KR20070090172A - 단백질 키나아제의 억제제로서 유용한피라졸로[1,5-ａ]피리미딘 - Google Patents
단백질 키나아제의 억제제로서 유용한피라졸로[1,5-ａ]피리미딘 Download PDFInfo
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- KR20070090172A KR20070090172A KR1020077012308A KR20077012308A KR20070090172A KR 20070090172 A KR20070090172 A KR 20070090172A KR 1020077012308 A KR1020077012308 A KR 1020077012308A KR 20077012308 A KR20077012308 A KR 20077012308A KR 20070090172 A KR20070090172 A KR 20070090172A
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Landscapes
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| US62544604P | 2004-11-04 | 2004-11-04 | |
| US60/625,446 | 2004-11-04 |
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| KR20070090172A true KR20070090172A (ko) | 2007-09-05 |
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| EP (1) | EP1812440B1 (https=) |
| JP (2) | JP5030229B2 (https=) |
| KR (1) | KR20070090172A (https=) |
| CN (1) | CN101094853B (https=) |
| AT (1) | ATE482213T1 (https=) |
| AU (1) | AU2005304784B2 (https=) |
| CA (1) | CA2586375A1 (https=) |
| DE (1) | DE602005023763D1 (https=) |
| DK (1) | DK1812440T3 (https=) |
| ES (1) | ES2354824T3 (https=) |
| IL (1) | IL182893A0 (https=) |
| MX (1) | MX337817B (https=) |
| NO (1) | NO20072795L (https=) |
| NZ (1) | NZ555236A (https=) |
| PT (1) | PT1812440E (https=) |
| RU (1) | RU2417996C2 (https=) |
| SI (1) | SI1812440T1 (https=) |
| WO (1) | WO2006052913A1 (https=) |
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20240155634A (ko) | 2023-04-20 | 2024-10-29 | 한국화학연구원 | 신규한 헤테로고리 화합물 또는 이의 약학적으로 허용가능한 염 및 이를 유효성분으로 포함하는 바이러스성 질환의 예방 또는 치료용 약학적 조성물 |
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| SE0104140D0 (sv) * | 2001-12-07 | 2001-12-07 | Astrazeneca Ab | Novel Compounds |
| PT1812440E (pt) * | 2004-11-04 | 2011-01-25 | Vertex Pharma | Pirazolo[1,5-a]pirimidinas úteis enquanto inibidores de proteínas cinases |
| SI1853588T1 (sl) * | 2005-02-16 | 2008-10-31 | Astrazeneca Ab | Kemične spojine |
| US20090156617A1 (en) * | 2005-05-12 | 2009-06-18 | Northrup Alan B | Tyrosine kinase inhibitors |
| US20080287437A1 (en) * | 2005-05-16 | 2008-11-20 | Astrazeneca Ab | Pyrazolylaminopyrimidine Derivatives Useful as Tyrosine Kinase Inhibitors |
| WO2007046867A2 (en) * | 2005-05-19 | 2007-04-26 | Xenon Pharmaceuticals Inc. | Piperidine derivatives and their uses as therapeutic agents |
| EP2354140A1 (en) * | 2005-05-20 | 2011-08-10 | Vertex Pharmaceuticals Incorporated | Pyrrolopyridines useful as inhibitors of protein kinase |
| JP2009513615A (ja) * | 2005-10-28 | 2009-04-02 | アストラゼネカ アクチボラグ | 癌の治療においてチロシンキナーゼ阻害剤として使用するための４−（３−アミノピラゾール）ピリミジン誘導体 |
| SG10202003901UA (en) | 2005-12-13 | 2020-05-28 | Incyte Holdings Corp | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as janus kinase inhibitors |
| GB0601638D0 (en) * | 2006-01-27 | 2006-03-08 | Merck Sharp & Dohme | Therapeutic treatment |
| US8198448B2 (en) | 2006-07-14 | 2012-06-12 | Amgen Inc. | Fused heterocyclic derivatives and methods of use |
| PE20080403A1 (es) | 2006-07-14 | 2008-04-25 | Amgen Inc | Derivados heterociclicos fusionados y metodos de uso |
| US8217177B2 (en) | 2006-07-14 | 2012-07-10 | Amgen Inc. | Fused heterocyclic derivatives and methods of use |
| CA2668286C (en) | 2006-11-03 | 2014-09-16 | Pharmacyclics, Inc. | Bruton's tyrosine kinase activity probe and method of using |
| MX2009010127A (es) * | 2007-03-22 | 2009-11-05 | Vertex Pharma | Compuestos utiles como inhibidores de janus cinasas. |
| JP2010524911A (ja) * | 2007-04-18 | 2010-07-22 | アストラゼネカ アクチボラグ | ５−アミノピラゾール−３−イル−３Ｈ−イミダゾ［４，５−ｂ］ピリジン誘導体と癌の治療のためのその使用 |
| UA99459C2 (en) * | 2007-05-04 | 2012-08-27 | Астразенека Аб | 9-(pyrazol-3-yl)- 9h-purine-2-amine and 3-(pyraz0l-3-yl)-3h-imidazo[4,5-b]pyridin-5-amine derivatives and their use for the treatment of cancer |
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- 2005-11-04 RU RU2007120518/04A patent/RU2417996C2/ru not_active IP Right Cessation
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- 2005-11-04 WO PCT/US2005/040344 patent/WO2006052913A1/en not_active Ceased
- 2005-11-04 KR KR1020077012308A patent/KR20070090172A/ko not_active Ceased
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
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| KR20240155634A (ko) | 2023-04-20 | 2024-10-29 | 한국화학연구원 | 신규한 헤테로고리 화합물 또는 이의 약학적으로 허용가능한 염 및 이를 유효성분으로 포함하는 바이러스성 질환의 예방 또는 치료용 약학적 조성물 |
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| CN101094853B (zh) | 2011-07-13 |
| WO2006052913A1 (en) | 2006-05-18 |
| EP1812440B1 (en) | 2010-09-22 |
| ZA200704476B (en) | 2008-09-25 |
| RU2007120518A (ru) | 2008-12-10 |
| MX337817B (es) | 2011-11-04 |
| DE602005023763D1 (de) | 2010-11-04 |
| US7528138B2 (en) | 2009-05-05 |
| AU2005304784B2 (en) | 2011-03-24 |
| US20060135537A1 (en) | 2006-06-22 |
| ATE482213T1 (de) | 2010-10-15 |
| CN101094853A (zh) | 2007-12-26 |
| JP2009067803A (ja) | 2009-04-02 |
| ES2354824T3 (es) | 2011-03-18 |
| CA2586375A1 (en) | 2006-05-18 |
| AU2005304784A1 (en) | 2006-05-18 |
| SI1812440T1 (sl) | 2011-04-29 |
| JP2008519059A (ja) | 2008-06-05 |
| MX2007005439A (es) | 2008-02-19 |
| NZ555236A (en) | 2010-10-29 |
| NO20072795L (no) | 2007-06-01 |
| JP5030229B2 (ja) | 2012-09-19 |
| PT1812440E (pt) | 2011-01-25 |
| DK1812440T3 (da) | 2011-01-31 |
| HK1113569A1 (en) | 2008-10-10 |
| IL182893A0 (en) | 2007-08-19 |
| EP1812440A1 (en) | 2007-08-01 |
| RU2417996C2 (ru) | 2011-05-10 |
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