FI971986A - Farmaseuttisia nanosuspensioita lääkeaineen antamiseen systeemeinä, joissa on kasvanut kyllästysliukoisuus ja liukenemisnopeus - Google Patents

Farmaseuttisia nanosuspensioita lääkeaineen antamiseen systeemeinä, joissa on kasvanut kyllästysliukoisuus ja liukenemisnopeus Download PDF

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Publication number
FI971986A
FI971986A FI971986A FI971986A FI971986A FI 971986 A FI971986 A FI 971986A FI 971986 A FI971986 A FI 971986A FI 971986 A FI971986 A FI 971986A FI 971986 A FI971986 A FI 971986A
Authority
FI
Finland
Prior art keywords
pct
active compound
particles
saturation solubility
sec
Prior art date
Application number
FI971986A
Other languages
English (en)
Swedish (sv)
Other versions
FI119465B (fi
FI971986A0 (fi
Inventor
Rainer H Mueller
Robert Becker
Bernd Kruss
Katrin Peters
Original Assignee
Medac Klinische Spezialpraep
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Filing date
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Application filed by Medac Klinische Spezialpraep filed Critical Medac Klinische Spezialpraep
Publication of FI971986A0 publication Critical patent/FI971986A0/fi
Publication of FI971986A publication Critical patent/FI971986A/fi
Application granted granted Critical
Publication of FI119465B publication Critical patent/FI119465B/fi

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B82—NANOTECHNOLOGY
    • B82Y—SPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00—Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dispersion Chemistry (AREA)
  • Dermatology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Emulsifying, Dispersing, Foam-Producing Or Wetting Agents (AREA)
  • Colloid Chemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI971986A 1994-11-11 1997-05-09 Menetelmä lääkesuspension valmistamiseksi FI119465B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE4440337A DE4440337A1 (de) 1994-11-11 1994-11-11 Pharmazeutische Nanosuspensionen zur Arzneistoffapplikation als Systeme mit erhöhter Sättigungslöslichkeit und Lösungsgeschwindigkeit
DE4440337 1994-11-11
EP9504401 1995-11-09
PCT/EP1995/004401 WO1996014830A1 (de) 1994-11-11 1995-11-09 Pharmazeutische nanosuspensionen zur arzneistoffapplikation als systeme mit erhöhter sättigungslöslichkeit und lösungsgeschwindigkeit

Publications (3)

Publication Number Publication Date
FI971986A0 FI971986A0 (fi) 1997-05-09
FI971986A true FI971986A (fi) 1997-07-08
FI119465B FI119465B (fi) 2008-11-28

Family

ID=6533079

Family Applications (1)

Application Number Title Priority Date Filing Date
FI971986A FI119465B (fi) 1994-11-11 1997-05-09 Menetelmä lääkesuspension valmistamiseksi

Country Status (19)

Country Link
US (1) US5858410A (fi)
EP (1) EP0790821B1 (fi)
JP (1) JP3977418B2 (fi)
KR (1) KR100480447B1 (fi)
CN (1) CN1210018C (fi)
AT (1) ATE278387T1 (fi)
AU (1) AU714978B2 (fi)
CA (1) CA2205046C (fi)
CZ (1) CZ293253B6 (fi)
DE (3) DE4440337A1 (fi)
EE (1) EE9700217A (fi)
ES (1) ES2229242T3 (fi)
FI (1) FI119465B (fi)
HU (1) HU228097B1 (fi)
MX (1) MX9703399A (fi)
NO (1) NO323143B1 (fi)
PL (1) PL320085A1 (fi)
SK (1) SK284541B6 (fi)
WO (1) WO1996014830A1 (fi)

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WO1996014830A1 (de) 1996-05-23
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HU228097B1 (en) 2012-10-29
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CN1210018C (zh) 2005-07-13
ES2229242T3 (es) 2005-04-16
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NO972142L (no) 1997-06-26
SK58497A3 (en) 1997-11-05
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US5858410A (en) 1999-01-12
DE4440337A1 (de) 1996-05-15
FI971986A0 (fi) 1997-05-09
EP0790821B1 (de) 2004-10-06
CN1172428A (zh) 1998-02-04
EP0790821A1 (de) 1997-08-27
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ATE278387T1 (de) 2004-10-15
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