NO20051566L - PGD2 reseptor antagonister for behandling av inflammatoriske sykdommer - Google Patents

PGD2 reseptor antagonister for behandling av inflammatoriske sykdommer

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Publication number
NO20051566L
NO20051566L NO20051566A NO20051566A NO20051566L NO 20051566 L NO20051566 L NO 20051566L NO 20051566 A NO20051566 A NO 20051566A NO 20051566 A NO20051566 A NO 20051566A NO 20051566 L NO20051566 L NO 20051566L
Authority
NO
Norway
Prior art keywords
treatment
receptor antagonists
inflammatory diseases
pgd2 receptor
compounds
Prior art date
Application number
NO20051566A
Other languages
English (en)
Norwegian (no)
Inventor
Kenneth G Carson
Shomir Ghosh
Amy M Elder
Kevin Sprott
Sean Harrison
Original Assignee
Millennium Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Millennium Pharm Inc filed Critical Millennium Pharm Inc
Publication of NO20051566L publication Critical patent/NO20051566L/no

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/50Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 4
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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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NO20051566A 2002-10-04 2005-03-23 PGD2 reseptor antagonister for behandling av inflammatoriske sykdommer NO20051566L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US41650102P 2002-10-04 2002-10-04
PCT/US2003/031542 WO2004032848A2 (fr) 2002-10-04 2003-10-03 Antagonistes vis-a-vis du recepteur pgd2 pour le traitement de maladies inflammatoires

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NO20051566L true NO20051566L (no) 2005-06-15

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NO20051566A NO20051566L (no) 2002-10-04 2005-03-23 PGD2 reseptor antagonister for behandling av inflammatoriske sykdommer

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US (2) US7211672B2 (fr)
EP (1) EP1556047A4 (fr)
JP (2) JP2006508077A (fr)
KR (1) KR20050055747A (fr)
CN (1) CN100363348C (fr)
AU (1) AU2003277285B2 (fr)
BR (1) BR0315041A (fr)
CA (1) CA2500582A1 (fr)
EA (1) EA011385B1 (fr)
MX (1) MXPA05003456A (fr)
NO (1) NO20051566L (fr)
PL (1) PL376156A1 (fr)
WO (1) WO2004032848A2 (fr)
ZA (1) ZA200502692B (fr)

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US20040082609A1 (en) 2004-04-29
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