MX375476B - Composición farmacéutica que comprende empagliflozina, métodos para tratamiento y sus usos. - Google Patents

Composición farmacéutica que comprende empagliflozina, métodos para tratamiento y sus usos.

Info

Publication number
MX375476B
MX375476B MX2015013939A MX2015013939A MX375476B MX 375476 B MX375476 B MX 375476B MX 2015013939 A MX2015013939 A MX 2015013939A MX 2015013939 A MX2015013939 A MX 2015013939A MX 375476 B MX375476 B MX 375476B
Authority
MX
Mexico
Prior art keywords
empagliflozin
therapeutic uses
type
diabetes
ckd
Prior art date
Application number
MX2015013939A
Other languages
English (en)
Other versions
MX2015013939A (es
Inventor
Hans-Juergen Woerle
Eynatten Maximilian Von
Sreeraj Macha
Uli Broedl
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=51787230&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX375476(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of MX2015013939A publication Critical patent/MX2015013939A/es
Publication of MX375476B publication Critical patent/MX375476B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Biophysics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se refiere a determinados inhibidores de SGLT-2 para tratar y/o prevenir trastornos metabólicos, tales como diabetes mellitus tipo 2 o tipo 1, o prediabetes, en pacientes con insuficiencia renal o enfermedad renal crónica (CKD).
MX2015013939A 2013-04-05 2014-04-03 Composición farmacéutica que comprende empagliflozina, métodos para tratamiento y sus usos. MX375476B (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201361808804P 2013-04-05 2013-04-05
CA2812519A CA2812519A1 (en) 2013-04-05 2013-04-10 Pharmaceutical composition, methods for treating and uses thereof
US201361908991P 2013-11-26 2013-11-26
PCT/EP2014/056657 WO2014161919A1 (en) 2013-04-05 2014-04-03 Therapeutic uses of empagliflozin

Publications (2)

Publication Number Publication Date
MX2015013939A MX2015013939A (es) 2016-07-20
MX375476B true MX375476B (es) 2025-03-06

Family

ID=51787230

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2015013939A MX375476B (es) 2013-04-05 2014-04-03 Composición farmacéutica que comprende empagliflozina, métodos para tratamiento y sus usos.
MX2020010004A MX2020010004A (es) 2013-04-05 2015-10-01 Composicion farmaceutica que comprende empagliflozina, metodos para tratamiento y sus usos.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2020010004A MX2020010004A (es) 2013-04-05 2015-10-01 Composicion farmaceutica que comprende empagliflozina, metodos para tratamiento y sus usos.

Country Status (15)

Country Link
US (1) US12433906B2 (es)
EP (2) EP3456332A1 (es)
JP (1) JP6177992B2 (es)
KR (3) KR20210130844A (es)
CN (2) CN105377267A (es)
AU (1) AU2014247092B2 (es)
CA (3) CA2812519A1 (es)
DK (1) DK2981271T3 (es)
EA (1) EA033397B1 (es)
LT (1) LT2981271T (es)
MX (2) MX375476B (es)
PL (1) PL2981271T3 (es)
RS (1) RS58097B1 (es)
SI (1) SI2981271T1 (es)
WO (1) WO2014161919A1 (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
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PT2981271T (pt) 2013-04-05 2019-02-19 Boehringer Ingelheim Int Utilizações terapêuticas de empagliflozina
HK1213818A1 (zh) 2013-04-05 2016-07-15 勃林格殷格翰国际有限公司 依帕列净的治疗用途
US11813275B2 (en) 2013-04-05 2023-11-14 Boehringer Ingelheim International Gmbh Pharmaceutical composition, methods for treating and uses thereof
CA2812519A1 (en) 2013-04-05 2014-10-05 Boehringer Ingelheim International Gmbh Pharmaceutical composition, methods for treating and uses thereof
EA033286B1 (ru) 2013-04-18 2019-09-30 Бёрингер Ингельхайм Интернациональ Гмбх Способ лечения или отсрочки развития хронической болезни почек
CN105769782A (zh) * 2014-12-23 2016-07-20 中美华世通生物医药科技（武汉）有限公司 恩格列净片及其制备方法和用途
CN106880595A (zh) * 2015-12-10 2017-06-23 常州方楠医药技术有限公司 一种无定型依帕列净的固体分散体及其制备方法
JP7625363B2 (ja) * 2016-11-10 2025-02-03 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 医薬組成物、治療方法及びその使用
BR112020006472A2 (pt) 2017-10-02 2020-10-06 Poxel método para tratamento ou prevenção de insuficiência cardíaca com fração de ejeção preservada (icfep)
WO2019228365A1 (zh) 2018-05-31 2019-12-05 华领医药技术（上海）有限公司 含有葡萄糖激酶激活剂和dpp-iv抑制剂的药物组合、组合物和复方制剂及其制备方法和用途
BR112020024643A2 (pt) 2018-06-06 2021-03-02 Metavant Sciences Gmbh método de tratamento de pré-diabetes ou diabetes mellitus tipo 1 ou tipo 2, método de melhoria do controle glicêmico em um sujeito tendo pré-diabetes ou diabetes tipo 1 ou tipo 2, imeglimina para uso em um método para tratamento de pré-diabetes ou diabetes mellitus tipo 1 ou tipo 2 de um sujeito, imeglimina para uso em um método para melhoria do controle glicêmico em um sujeito tendo pré-diabetes ou diabetes tipo 1 ou tipo 2, uso de imeglimina para a fabricação de um medicamento para o tratamento de um sujeito tendo pré-diabetes ou diabetes mellitus tipo 1 ou tipo 2 e uso de imeglimina para a fabricação de um medicamento para melhoria do controle glicêmico em um sujeito tendo pré-diabetes ou diabetes tipo 1 ou tipo 2
EP3806828A1 (en) 2018-06-14 2021-04-21 Poxel Film-coated tablet comprising a triazine derivative for use in the treatment of diabetes
CN110141555A (zh) * 2019-06-21 2019-08-20 江苏豪森药业集团有限公司 一种恩格列净片及其制备方法
CN110721170A (zh) * 2019-10-24 2020-01-24 安徽九华华源药业有限公司 一种恩格列净片剂及其制备方法
WO2022065895A1 (ko) * 2020-09-24 2022-03-31 동아에스티 주식회사 Sglt-2 억제제인 엠파글리플로진 유도체의 신규염 및 염의 수화물

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