NL300348I2 - 42-rapamycine-hydroxyester, werkwijze voor de bereiding daarvan en farmaceutische preparaten die de ester bevatten - Google Patents

42-rapamycine-hydroxyester, werkwijze voor de bereiding daarvan en farmaceutische preparaten die de ester bevatten

Info

Publication number
NL300348I2
NL300348I2 NL300348C NL300348C NL300348I2 NL 300348 I2 NL300348 I2 NL 300348I2 NL 300348 C NL300348 C NL 300348C NL 300348 C NL300348 C NL 300348C NL 300348 I2 NL300348 I2 NL 300348I2
Authority
NL
Netherlands
Prior art keywords
alkyl
hydrogen
alkynyl
alkenyl
tri
Prior art date
Application number
NL300348C
Other languages
English (en)
Other versions
NL300348I1 (nl
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22860462&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NL300348(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of NL300348I1 publication Critical patent/NL300348I1/nl
Publication of NL300348I2 publication Critical patent/NL300348I2/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Vascular Medicine (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Domestic Plumbing Installations (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NL300348C 1994-04-18 2008-05-15 42-rapamycine-hydroxyester, werkwijze voor de bereiding daarvan en farmaceutische preparaten die de ester bevatten NL300348I2 (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/229,261 US5362718A (en) 1994-04-18 1994-04-18 Rapamycin hydroxyesters
PCT/US1995/004603 WO1995028406A1 (en) 1994-04-18 1995-04-14 Rapamycin hydroxyesters, process for their preparation and pharmaceutical compositions containing them

Publications (2)

Publication Number Publication Date
NL300348I1 NL300348I1 (nl) 2008-07-01
NL300348I2 true NL300348I2 (nl) 2008-09-01

Family

ID=22860462

Family Applications (1)

Application Number Title Priority Date Filing Date
NL300348C NL300348I2 (nl) 1994-04-18 2008-05-15 42-rapamycine-hydroxyester, werkwijze voor de bereiding daarvan en farmaceutische preparaten die de ester bevatten

Country Status (30)

Country Link
US (2) US5362718A (nl)
EP (3) EP0763039B3 (nl)
JP (1) JP3725901B2 (nl)
KR (1) KR100330800B1 (nl)
CN (1) CN1059905C (nl)
AT (3) ATE537176T1 (nl)
BR (1) BR9507323A (nl)
CA (1) CA2187024C (nl)
CY (2) CY2378B1 (nl)
CZ (1) CZ284567B6 (nl)
DE (3) DE69535363T2 (nl)
DK (2) DK1266899T3 (nl)
ES (3) ES2191704T7 (nl)
FR (1) FR08C0018I2 (nl)
HK (2) HK1048816B (nl)
HU (1) HU225915B1 (nl)
IL (1) IL113179A (nl)
LU (1) LU91438I2 (nl)
LV (1) LV13038B (nl)
MX (1) MX9604694A (nl)
NL (1) NL300348I2 (nl)
NZ (1) NZ283988A (nl)
PL (1) PL183178B1 (nl)
PT (2) PT763039E (nl)
RU (1) RU2134267C1 (nl)
SI (2) SI0763039T1 (nl)
SK (1) SK281787B6 (nl)
TW (1) TW275631B (nl)
WO (1) WO1995028406A1 (nl)
ZA (1) ZA953090B (nl)

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