NO314783B1 - Farmasoytiske formuleringer inneholdende darifenacin - Google Patents
Farmasoytiske formuleringer inneholdende darifenacin Download PDFInfo
- Publication number
- NO314783B1 NO314783B1 NO19981073A NO981073A NO314783B1 NO 314783 B1 NO314783 B1 NO 314783B1 NO 19981073 A NO19981073 A NO 19981073A NO 981073 A NO981073 A NO 981073A NO 314783 B1 NO314783 B1 NO 314783B1
- Authority
- NO
- Norway
- Prior art keywords
- darifenacin
- pharmaceutically acceptable
- released
- dosage form
- acceptable salt
- Prior art date
Links
- HXGBXQDTNZMWGS-RUZDIDTESA-N darifenacin Chemical compound C=1C=CC=CC=1C([C@H]1CN(CCC=2C=C3CCOC3=CC=2)CC1)(C(=O)N)C1=CC=CC=C1 HXGBXQDTNZMWGS-RUZDIDTESA-N 0.000 title claims description 59
- 229960002677 darifenacin Drugs 0.000 title claims description 56
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- UQAVIASOPREUIT-VQIWEWKSSA-N darifenacin hydrobromide Chemical compound Br.C=1C=CC=CC=1C([C@H]1CN(CCC=2C=C3CCOC3=CC=2)CC1)(C(=O)N)C1=CC=CC=C1 UQAVIASOPREUIT-VQIWEWKSSA-N 0.000 claims description 8
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Classifications
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0031—Rectum, anus
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Inorganic Chemistry (AREA)
- Urology & Nephrology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9518953.6A GB9518953D0 (en) | 1995-09-15 | 1995-09-15 | Pharmaceutical formulations |
| PCT/EP1996/003719 WO1997009980A1 (en) | 1995-09-15 | 1996-08-21 | Pharmaceutical formulations containing darifenacin |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO981073D0 NO981073D0 (no) | 1998-03-11 |
| NO981073L NO981073L (no) | 1998-03-11 |
| NO314783B1 true NO314783B1 (no) | 2003-05-26 |
Family
ID=10780813
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO19981073A NO314783B1 (no) | 1995-09-15 | 1998-03-11 | Farmasoytiske formuleringer inneholdende darifenacin |
| NO2005009C NO2005009I2 (no) | 1995-09-15 | 2005-04-08 | Emselex-darifenacin. Iupac-navn: (S)-2-ä1-Ä2-(2,3 -dihydrobenzofuran-5-yl)etylÜ-3-pyrrolidinylü-2,2-difenylacetamid |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO2005009C NO2005009I2 (no) | 1995-09-15 | 2005-04-08 | Emselex-darifenacin. Iupac-navn: (S)-2-ä1-Ä2-(2,3 -dihydrobenzofuran-5-yl)etylÜ-3-pyrrolidinylü-2,2-difenylacetamid |
Country Status (32)
| Country | Link |
|---|---|
| US (1) | US6106864A (ru) |
| EP (2) | EP1245231B1 (ru) |
| JP (1) | JP3403203B2 (ru) |
| KR (1) | KR100348585B1 (ru) |
| CN (1) | CN1303998C (ru) |
| AR (1) | AR005231A1 (ru) |
| AT (2) | ATE233090T1 (ru) |
| BR (2) | BR9610153A (ru) |
| CA (1) | CA2230314C (ru) |
| CO (1) | CO4750822A1 (ru) |
| CY (3) | CY2468B1 (ru) |
| CZ (1) | CZ294024B6 (ru) |
| DE (4) | DE69626397T2 (ru) |
| DK (2) | DK0850059T3 (ru) |
| EG (1) | EG23826A (ru) |
| ES (2) | ES2188782T3 (ru) |
| FR (1) | FR05C0019I2 (ru) |
| GB (1) | GB9518953D0 (ru) |
| HU (2) | HU227397B1 (ru) |
| IL (1) | IL122746A (ru) |
| LU (1) | LU91163I2 (ru) |
| MY (1) | MY125662A (ru) |
| NL (1) | NL300190I2 (ru) |
| NO (2) | NO314783B1 (ru) |
| NZ (1) | NZ316924A (ru) |
| PL (1) | PL185604B1 (ru) |
| PT (1) | PT1245231E (ru) |
| RU (1) | RU2163803C2 (ru) |
| TR (1) | TR199800461T1 (ru) |
| TW (1) | TW442300B (ru) |
| WO (1) | WO1997009980A1 (ru) |
| ZA (1) | ZA967745B (ru) |
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| US5233053A (en) * | 1989-03-17 | 1993-08-03 | Pfizer Inc. | Pyrrolidine derivatives |
| GB8906166D0 (en) * | 1989-03-17 | 1989-05-04 | Pfizer Ltd | Therapeutic agents |
| PT93637A (pt) * | 1989-04-20 | 1990-11-20 | Procter & Gamble | Metodo para o tratamento de desordens funcionais intestinais/colonicas, especialmente o sindrome de irritacao intestinal |
| GB9400600D0 (en) * | 1994-01-14 | 1994-03-09 | Pfizer Ltd | Treatment of motion seckness |
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