasol Gmbh | Verfahren zur schonenden Herstellung von hochfeinen Mikropartikeln und Nanopartikeln |
| EP1214059B1 (en) * | 1999-09-21 | 2005-05-25 | Skyepharma Canada Inc. | Surface modified particulate compositions of biologically active substances |
| US7732404B2 (en) * | 1999-12-30 | 2010-06-08 | Dexcel Ltd | Pro-nanodispersion for the delivery of cyclosporin |
| US20040009229A1 (en) * | 2000-01-05 | 2004-01-15 | Unger Evan Charles | Stabilized nanoparticle formulations of camptotheca derivatives |
| AU2001245947A1 (en) * | 2000-03-23 | 2001-10-03 | Collaborative Technologies, Inc | Method for preparing high pressure/high shear dispersions containing physiologically active ingredients |
| US8404217B2 (en) * | 2000-05-10 | 2013-03-26 | Novartis Ag | Formulation for pulmonary administration of antifungal agents, and associated methods of manufacture and use |
| US6495164B1 (en) * | 2000-05-25 | 2002-12-17 | Alkermes Controlled Therapeutics, Inc. I | Preparation of injectable suspensions having improved injectability |
| USRE44145E1 (en) | 2000-07-07 | 2013-04-09 | A.V. Topchiev Institute Of Petrochemical Synthesis | Preparation of hydrophilic pressure sensitive adhesives having optimized adhesive properties |
| DE10036871A1 (de) | 2000-07-28 | 2002-02-14 | Pharmasol Gmbh | Dispersionen zur Formulierung wenig oder schwer löslicher Wirkstoffe |
| US6623765B1 (en) * | 2000-08-01 | 2003-09-23 | University Of Florida, Research Foundation, Incorporated | Microemulsion and micelle systems for solubilizing drugs |
| DE10043321B4 (de) * | 2000-08-24 | 2005-07-28 | Neurobiotec Gmbh | Verwendung eines transdermalen therapeutischen Systems zur Behandlung der Parkinsonschen Krankheit, zur Behandlung und Prävention des prämenstruellen Syndroms und zur Lactationshemmung |
| DE10053397A1 (de) * | 2000-10-20 | 2002-05-02 | Schering Ag | Verwendung eines dopaminergen Wirkstoffes zur Behandlung von dopaminerg behandelbaren Erkrankungen |
| CA2420597C (en) | 2000-08-31 | 2011-05-17 | Rtp Pharma Inc. | Milled particles |
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| WO2018129555A1 (en) | 2017-01-09 | 2018-07-12 | Temple University - Of The Commonwealth System Of Higher Education | Methods and compositions for treatment of non-alcoholic steatohepatitis |
| WO2018222583A1 (en) * | 2017-05-30 | 2018-12-06 | Rho Pharmaceuticals, Llc | In-vial deposition of a stable, sterile and crystalline o-acetyl salicylic acid (aspirin) |
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| US10973798B2 (en) * | 2018-12-23 | 2021-04-13 | SRM Institute of Science and Technology | Dispersion of formononetin solid lipid nanoparticles and process for its preparation |
| US11788091B2 (en) | 2019-08-21 | 2023-10-17 | University Of Virginia Patent Foundation | Methods and compositions for diagnosing and treating prostate cancer based on long noncoding RNA overlapping the LCK gene that regulates prostate cancer cell growth |
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| CN114099441A (zh) * | 2021-12-22 | 2022-03-01 | 金河牧星（重庆）生物科技有限公司 | 一种盐酸金霉素干混悬剂及其制备方法和应用 |
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| JPS60150221A (ja) * | 1984-01-14 | 1985-08-07 | Sanee Denki Kk | 磁気ヘツド |
| JPS60258110A (ja) * | 1984-06-05 | 1985-12-20 | Daigo Eiyou Kagaku Kk | 静脈注射可能なプロゲステロン乳化注射液 |
| JPH0774145B2 (ja) * | 1986-12-15 | 1995-08-09 | 株式会社資生堂 | 結晶性薬物含有乳化組成物 |
| HU205861B (en) * | 1986-12-19 | 1992-07-28 | Sandoz Ag | Process for producing hydrosole of pharmaceutically effective material |
| US4879308A (en) * | 1987-08-11 | 1989-11-07 | Lyphomed, Inc. | Aqueous nitroglycerin injection and manufacturing process |
| EP0361928B1 (en) * | 1988-09-29 | 1994-04-27 | Shiseido Company Limited | Emulsified composition |
