DK3625224T3 - N-substituerede indolderivater - Google Patents

N-substituerede indolderivater Download PDF

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Publication number
DK3625224T3
DK3625224T3 DK18725223.4T DK18725223T DK3625224T3 DK 3625224 T3 DK3625224 T3 DK 3625224T3 DK 18725223 T DK18725223 T DK 18725223T DK 3625224 T3 DK3625224 T3 DK 3625224T3
Authority
DK
Denmark
Prior art keywords
substituted content
derivatives
content derivatives
substituted
content
Prior art date
Application number
DK18725223.4T
Other languages
English (en)
Inventor
Heinz Fretz
Isabelle Lyothier
Julien Pothier
Sylvia Richard-Bildstein
Thierry Sifferlen
Original Assignee
Idorsia Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idorsia Pharmaceuticals Ltd filed Critical Idorsia Pharmaceuticals Ltd
Application granted granted Critical
Publication of DK3625224T3 publication Critical patent/DK3625224T3/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
DK18725223.4T 2017-05-18 2018-05-17 N-substituerede indolderivater DK3625224T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP2017062008 2017-05-18
PCT/EP2018/062865 WO2018210995A1 (en) 2017-05-18 2018-05-17 N-substituted indole derivatives

Publications (1)

Publication Number Publication Date
DK3625224T3 true DK3625224T3 (da) 2021-11-08

Family

ID=62186481

Family Applications (1)

Application Number Title Priority Date Filing Date
DK18725223.4T DK3625224T3 (da) 2017-05-18 2018-05-17 N-substituerede indolderivater

Country Status (32)

Country Link
US (2) US20200069686A1 (da)
EP (1) EP3625224B1 (da)
JP (1) JP7065117B2 (da)
KR (1) KR102650756B1 (da)
CN (1) CN110621666A (da)
AR (1) AR111806A1 (da)
AU (1) AU2018269667B2 (da)
BR (1) BR112019024114A2 (da)
CA (1) CA3063637A1 (da)
CL (1) CL2019003257A1 (da)
CO (1) CO2019010804A2 (da)
CR (1) CR20190567A (da)
CY (1) CY1124528T1 (da)
DK (1) DK3625224T3 (da)
EA (1) EA039630B1 (da)
ES (1) ES2894124T3 (da)
HR (1) HRP20211532T1 (da)
HU (1) HUE056406T2 (da)
IL (1) IL270616B (da)
LT (1) LT3625224T (da)
MA (1) MA49127B1 (da)
MX (1) MX2019013639A (da)
PE (1) PE20191787A1 (da)
PH (1) PH12019502562A1 (da)
PL (1) PL3625224T3 (da)
PT (1) PT3625224T (da)
RS (1) RS62441B1 (da)
SG (1) SG11201908660RA (da)
SI (1) SI3625224T1 (da)
TW (1) TWI768043B (da)
UA (1) UA124748C2 (da)
WO (1) WO2018210995A1 (da)

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US11446298B2 (en) 2017-05-18 2022-09-20 Idorsia Pharmaceuticals Ltd Pyrimidine derivatives
US11325899B2 (en) 2017-05-18 2022-05-10 Idorsia Pharmaceuticals Ltd Benzofurane and benzothiophene derivatives as PGE2 receptor modulators
AR111941A1 (es) 2017-05-18 2019-09-04 Idorsia Pharmaceuticals Ltd Derivados de pirimidina como moduladores del receptor de pge2
WO2021060281A1 (ja) * 2019-09-24 2021-04-01 Ａｇｃ株式会社 プロスタグランジンｅ２レセプターｅｐ２／ｅｐ４デュアルアンタゴニスト
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Also Published As

Publication number Publication date
IL270616B (en) 2022-01-01
WO2018210995A1 (en) 2018-11-22
PH12019502562A1 (en) 2020-07-20
SG11201908660RA (en) 2019-10-30
PE20191787A1 (es) 2019-12-24
MA49127A (fr) 2021-05-26
KR102650756B1 (ko) 2024-03-22
AU2018269667A1 (en) 2019-10-24
US20200069686A1 (en) 2020-03-05
EP3625224A1 (en) 2020-03-25
MX2019013639A (es) 2020-01-21
HRP20211532T1 (hr) 2022-01-07
LT3625224T (lt) 2021-10-25
UA124748C2 (uk) 2021-11-10
CA3063637A1 (en) 2018-11-22
CN110621666A (zh) 2019-12-27
JP7065117B2 (ja) 2022-05-11
US20230165859A1 (en) 2023-06-01
SI3625224T1 (sl) 2021-11-30
KR20200006589A (ko) 2020-01-20
TW201900637A (zh) 2019-01-01
ES2894124T3 (es) 2022-02-11
EA039630B1 (ru) 2022-02-18
BR112019024114A2 (pt) 2020-06-02
JP2020520359A (ja) 2020-07-09
EP3625224B1 (en) 2021-08-04
HUE056406T2 (hu) 2022-02-28
TWI768043B (zh) 2022-06-21
AU2018269667B2 (en) 2022-02-03
CY1124528T1 (el) 2022-07-22
CO2019010804A2 (es) 2019-10-09
EA201992679A1 (ru) 2020-05-06
PT3625224T (pt) 2021-10-06
AR111806A1 (es) 2019-08-21
RS62441B1 (sr) 2021-11-30
CL2019003257A1 (es) 2020-03-27
PL3625224T3 (pl) 2022-01-10
CR20190567A (es) 2020-02-10
MA49127B1 (fr) 2022-05-31

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