NO20065864L - Femleddete heterosykler anvendelige som serinproteaseinhibitorer - Google Patents

Femleddete heterosykler anvendelige som serinproteaseinhibitorer

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Publication number
NO20065864L
NO20065864L NO20065864A NO20065864A NO20065864L NO 20065864 L NO20065864 L NO 20065864L NO 20065864 A NO20065864 A NO 20065864A NO 20065864 A NO20065864 A NO 20065864A NO 20065864 L NO20065864 L NO 20065864L
Authority
NO
Norway
Prior art keywords
factor
formula
compounds
serine protease
protease inhibitors
Prior art date
Application number
NO20065864A
Other languages
English (en)
Norwegian (no)
Inventor
Jon J Hangeland
James R Corte
Mimi L Quan
Joanne M Smallheer
Gregory S Bisacchi
Todd J Friends
Zhong Sun
Karen A Rossi
Cullen L Cavallaro
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35481430&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20065864(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20065864L publication Critical patent/NO20065864L/no

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    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

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KR20080087817A (ko) 2005-12-14 2008-10-01 브리스톨-마이어스 스큅 컴퍼니 인자 ｘｉａ 억제제로서 아릴프로피온아미드,아릴아크릴아미드, 아릴프로핀아미드 또는 아릴메틸우레아유사체

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IL179844A0 (en) 2007-07-04
US10112936B2 (en) 2018-10-30
EP1773786B1 (de) 2017-04-26
EP1773786A2 (de) 2007-04-18
ES2628279T3 (es) 2017-08-02
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WO2005123050A2 (en) 2005-12-29
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US7453002B2 (en) 2008-11-18
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