MX367131B - Sales de xantilio 3,6-disustituidas. - Google Patents

Sales de xantilio 3,6-disustituidas.

Info

Publication number
MX367131B
MX367131B MX2014012523A MX2014012523A MX367131B MX 367131 B MX367131 B MX 367131B MX 2014012523 A MX2014012523 A MX 2014012523A MX 2014012523 A MX2014012523 A MX 2014012523A MX 367131 B MX367131 B MX 367131B
Authority
MX
Mexico
Prior art keywords
medicaments
compounds
disubstituted
xanthylium salts
salts
Prior art date
Application number
MX2014012523A
Other languages
English (en)
Inventor
Clunas Scott
Mervyn David Storey John
Horsley David
Robert Harrington Charles
Michel Wischik Claude
Elizabeth Rickard Janet
Original Assignee
Wista Lab Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wista Lab Ltd filed Critical Wista Lab Ltd
Publication of MX367131B publication Critical patent/MX367131B/es

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    • C07D311/78—Ring systems having three or more relevant rings
    • C07D311/80—Dibenzopyrans; Hydrogenated dibenzopyrans
    • C07D311/82—Xanthenes
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    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
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    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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Abstract

Esta invención se refiere generalmente a procedimientos, usos, métodos y materiales que utilizan compuestos de xantilio particulares, incluyendo compuestos de la fórmula (I) y (II), como se definen más en la presente. (ver Fórmulas) Estos compuestos son útiles como fármacos, por ejemplo, en el tratamiento de tauopatías, tales como enfermedad de Alzheimer.
MX2014012523A 2008-12-10 2009-12-10 Sales de xantilio 3,6-disustituidas. MX367131B (es)

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PCT/GB2009/002865 WO2010067078A2 (en) 2008-12-10 2009-12-10 3,6-disubstituted xanthylium salts as medicaments

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EP3689346A1 (en) 2020-08-05
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