NL1015744C2 - Werkwijze voor de bereiding van 2-(6-gesubstitueerde-1,3-dioxan-4-yl) azijnzuurderivaten. - Google Patents

Werkwijze voor de bereiding van 2-(6-gesubstitueerde-1,3-dioxan-4-yl) azijnzuurderivaten. Download PDF

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Publication number
NL1015744C2
NL1015744C2 NL1015744A NL1015744A NL1015744C2 NL 1015744 C2 NL1015744 C2 NL 1015744C2 NL 1015744 A NL1015744 A NL 1015744A NL 1015744 A NL1015744 A NL 1015744A NL 1015744 C2 NL1015744 C2 NL 1015744C2
Authority
NL
Netherlands
Prior art keywords
formula
substituted
acetic acid
dioxan
group
Prior art date
Application number
NL1015744A
Other languages
English (en)
Dutch (nl)
Inventor
Daniel Mink
Jacob Hermanus Matthe Kooistra
Hubertus Josephus Mari Zeegers
Joannes Maria Cornelis Mulders
Original Assignee
Dsm Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to NL1015744A priority Critical patent/NL1015744C2/nl
Application filed by Dsm Nv filed Critical Dsm Nv
Priority to AT01953373T priority patent/ATE340790T1/de
Priority to CN2007101118797A priority patent/CN101081842B/zh
Priority to CZ20030163A priority patent/CZ302718B6/cs
Priority to BR0112535-4A priority patent/BR0112535A/pt
Priority to ES01953373T priority patent/ES2272506T3/es
Priority to CNB2005100657442A priority patent/CN100378091C/zh
Priority to PCT/NL2001/000535 priority patent/WO2002006266A1/en
Priority to KR1020087019878A priority patent/KR20080078925A/ko
Priority to CA002415963A priority patent/CA2415963C/en
Priority to KR1020077027471A priority patent/KR20070121063A/ko
Priority to DE60123444T priority patent/DE60123444T2/de
Priority to IL15398001A priority patent/IL153980A0/xx
Priority to DK01953373T priority patent/DK1317440T3/da
Priority to NZ523703A priority patent/NZ523703A/en
Priority to SK123-2010A priority patent/SK287756B6/sk
Priority to PL359332A priority patent/PL207115B1/pl
Priority to ES06010837T priority patent/ES2387313T3/es
Priority to EP01953373A priority patent/EP1317440B1/en
Priority to HU0303166A priority patent/HUP0303166A3/hu
Priority to EP06010837A priority patent/EP1700854B1/en
Priority to PT01953373T priority patent/PT1317440E/pt
Priority to US10/333,351 priority patent/US6870059B2/en
Priority to MXPA03000498A priority patent/MXPA03000498A/es
Priority to KR1020027017684A priority patent/KR100865016B1/ko
Priority to CN01812999A priority patent/CN1443183A/zh
Priority to AU2001275830A priority patent/AU2001275830B2/en
Priority to AU7583001A priority patent/AU7583001A/xx
Priority to SK35-2003A priority patent/SK287755B6/sk
Priority to EEP200300024A priority patent/EE200300024A/xx
Priority to RU2003104825/04A priority patent/RU2266903C2/ru
Priority to JP2002512170A priority patent/JP5006499B2/ja
Priority to UA2003010456A priority patent/UA77944C2/uk
Publication of NL1015744C2 publication Critical patent/NL1015744C2/nl
Application granted granted Critical
Priority to NO20030025A priority patent/NO328935B1/no
Priority to IS6680A priority patent/IS2386B/is
Priority to IL153980A priority patent/IL153980A/en
Priority to ZA200300478A priority patent/ZA200300478B/en
Priority to US11/053,090 priority patent/US7642363B2/en
Priority to IL177824A priority patent/IL177824A0/en
Priority to CY20061101848T priority patent/CY1105881T1/el
Priority to HK07102328.2A priority patent/HK1097260A1/xx
Priority to IS8690A priority patent/IS8690A/is
Priority to US12/625,156 priority patent/US7989643B2/en
Priority to US13/166,607 priority patent/US20110251406A1/en
Priority to JP2011267056A priority patent/JP2012111757A/ja

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/30—Oxygen atoms, e.g. delta-lactones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/04—1,3-Dioxanes; Hydrogenated 1,3-dioxanes
    • C07D319/06—1,3-Dioxanes; Hydrogenated 1,3-dioxanes not condensed with other rings
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10T—TECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
    • Y10T428/00—Stock material or miscellaneous articles
    • Y10T428/29—Coated or structually defined flake, particle, cell, strand, strand portion, rod, filament, macroscopic fiber or mass thereof
    • Y10T428/2982—Particulate matter [e.g., sphere, flake, etc.]

