MX2015011955A - Lipidos y composiciones de lipidos para el suministro de agentes activos. - Google Patents

Lipidos y composiciones de lipidos para el suministro de agentes activos.

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Publication number
MX2015011955A
MX2015011955A MX2015011955A MX2015011955A MX2015011955A MX 2015011955 A MX2015011955 A MX 2015011955A MX 2015011955 A MX2015011955 A MX 2015011955A MX 2015011955 A MX2015011955 A MX 2015011955A MX 2015011955 A MX2015011955 A MX 2015011955A
Authority
MX
Mexico
Prior art keywords
delivery
active agents
lipids
lipid compositions
formula
Prior art date
Application number
MX2015011955A
Other languages
English (en)
Inventor
Chandra Vargeese
Jeremy Lee Baryza
Rohan Eric John Beckwith
Keith Bowman
Crystal Byers
Tanzina Fazal
Gabriel Grant Gamber
Cameron Chuck-Munn Lee
Ritesh Bhanudasji Tichkule
Laura West
Shuangxi Wang
Thomas Zabawa
Junping Zhao
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MX2015011955A publication Critical patent/MX2015011955A/es

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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
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    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
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Abstract

Esta invención proporciona un compuesto de la fórmula (I): (ver Fórmula) o una sal farmacéuticamente aceptable del mismo, en donde R1-R4, L y X se definen en la presente. Los compuestos de la fórmula (I) y las sales farmacéuticamente aceptables de los mismos son lípidos catiónicos útiles en el suministro de agentes biológicamente activos a las células y los tejidos.
MX2015011955A 2013-03-08 2014-03-06 Lipidos y composiciones de lipidos para el suministro de agentes activos. MX2015011955A (es)

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