ME00058B - Derivati aminoindazola, postupak izrade i međuproizvodi ovog postupka kao medicinski produkti i farmaceutske kompozicije koje ih sadrži - Google Patents

Derivati aminoindazola, postupak izrade i međuproizvodi ovog postupka kao medicinski produkti i farmaceutske kompozicije koje ih sadrži

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Publication number
ME00058B
ME00058B MEP-2008-161A MEP2008161A ME00058B ME 00058 B ME00058 B ME 00058B ME P2008161 A MEP2008161 A ME P2008161A ME 00058 B ME00058 B ME 00058B
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ME
Montenegro
Prior art keywords
procedure
heteroarylalkyl
derivatives
aminoindasol
intermediates
Prior art date
Application number
MEP-2008-161A
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English (en)
French (fr)
Inventor
Rosset Gilles Dutruc
Dominique Lesuisse
Thomas Rooney
Franck Halley
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Aventis Pharma Sa
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Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of ME00058B publication Critical patent/ME00058B/me

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    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
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Abstract

Pronalazak se odnosi na nove derivate indazola koji imaju opštu formulu (I): pri čemu je R O, S ili NH; R3 je alkil, aril,arilalkil, heteroaril, heteroarilalkil, aril, heterociklil, cikloalkil, alkenil itd., radikal; navedeni radikali su opciono supstituisanisa 1 ili više supstituenata; R4, R5, R6 i R7 su nezavisno izabrani od sledećih radikala: vodonika, halogena, CN, N02, NH2,OH, COOH, C(O)OR8, -O-C(O)R8, NR8R9, NHC(O)R8, C(O)NR8R9, NHC(S)R8, C(S)NR8R9, SR8, S(O)R8, S02R8,NHS02R8, S02NR8R9, trifluorometil, trifluorometoksi, alkil, alkoksi, aril, arilalkil, heteroaril, heteroarilalkil, heterociklil,cikloalkil, alkenil itd., navedeni radikali su opciono supstituisani sa 1 ili više supstituenata.
MEP-2008-161A 2002-03-11 2003-03-07 Derivati aminoindazola, postupak izrade i međuproizvodi ovog postupka kao medicinski produkti i farmaceutske kompozicije koje ih sadrži ME00058B (me)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR0202997A FR2836915B1 (fr) 2002-03-11 2002-03-11 Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
PCT/FR2003/000752 WO2003078403A2 (fr) 2002-03-11 2003-03-07 Derives d’aminoindazoles comme inhibiteurs de proteine-kinase
EP03744396.7A EP1487804B1 (fr) 2002-03-11 2003-03-07 Derives d'aminoindazoles comme inhibiteurs de proteine-kinase

Publications (1)

Publication Number Publication Date
ME00058B true ME00058B (me) 2010-10-10

Family

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Application Number Title Priority Date Filing Date
MEP-2008-161A ME00058B (me) 2002-03-11 2003-03-07 Derivati aminoindazola, postupak izrade i međuproizvodi ovog postupka kao medicinski produkti i farmaceutske kompozicije koje ih sadrži
MEP-161/08A MEP16108A (en) 2002-03-11 2003-03-07 Derives d'aminoindazoles comme inhibiteurs de proteine-kinase

Family Applications After (1)

Application Number Title Priority Date Filing Date
MEP-161/08A MEP16108A (en) 2002-03-11 2003-03-07 Derives d'aminoindazoles comme inhibiteurs de proteine-kinase

Country Status (30)

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US (1) US6949579B2 (me)
EP (1) EP1487804B1 (me)
JP (2) JP4648630B2 (me)
KR (1) KR101068770B1 (me)
CN (2) CN1656078A (me)
AR (1) AR038915A1 (me)
AU (1) AU2003242809B8 (me)
BR (1) BR0308373A (me)
CA (1) CA2478542C (me)
FR (1) FR2836915B1 (me)
GT (1) GT200300057A (me)
HR (1) HRP20040824B1 (me)
IL (2) IL163831A0 (me)
JO (1) JO2326B1 (me)
MA (1) MA27230A1 (me)
ME (2) ME00058B (me)
MX (1) MXPA04007478A (me)
MY (1) MY138269A (me)
NO (1) NO329384B1 (me)
NZ (1) NZ535147A (me)
PA (1) PA8568301A1 (me)
PE (1) PE20040155A1 (me)
PL (1) PL370478A1 (me)
RS (1) RS52396B (me)
RU (1) RU2345070C2 (me)
SV (1) SV2003001494A (me)
TW (1) TWI329103B (me)
UY (1) UY27713A1 (me)
WO (1) WO2003078403A2 (me)
ZA (1) ZA200406687B (me)

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