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
NL1015744A 2000-07-19 2000-07-19 Werkwijze voor de bereiding van 2-(6-gesubstitueerde-1,3-dioxan-4-yl) azijnzuurderivaten. NL1015744C2 (nl)

Priority Applications (45)

Application Number Priority Date Filing Date Title
NL1015744A NL1015744C2 (nl) 2000-07-19 2000-07-19 Werkwijze voor de bereiding van 2-(6-gesubstitueerde-1,3-dioxan-4-yl) azijnzuurderivaten.
ES06010837T ES2387313T3 (es) 2000-07-19 2001-07-12 Intermedios para la preparación de derivados de ácido 2-(6-sustituido-1,3-dioxan-4-il)acético
CZ20030163A CZ302718B6 (cs) 2000-07-19 2001-07-12 Zpusob prípravy derivátu 2-(6-substituované-1,3-dioxan-4-yl)octové kyseliny
BR0112535-4A BR0112535A (pt) 2000-07-19 2001-07-12 Processo para a preparação de derivados de ácido 2-(6-substituìdo-1,3-dioxana-4-il)acético
ES01953373T ES2272506T3 (es) 2000-07-19 2001-07-12 Procedimiento para la preparacion de derivados de acido 2-(6-sustituido-1,3-dioxan-4-il)acetico.
CNB2005100657442A CN100378091C (zh) 2000-07-19 2001-07-12 2－（6－取代的1，3－二烷－4－基）乙酸衍生物的制备方法
PCT/NL2001/000535 WO2002006266A1 (en) 2000-07-19 2001-07-12 Process for the preparation of 2-(6-substituted-1,3-dioxane-4-yl)acetic acid derivatives
KR1020087019878A KR20080078925A (ko) 2000-07-19 2001-07-12 2-(6-치환-1,3-디옥산-4-일)아세트산 유도체
CA002415963A CA2415963C (en) 2000-07-19 2001-07-12 Process for the preparation of 2-(6-substituted-1,3-dioxane-4-yl)acetic acid derivatives
KR1020077027471A KR20070121063A (ko) 2000-07-19 2001-07-12 2-(6-치환-1,3-디옥산-4-일)아세트산 유도체의 제조위한개시 화합물
DE60123444T DE60123444T2 (de) 2000-07-19 2001-07-12 Verfahren zu herstellung von 2-(6-substituierte-1,3-dioxan-4-yl)essigsäurederivate
IL15398001A IL153980A0 (en) 2000-07-19 2001-07-12 Process for the preparation of 2-(6-substituted-1,3-dioxane-4-yl) acetic acid derivatives
DK01953373T DK1317440T3 (da) 2000-07-19 2001-07-12 Fremgangsmåde til fremstilling af 2- (6-substitueret 1,3-dioxan-4yl) eddikesyrederivater
NZ523703A NZ523703A (en) 2000-07-19 2001-07-12 Process for the preparation of 2-(6-substituted-1,3-dioxane-4-yl)acetic acid derivatives
SK123-2010A SK287756B6 (sk) 2000-07-19 2001-07-12 Deriváty 2-(6-substituovanej-1,3-dioxán-4-yl)octovej kyseliny, soli týchto derivátov a východiskové produkty použité pri spôsobe výroby týchto derivátov
PL359332A PL207115B1 (pl) 2000-07-19 2001-07-12 Sposób wytwarzania pochodnych kwasu 2-(6-podstawiony-1,3-dioksan-4-ylo)octowego
CN01812999A CN1443183A (zh) 2000-07-19 2001-07-12 2－(6－取代的1,3－二噁烷－4－基)乙酸衍生物的制备方法
CN2007101118797A CN101081842B (zh) 2000-07-19 2001-07-12 2-(6-取代的1,3-二噁烷-4-基)乙酸衍生物的制备方法
HU0303166A HUP0303166A3 (en) 2000-07-19 2001-07-12 Process for the preparation of 2-(6-substituted-1,3-dioxane-4-yl)acetic acid derivatives
EP06010837A EP1700854B1 (en) 2000-07-19 2001-07-12 Intermediates for the preparation of 2-(6-substituted-1,3-dioxane-4-yl) acetic acid derivatives
PT01953373T PT1317440E (pt) 2000-07-19 2001-07-12 Processo para a preparação de derivados do ácido 2- ( 6- substituídos-1,3- dioxano-4-il ) acético
US10/333,351 US6870059B2 (en) 2000-07-19 2001-07-12 Process for the preparation of 2-(6-substituted-1,-3-dioxane-4-yl)acetic acid derivatives
