NO171680C - Analogifremgangsmaate for fremstilling av terapeutisk aktiv morfolinoethylester av mycofenolsyre og derivater derav - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktiv morfolinoethylester av mycofenolsyre og derivater derav

Info

Publication number
NO171680C
NO171680C NO875240A NO875240A NO171680C NO 171680 C NO171680 C NO 171680C NO 875240 A NO875240 A NO 875240A NO 875240 A NO875240 A NO 875240A NO 171680 C NO171680 C NO 171680C
Authority
NO
Norway
Prior art keywords
morpholinoethylesters
derivatives
preparation
mycophenolic acid
therapeutic active
Prior art date
Application number
NO875240A
Other languages
English (en)
Norwegian (no)
Other versions
NO875240L (no
NO171680B (no
NO875240D0 (no
Inventor
Peter H Nelson
Chee-Liang Leo Gu
Anthony C Allison
Elsie M Eugui
William A Lee
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21733252&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO171680(C) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of NO875240D0 publication Critical patent/NO875240D0/no
Publication of NO875240L publication Critical patent/NO875240L/no
Publication of NO171680B publication Critical patent/NO171680B/no
Publication of NO171680C publication Critical patent/NO171680C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Furan Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Saccharide Compounds (AREA)
NO875240A 1987-01-30 1987-12-15 Analogifremgangsmaate for fremstilling av terapeutisk aktiv morfolinoethylester av mycofenolsyre og derivater derav NO171680C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/008,717 US4753935A (en) 1987-01-30 1987-01-30 Morpholinoethylesters of mycophenolic acid and pharmaceutical compositions

Publications (4)

Publication Number Publication Date
NO875240D0 NO875240D0 (no) 1987-12-15
NO875240L NO875240L (no) 1988-08-01
NO171680B NO171680B (no) 1993-01-11
NO171680C true NO171680C (no) 1993-04-21

Family

ID=21733252

Family Applications (2)

Application Number Title Priority Date Filing Date
NO875240A NO171680C (no) 1987-01-30 1987-12-15 Analogifremgangsmaate for fremstilling av terapeutisk aktiv morfolinoethylester av mycofenolsyre og derivater derav
NO1997007C NO1997007I1 (no) 1987-01-30 1997-07-01 Mykofenolatmofetil eller et farmasøytisk akseptabelt salt derav

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO1997007C NO1997007I1 (no) 1987-01-30 1997-07-01 Mykofenolatmofetil eller et farmasøytisk akseptabelt salt derav

Country Status (26)

Country Link
US (7) US4753935A (fi)
EP (1) EP0281713B1 (fi)
JP (1) JPS63188672A (fi)
KR (1) KR940003758B1 (fi)
AT (1) ATE68180T1 (fi)
AU (1) AU599728B2 (fi)
CA (1) CA1333285C (fi)
DE (2) DE3773660D1 (fi)
DK (1) DK166675B1 (fi)
ES (1) ES2038190T3 (fi)
FI (1) FI85141C (fi)
GE (1) GEP20094816B (fi)
GR (1) GR3002866T3 (fi)
HK (1) HK125893A (fi)
HU (2) HU201927B (fi)
IE (1) IE60750B1 (fi)
IL (1) IL84833A (fi)
LU (1) LU88795I2 (fi)
LV (1) LV5748B4 (fi)
MX (1) MX9203163A (fi)
NL (1) NL960019I2 (fi)
NO (2) NO171680C (fi)
NZ (1) NZ222922A (fi)
PH (1) PH23819A (fi)
PT (1) PT86343B (fi)
ZA (1) ZA879414B (fi)

