ZA200502692B - PGD2 receptor antagonists for the treatment of inflammatory diseases - Google Patents

PGD2 receptor antagonists for the treatment of inflammatory diseases Download PDF

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Publication number
ZA200502692B
ZA200502692B ZA200502692A ZA200502692A ZA200502692B ZA 200502692 B ZA200502692 B ZA 200502692B ZA 200502692 A ZA200502692 A ZA 200502692A ZA 200502692 A ZA200502692 A ZA 200502692A ZA 200502692 B ZA200502692 B ZA 200502692B
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South Africa
Prior art keywords
phenyl
methyl
tetrahydro
group
quinolinyl
Prior art date
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ZA200502692A
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English (en)
Inventor
Ghosh Shomir
Amy M Elder
Kennth G Carson
Sprott Kevin
Harrison Sean
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Millennium Pharm Inc
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Publication of ZA200502692B publication Critical patent/ZA200502692B/en

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    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/50—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 4
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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ZA200502692A 2002-10-04 2005-04-04 PGD2 receptor antagonists for the treatment of inflammatory diseases ZA200502692B (en)

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US (2) US7211672B2 (fr)
EP (1) EP1556047A4 (fr)
JP (2) JP2006508077A (fr)
KR (1) KR20050055747A (fr)
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