AT01953373T ATE340790T1 (de) 2000-07-19 2001-07-12 Verfahren zu herstellung von 2-(6-substituierte-1,3-dioxan-4-yl)essigsäurede ivate
EP01953373A EP1317440B1 (en) 2000-07-19 2001-07-12 Process for the preparation of 2-(6-substituted-1,3-dioxane-4-yl)acetic acid derivatives
MXPA03000498A MXPA03000498A (es) 2000-07-19 2001-07-12 Procedimiento para la preparacion de derivados de acido 2-(6-sustituido-1,3-dioxan-4-il)acetico.
AU2001275830A AU2001275830B2 (en) 2000-07-19 2001-07-12 Process for the preparation of 2-(6-substituted-1,3-dioxane-4-yl)acetic acid derivatives
AU7583001A AU7583001A (en) 2000-07-19 2001-07-12 Process for the preparation of 2-(6-substituted-1,3-dioxane-4-yl)acetic acid derivatives
SK35-2003A SK287755B6 (sk) 2000-07-19 2001-07-12 Spôsob prípravy derivátov 2-(6-substituovaných-1,3-dioxán-4- yl)octovej kyseliny
EEP200300024A EE200300024A (et) 2000-07-19 2001-07-12 Meetod 2-(6-asendatud-1,3-dioksaan-4-üül)etaanhappe derivaadi valmistamiseks, lähteühend ning lõppsaadused
RU2003104825/04A RU2266903C2 (ru) 2000-07-19 2001-07-12 Способ получения производных 2-(6-замещенной-1,3-диоксан-4-ил)уксусной кислоты
JP2002512170A JP5006499B2 (ja) 2000-07-19 2001-07-12 ２−（６−置換−１，３−ジオキサン−４−イル）酢酸誘導体の製造法
KR1020027017684A KR100865016B1 (ko) 2000-07-19 2001-07-12 2-(6-치환-1,3-디옥산-4-일)아세트산 유도체의 제조방법
UA2003010456A UA77944C2 (en) 2000-07-19 2001-12-07 Processes for preparation of derivatives of 2-(6-substituted-1,3-dioxan-4-yl) acetic acid, these derivatives and intermediary compound
NO20030025A NO328935B1 (no) 2000-07-19 2003-01-03 Fremgangsmate ved fremstillingen av 2-(6-substituerte-1,3-dioksan-4-yl)eddiksyrederivater
IS6680A IS2386B (is) 2000-07-19 2003-01-15 Aðferð til að framleiða 2-(6-útskiptar-1,3-díoxan-4-ýl)ediksýruafleiður
IL153980A IL153980A (en) 2000-07-19 2003-01-16 Process for the preparation of a history of 2- (6-converted3,1-dioxane-4-il) Acetic acid
ZA200300478A ZA200300478B (en) 2000-07-19 2003-01-17 Process for the preparation of 2-(6-substituted-1,3-dioxane-4-yl)acetic acid derivatives.
US11/053,090 US7642363B2 (en) 2000-07-19 2005-02-07 Process for the preparation of 2-(6-substituted-1,3-dioxane-4-YL) acetic acid derivatives
IL177824A IL177824A0 (en) 2000-07-19 2006-08-31 Process for the preparation of 2-(6-substituted-1,3-dioxane-4-yl) acetic acid derivatives
CY20061101848T CY1105881T1 (el) 2000-07-19 2006-12-21 Διαδικασια για την παρασκευη παραγωγων 2-(6-υποκατεστημενου-1,3-διοξανο-4υλ)οξικου οξεως
HK07102328.2A HK1097260A1 (en) 2000-07-19 2007-03-01 Intermediates for the preparation of 2-(6-substituted-1,3-dioxane-4-yl) acetic acid derivatives
IS8690A IS8690A (is) 2000-07-19 2007-11-15 Aðferð til að framleiða 2- (6-útskiptar-1,3-díoxan-4-ýl)ediksýruafleiður
US12/625,156 US7989643B2 (en) 2000-07-19 2009-11-24 Process for the preparation of 2-(6-substituted-1,3-dioxane-4-yl)acetic acid derivatives
US13/166,607 US20110251406A1 (en) 2000-07-19 2011-06-22 Process for the preparation of 2-(6-substituted-1,-3-dioxane-4-yl) acetic acid derivatives
JP2011267056A JP2012111757A (ja) 2000-07-19 2011-12-06 ２−（６−置換−１，３−ジオキサン−４−イル）酢酸誘導体およびその製造中間体

