KR20070090172A - 단백질 키나아제의 억제제로서 유용한피라졸로[1,5-ａ]피리미딘 - Google Patents
단백질 키나아제의 억제제로서 유용한피라졸로[1,5-ａ]피리미딘 Download PDFInfo
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- KR20070090172A KR20070090172A KR1020077012308A KR20077012308A KR20070090172A KR 20070090172 A KR20070090172 A KR 20070090172A KR 1020077012308 A KR1020077012308 A KR 1020077012308A KR 20077012308 A KR20077012308 A KR 20077012308A KR 20070090172 A KR20070090172 A KR 20070090172A
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Landscapes
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| US62544604P | 2004-11-04 | 2004-11-04 | |
| US60/625,446 | 2004-11-04 |
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| KR20070090172A true KR20070090172A (ko) | 2007-09-05 |
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| EP (1) | EP1812440B1 (https=) |
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| AT (1) | ATE482213T1 (https=) |
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| DK (1) | DK1812440T3 (https=) |
| ES (1) | ES2354824T3 (https=) |
| IL (1) | IL182893A0 (https=) |
| MX (1) | MX337817B (https=) |
| NO (1) | NO20072795L (https=) |
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| RU (1) | RU2417996C2 (https=) |
| SI (1) | SI1812440T1 (https=) |
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20240155634A (ko) | 2023-04-20 | 2024-10-29 | 한국화학연구원 | 신규한 헤테로고리 화합물 또는 이의 약학적으로 허용가능한 염 및 이를 유효성분으로 포함하는 바이러스성 질환의 예방 또는 치료용 약학적 조성물 |
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| ATE482213T1 (de) * | 2004-11-04 | 2010-10-15 | Vertex Pharma | Als inhibitoren von proteinkinasen geeignete pyrazoloä1,5-aüpyrimidine |
| PT1853588E (pt) * | 2005-02-16 | 2008-08-25 | Astrazeneca Ab | Compostos químicos |
| US20090156617A1 (en) * | 2005-05-12 | 2009-06-18 | Northrup Alan B | Tyrosine kinase inhibitors |
| EP1899323A2 (en) * | 2005-05-16 | 2008-03-19 | AstraZeneca AB | Pyrazolylaminopyrimidine derivatives useful as tyrosine kinase inhibitors |
| WO2007046867A2 (en) * | 2005-05-19 | 2007-04-26 | Xenon Pharmaceuticals Inc. | Piperidine derivatives and their uses as therapeutic agents |
| WO2006127587A1 (en) * | 2005-05-20 | 2006-11-30 | Vertex Pharmaceuticals Incorporated | Pyrrolopyridines useful as inhibitors of protein kinase |
| WO2007049041A1 (en) * | 2005-10-28 | 2007-05-03 | Astrazeneca Ab | 4- (3-aminopyrazole) pyrimidine derivatives for use as tyrosine kinase inhibitors in the treatment of cancer |
| EP2455382B1 (en) | 2005-12-13 | 2016-10-26 | Incyte Holdings Corporation | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors |
| GB0601638D0 (en) * | 2006-01-27 | 2006-03-08 | Merck Sharp & Dohme | Therapeutic treatment |
| PE20080403A1 (es) * | 2006-07-14 | 2008-04-25 | Amgen Inc | Derivados heterociclicos fusionados y metodos de uso |
| US8198448B2 (en) | 2006-07-14 | 2012-06-12 | Amgen Inc. | Fused heterocyclic derivatives and methods of use |
| US8217177B2 (en) | 2006-07-14 | 2012-07-10 | Amgen Inc. | Fused heterocyclic derivatives and methods of use |
| CA2668286C (en) | 2006-11-03 | 2014-09-16 | Pharmacyclics, Inc. | Bruton's tyrosine kinase activity probe and method of using |
| CN101778825A (zh) * | 2007-03-22 | 2010-07-14 | 沃泰克斯药物股份有限公司 | 适用作詹纳斯激酶抑制剂的n-杂环类化合物 |
| WO2008129255A1 (en) * | 2007-04-18 | 2008-10-30 | Astrazeneca Ab | 5-aminopyrazol-3-yl-3h-imidazo [4,5-b] pyridine derivatives and their use for the treatment of cancer |
| UA99459C2 (en) * | 2007-05-04 | 2012-08-27 | Астразенека Аб | 9-(pyrazol-3-yl)- 9h-purine-2-amine and 3-(pyraz0l-3-yl)-3h-imidazo[4,5-b]pyridin-5-amine derivatives and their use for the treatment of cancer |
| US20100137398A1 (en) * | 2007-05-04 | 2010-06-03 | Novartis Ag | Use of hdac inhibitors for the treatment of gastrointestinal cancers |
| EP3070090B1 (en) | 2007-06-13 | 2018-12-12 | Incyte Holdings Corporation | Use of salts of the janus kinase inhibitor (r)-3-(4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h- pyrazol-1-yl)-3- cyclopentylpropanenitrile |
| CN101878217B (zh) * | 2007-09-28 | 2014-01-15 | 协和发酵麒麟株式会社 | 皮肤疾病的预防和/或治疗剂 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| KR20240155634A (ko) | 2023-04-20 | 2024-10-29 | 한국화학연구원 | 신규한 헤테로고리 화합물 또는 이의 약학적으로 허용가능한 염 및 이를 유효성분으로 포함하는 바이러스성 질환의 예방 또는 치료용 약학적 조성물 |
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| AU2005304784B2 (en) | 2011-03-24 |
| HK1113569A1 (en) | 2008-10-10 |
| CN101094853B (zh) | 2011-07-13 |
| MX337817B (es) | 2011-11-04 |
| IL182893A0 (en) | 2007-08-19 |
| DK1812440T3 (da) | 2011-01-31 |
| ES2354824T3 (es) | 2011-03-18 |
| ZA200704476B (en) | 2008-09-25 |
| JP5030229B2 (ja) | 2012-09-19 |
| MX2007005439A (es) | 2008-02-19 |
| CA2586375A1 (en) | 2006-05-18 |
| AU2005304784A1 (en) | 2006-05-18 |
| RU2417996C2 (ru) | 2011-05-10 |
| DE602005023763D1 (de) | 2010-11-04 |
| EP1812440A1 (en) | 2007-08-01 |
| US20060135537A1 (en) | 2006-06-22 |
| ATE482213T1 (de) | 2010-10-15 |
| PT1812440E (pt) | 2011-01-25 |
| CN101094853A (zh) | 2007-12-26 |
| NZ555236A (en) | 2010-10-29 |
| SI1812440T1 (sl) | 2011-04-29 |
| JP2008519059A (ja) | 2008-06-05 |
| NO20072795L (no) | 2007-06-01 |
| JP2009067803A (ja) | 2009-04-02 |
| EP1812440B1 (en) | 2010-09-22 |
| RU2007120518A (ru) | 2008-12-10 |
| US7528138B2 (en) | 2009-05-05 |
| WO2006052913A1 (en) | 2006-05-18 |
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