MA50245A - Inhibiteurs allostériques octahydrocyclopenta[c]pyrrole de shp2 - Google Patents

Inhibiteurs allostériques octahydrocyclopenta[c]pyrrole de shp2

Info

Publication number
MA50245A
MA50245A MA050245A MA50245A MA50245A MA 50245 A MA50245 A MA 50245A MA 050245 A MA050245 A MA 050245A MA 50245 A MA50245 A MA 50245A MA 50245 A MA50245 A MA 50245A
Authority
MA
Morocco
Prior art keywords
octahydrocyclopenta
shp2
pyrrole
allosteric inhibitors
allosteric
Prior art date
Application number
MA050245A
Other languages
English (en)
Inventor
Anthony Marfat
Frederick Nelson
Robert VOLKMANN
Panayiotis Zagouras
Original Assignee
Krouzon Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Krouzon Pharmaceuticals Inc filed Critical Krouzon Pharmaceuticals Inc
Publication of MA50245A publication Critical patent/MA50245A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
MA050245A 2017-09-11 2018-09-11 Inhibiteurs allostériques octahydrocyclopenta[c]pyrrole de shp2 MA50245A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201762556713P 2017-09-11 2017-09-11

Publications (1)

Publication Number Publication Date
MA50245A true MA50245A (fr) 2020-07-22

Family

ID=63794616

Family Applications (1)

Application Number Title Priority Date Filing Date
MA050245A MA50245A (fr) 2017-09-11 2018-09-11 Inhibiteurs allostériques octahydrocyclopenta[c]pyrrole de shp2

Country Status (8)

Country Link
US (1) US10435389B2 (fr)
EP (1) EP3681879A1 (fr)
JP (2) JP7447002B2 (fr)
CN (1) CN111201223B (fr)
CA (1) CA3074304A1 (fr)
MA (1) MA50245A (fr)
TW (1) TW201912639A (fr)
WO (1) WO2019051469A1 (fr)

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Also Published As

Publication number Publication date
CA3074304A1 (fr) 2019-03-14
US20190077792A1 (en) 2019-03-14
JP2020535218A (ja) 2020-12-03
TW201912639A (zh) 2019-04-01
CN111201223B (zh) 2024-07-09
JP7447002B2 (ja) 2024-03-11
JP2024059874A (ja) 2024-05-01
US10435389B2 (en) 2019-10-08
CN111201223A (zh) 2020-05-26
WO2019051469A1 (fr) 2019-03-14
EP3681879A1 (fr) 2020-07-22

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