NO20043726L - Heteroarylforbindelser anvendelige som inhibitorer av GSK-3 - Google Patents

Heteroarylforbindelser anvendelige som inhibitorer av GSK-3

Info

Publication number
NO20043726L
NO20043726L NO20043726A NO20043726A NO20043726L NO 20043726 L NO20043726 L NO 20043726L NO 20043726 A NO20043726 A NO 20043726A NO 20043726 A NO20043726 A NO 20043726A NO 20043726 L NO20043726 L NO 20043726L
Authority
NO
Norway
Prior art keywords
gsk
inhibitors
compounds useful
heteroaryl compounds
heteroaryl
Prior art date
Application number
NO20043726A
Other languages
English (en)
Norwegian (no)
Inventor
Michael J Arnost
Scott L Harbeson
Jeremy Green
Viadimir Savic
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of NO20043726L publication Critical patent/NO20043726L/no

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245—Oxadiazoles
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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  • Organic Chemistry (AREA)
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NO20043726A 2002-02-06 2004-09-06 Heteroarylforbindelser anvendelige som inhibitorer av GSK-3 NO20043726L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35484302P 2002-02-06 2002-02-06
PCT/US2003/003655 WO2003066629A2 (en) 2002-02-06 2003-02-06 Heteroaryl compounds useful as inhibitors of gsk-3

Publications (1)

Publication Number Publication Date
NO20043726L true NO20043726L (no) 2004-11-08

Family

ID=27734431

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20043726A NO20043726L (no) 2002-02-06 2004-09-06 Heteroarylforbindelser anvendelige som inhibitorer av GSK-3

Country Status (13)

Country Link
US (2) US20040034037A1 (ja)
EP (2) EP2322521B1 (ja)
JP (2) JP4656838B2 (ja)
KR (1) KR20040084896A (ja)
AU (1) AU2003215087B2 (ja)
CA (1) CA2475633C (ja)
ES (1) ES2437391T3 (ja)
MX (1) MXPA04007697A (ja)
NO (1) NO20043726L (ja)
PL (1) PL372198A1 (ja)
RU (1) RU2004126671A (ja)
SG (1) SG159380A1 (ja)
WO (1) WO2003066629A2 (ja)

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