MA45588A - Formes solides d'un stimulateur de la gcs - Google Patents

Formes solides d'un stimulateur de la gcs

Info

Publication number
MA45588A
MA45588A MA045588A MA45588A MA45588A MA 45588 A MA45588 A MA 45588A MA 045588 A MA045588 A MA 045588A MA 45588 A MA45588 A MA 45588A MA 45588 A MA45588 A MA 45588A
Authority
MA
Morocco
Prior art keywords
gcs
stimulator
solid forms
solid
forms
Prior art date
Application number
MA045588A
Other languages
English (en)
Inventor
Ahmad Hashash
Robert C Livingston
Kwame Wiredu Nti-Addae
Vasu Sethuraman
Song Xue
Original Assignee
Ironwood Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ironwood Pharmaceuticals Inc filed Critical Ironwood Pharmaceuticals Inc
Publication of MA45588A publication Critical patent/MA45588A/fr

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
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    • C07B2200/13Crystalline forms, e.g. polymorphs
MA045588A 2016-07-07 2017-07-06 Formes solides d'un stimulateur de la gcs MA45588A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201662359466P 2016-07-07 2016-07-07

Publications (1)

Publication Number Publication Date
MA45588A true MA45588A (fr) 2019-05-15

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Application Number Title Priority Date Filing Date
MA045588A MA45588A (fr) 2016-07-07 2017-07-06 Formes solides d'un stimulateur de la gcs

Country Status (16)

Country Link
US (3) US10889577B2 (fr)
EP (1) EP3481820B1 (fr)
JP (2) JP2019524710A (fr)
KR (2) KR20230074840A (fr)
CN (1) CN109563087A (fr)
AU (1) AU2017292818B2 (fr)
BR (1) BR112019000293A2 (fr)
CA (1) CA3029333A1 (fr)
CL (1) CL2019000018A1 (fr)
EA (1) EA039753B1 (fr)
IL (1) IL263996B2 (fr)
JO (1) JOP20180127A1 (fr)
MA (1) MA45588A (fr)
MX (2) MX2019000115A (fr)
TW (1) TWI774683B (fr)
WO (1) WO2018009609A1 (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG10202100168XA (en) * 2016-07-07 2021-02-25 Cyclerion Therapeutics Inc Novel processes for preparation of soluble guanylate cyclase stimulators
EP3481820B1 (fr) * 2016-07-07 2023-10-18 Cyclerion Therapeutics, Inc. Formes solides d'un stimulateur de la gcs
MA45603A (fr) * 2016-07-07 2019-05-15 Ironwood Pharmaceuticals Inc Nouveaux procédés de préparation de stimulateurs de la guanylate cyclase soluble
WO2019161534A1 (fr) * 2018-02-22 2019-08-29 Ironwood Pharmaceuticals, Inc. Nouveaux procédés et intermédiaires pour la préparation de stimulateurs de guanylate cyclase soluble
CN109503574B (zh) * 2018-12-14 2021-07-06 中国人民解放军军事科学院军事医学研究院 抗肺动脉高压药物sgc-003的多晶型晶体变体及其制备方法
CN110862424A (zh) * 2019-12-03 2020-03-06 海南顿斯医药科技有限公司 一种硫酸阿米卡星化合物
WO2023009710A1 (fr) * 2021-07-28 2023-02-02 Cyclerion Therapeutics, Inc. Traitement de hfpef chez des femmes post-ménopausées avec un stimulateur sgc
CN114199812A (zh) * 2021-12-28 2022-03-18 南通联亚药业有限公司 一种盐酸美金刚缓释制剂中盐酸美金刚的检测方法

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TW201805283A (zh) 2018-02-16
BR112019000293A2 (pt) 2019-04-16
US10889577B2 (en) 2021-01-12
IL263996A (en) 2019-01-31
AU2017292818A1 (en) 2019-01-31
US20190169179A1 (en) 2019-06-06
CA3029333A1 (fr) 2018-01-11
IL263996B2 (en) 2024-03-01
EA039753B1 (ru) 2022-03-10
KR20230074840A (ko) 2023-05-31
IL263996B1 (en) 2023-11-01
MX2022001565A (es) 2022-03-02
EP3481820A1 (fr) 2019-05-15
KR20190025989A (ko) 2019-03-12
WO2018009609A1 (fr) 2018-01-11
CL2019000018A1 (es) 2019-05-03
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AU2017292818B2 (en) 2021-10-21
MX2019000115A (es) 2019-04-22
JP2019524710A (ja) 2019-09-05
US20210188830A1 (en) 2021-06-24
US11572358B2 (en) 2023-02-07
US20240059683A1 (en) 2024-02-22
EP3481820B1 (fr) 2023-10-18
JOP20180127A1 (ar) 2019-01-30

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