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
NL1015744A NL1015744C2 (nl) 2000-07-19 2000-07-19 Werkwijze voor de bereiding van 2-(6-gesubstitueerde-1,3-dioxan-4-yl) azijnzuurderivaten.
NL1015744 2000-07-19

Publications (1)

Publication Number Publication Date
NL1015744C2 true NL1015744C2 (nl) 2002-01-22

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
NL1015744A NL1015744C2 (nl) 2000-07-19 2000-07-19 Werkwijze voor de bereiding van 2-(6-gesubstitueerde-1,3-dioxan-4-yl) azijnzuurderivaten.

Country Status (30)

Country Link
US (4) US6870059B2 (da)
EP (2) EP1700854B1 (da)
JP (2) JP5006499B2 (da)
KR (3) KR20070121063A (da)
CN (3) CN1443183A (da)
AT (1) ATE340790T1 (da)
AU (2) AU7583001A (da)
BR (1) BR0112535A (da)
CA (1) CA2415963C (da)
CY (1) CY1105881T1 (da)
CZ (1) CZ302718B6 (da)
DE (1) DE60123444T2 (da)
DK (1) DK1317440T3 (da)
EE (1) EE200300024A (da)
ES (2) ES2272506T3 (da)
HK (1) HK1097260A1 (da)
HU (1) HUP0303166A3 (da)
IL (3) IL153980A0 (da)
IS (2) IS2386B (da)
MX (1) MXPA03000498A (da)
NL (1) NL1015744C2 (da)
NO (1) NO328935B1 (da)
NZ (1) NZ523703A (da)
PL (1) PL207115B1 (da)
PT (1) PT1317440E (da)
RU (1) RU2266903C2 (da)
SK (2) SK287756B6 (da)
UA (1) UA77944C2 (da)
WO (1) WO2002006266A1 (da)
ZA (1) ZA200300478B (da)

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EP2614057B1 (en) 2010-09-09 2015-10-21 DSM Sinochem Pharmaceuticals Netherlands B.V. Salts of 7-amino-3,5-dihydroxyheptanoic acid esters
US20130178636A1 (en) 2010-09-16 2013-07-11 Dsm Sinochem Pharmaceuticals Netherlands B.V. Esters of hexanoic acids as intermediates for the preparation of atorvastatin
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HUE030590T2 (en) 2011-01-18 2017-05-29 Dsm Sinochem Pharm Nl Bv Process for the production of diol sulfones
EP2665723B1 (en) 2011-01-18 2015-07-22 DSM Sinochem Pharmaceuticals Netherlands B.V. Process for the preparation of statins in the presence of base
MX359424B (es) 2011-12-09 2018-09-12 Dsm Sinochem Pharm Nl Bv Proceso para la preparación de un precursor de estatina.
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JP6065862B2 (ja) * 2013-04-10 2017-01-25 信越化学工業株式会社 パターン形成方法、レジスト組成物、高分子化合物及び単量体
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