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CN102952105A (zh) * 2011-08-26 2013-03-06 中国科学院上海药物研究所 一类霉酚酸衍生物、其制备方法和用途
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US8669281B1 (en) 2013-03-14 2014-03-11 Alkermes Pharma Ireland Limited Prodrugs of fumarates and their use in treating various diseases
CA2906580C (en) 2013-03-14 2019-10-29 Alkermes Pharma Ireland Limited Prodrugs of fumarates and their use in treating various diseases
US10369133B2 (en) 2013-07-23 2019-08-06 The University Of Tennessee Research Foundation Immunosuppressive compounds and therapeutics
CA2935905C (en) * 2014-01-10 2019-02-05 Fujifilm Corporation Method and apparatus for predicting effective dose or sensitivity of 5-hydroxy-1h-imidazole-4-carboxamide, method for determining amount of xanthosine monophosphate, and treatmentagent and method for treating myelodysplastic syndrome
WO2015127450A1 (en) 2014-02-24 2015-08-27 Alkermes Pharma Ireland Limited Sulfonamide and sulfinamide prodrugs of fumarates and their use in treating various diseases
US10603299B2 (en) 2016-06-02 2020-03-31 Steven Baranowitz Prevention and treatment of viral infections
WO2017210262A1 (en) 2016-06-02 2017-12-07 Steven Baranowitz Prevention and treatment of viral infections
US12011429B2 (en) 2016-06-02 2024-06-18 Steven Baranowitz Prevention and treatment of viral infections
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US10835489B2 (en) * 2018-03-09 2020-11-17 University Of Saskatchewan Modified release formulations of mycophenolate mofetil
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CN112121173B (zh) * 2020-08-22 2022-05-06 浙江大学 脂肪酸修饰的免疫抑制剂mmf及fk506纳米制剂及其制备方法和应用
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Also Published As

Publication number Publication date
NO875240L (no) 1988-08-01
US4753935A (en) 1988-06-28
NO171680B (no) 1993-01-11
DE3773660D1 (de) 1991-11-14
EP0281713B1 (en) 1991-10-09
IL84833A0 (en) 1988-06-30
US4808592A (en) 1989-02-28
AU599728B2 (en) 1990-07-26
PH23819A (en) 1989-11-23
CA1333285C (en) 1994-11-29
IE873397L (en) 1988-07-30
FI875502A0 (fi) 1987-12-15
DE19675020I2 (de) 2002-11-07
LU88795I2 (fr) 1996-11-05
HU201927B (en) 1991-01-28
KR940003758B1 (ko) 1994-04-30
EP0281713A1 (en) 1988-09-14
IE60750B1 (en) 1994-08-10
LV5748A4 (lv) 1996-10-20
ATE68180T1 (de) 1991-10-15
US4952579A (en) 1990-08-28
DK658787D0 (da) 1987-12-15
FI85141B (fi) 1991-11-29
IL84833A (en) 1992-03-29
MX9203163A (es) 1992-07-31
FI875502A (fi) 1988-07-31
LV5748B4 (lv) 1997-02-20
NL960019I1 (nl) 1996-10-01
GR3002866T3 (en) 1993-01-25
FI85141C (fi) 1992-03-10
US4992467A (en) 1991-02-12
NO875240D0 (no) 1987-12-15
US4786637A (en) 1988-11-22
KR880009016A (ko) 1988-09-13
US4868153A (en) 1989-09-19
NO1997007I1 (no) 1997-07-01
HK125893A (en) 1993-11-19
AU8254087A (en) 1988-08-04
HUT47567A (en) 1989-03-28
JPS63188672A (ja) 1988-08-04
DK166675B1 (da) 1993-06-28
NZ222922A (en) 1990-09-26
DK658787A (da) 1988-07-31
GEP20094816B (en) 2009-11-10
PT86343B (pt) 1991-02-08
US4948793A (en) 1990-08-14
ES2038190T3 (es) 1993-07-16
HU210350A9 (en) 1995-03-28
NL960019I2 (nl) 1997-06-02
PT86343A (en) 1988-01-01
JPH0571591B2 (fi) 1993-10-07
ZA879414B (en) 1989-08-30

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