| ATE94057T1 (de) * | 1988-12-20 | 1993-09-15 | Medicontrol Corp | Durch hitze dehydratisierte emulsionen. |
| US5145684A (en) * | 1991-01-25 | 1992-09-08 | Sterling Drug Inc. | Surface modified drug nanoparticles |
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| IL101387A (en) * | 1992-03-26 | 1999-11-30 | Pharmos Ltd | Emulsion with enhanced topical and/or transdermal systemic effect utilizing submicron oil droplets |
| DE4217842A1 (de) * | 1992-05-29 | 1993-12-02 | Dietl Hans | Calciumantagonisten enthaltende pharmazeutische Zubereitung zur intravenösen und intrakoronaren Applikation sowie Verfahren zu ihrer Herstellung |
| JPH06126143A (ja) * | 1992-10-14 | 1994-05-10 | Mitsubishi Heavy Ind Ltd | 凝集体含有液状混合物の分散方法 |
| AU660852B2 (en) * | 1992-11-25 | 1995-07-06 | Elan Pharma International Limited | Method of grinding pharmaceutical substances |
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-
1994
- 1994-11-11 DE DE4440337A patent/DE4440337A1/de not_active Withdrawn
-
1995
- 1995-11-09 CA CA002205046A patent/CA2205046C/en not_active Expired - Lifetime
- 1995-11-09 EE EE9700217A patent/EE9700217A/xx unknown
- 1995-11-09 EP EP95938439A patent/EP0790821B1/de not_active Expired - Lifetime
- 1995-11-09 JP JP51571196A patent/JP3977418B2/ja not_active Expired - Lifetime
- 1995-11-09 DE DE59510954T patent/DE59510954D1/de not_active Expired - Lifetime
- 1995-11-09 HU HU9702018A patent/HU228097B1/hu unknown
- 1995-11-09 AU AU39827/95A patent/AU714978B2/en not_active Expired
- 1995-11-09 SK SK584-97A patent/SK284541B6/sk not_active IP Right Cessation
- 1995-11-09 AT AT95938439T patent/ATE278387T1/de not_active IP Right Cessation
- 1995-11-09 CN CNB951973010A patent/CN1210018C/zh not_active Expired - Lifetime
- 1995-11-09 KR KR1019970703160A patent/KR100480447B1/ko not_active IP Right Cessation
- 1995-11-09 US US08/836,305 patent/US5858410A/en not_active Expired - Lifetime
- 1995-11-09 DE DE19581305T patent/DE19581305D2/de not_active Ceased
- 1995-11-09 WO PCT/EP1995/004401 patent/WO1996014830A1/de active IP Right Grant
- 1995-11-09 ES ES95938439T patent/ES2229242T3/es not_active Expired - Lifetime
- 1995-11-09 CZ CZ19971426A patent/CZ293253B6/cs not_active IP Right Cessation
- 1995-11-09 PL PL95320085A patent/PL320085A1/xx unknown
-
1997
- 1997-05-09 NO NO19972142A patent/NO323143B1/no not_active IP Right Cessation
- 1997-05-09 FI FI971986A patent/FI119465B/fi not_active IP Right Cessation
- 1997-05-09 MX MX9703399A patent/MX9703399A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI119465B (fi) | 2008-11-28 |
| JPH10508614A (ja) | 1998-08-25 |
| WO1996014830A1 (de) | 1996-05-23 |
| CZ293253B6 (cs) | 2004-03-17 |
| HU228097B1 (en) | 2012-10-29 |
| FI971986A (fi) | 1997-07-08 |
| CA2205046C (en) | 2002-05-14 |
| CZ142697A3 (en) | 1997-10-15 |
| SK284541B6 (sk) | 2005-06-02 |
| HUT77526A (hu) | 1998-05-28 |
| CA2205046A1 (en) | 1996-05-23 |
| CN1210018C (zh) | 2005-07-13 |
| ES2229242T3 (es) | 2005-04-16 |
| KR100480447B1 (ko) | 2005-09-20 |
| NO972142L (no) | 1997-06-26 |
| SK58497A3 (en) | 1997-11-05 |
| KR970706795A (ko) | 1997-12-01 |
| AU714978B2 (en) | 2000-01-13 |
| US5858410A (en) | 1999-01-12 |
| DE4440337A1 (de) | 1996-05-15 |
| FI971986A0 (fi) | 1997-05-09 |
| EP0790821B1 (de) | 2004-10-06 |
| CN1172428A (zh) | 1998-02-04 |
| EP0790821A1 (de) | 1997-08-27 |
| NO972142D0 (no) | 1997-05-09 |
| JP3977418B2 (ja) | 2007-09-19 |
| ATE278387T1 (de) | 2004-10-15 |
| PL320085A1 (en) | 1997-09-15 |
| EE9700217A (et) | 1998-02-16 |
| DE19581305D2 (de) | 1998-11-05 |
| DE59510954D1 (de) | 2004-11-11 |
| AU3982795A (en) | 1996-06-06 |
| MX9703399A (es) | 1998-07-31 |
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| MK1K | Patent expired |