KR101290925B1 - 코팅된 정제 제형 및 방법 - Google Patents

코팅된 정제 제형 및 방법 Download PDF

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Publication number
KR101290925B1
KR101290925B1 KR1020067024818A KR20067024818A KR101290925B1 KR 101290925 B1 KR101290925 B1 KR 101290925B1 KR 1020067024818 A KR1020067024818 A KR 1020067024818A KR 20067024818 A KR20067024818 A KR 20067024818A KR 101290925 B1 KR101290925 B1 KR 101290925B1
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KR
South Korea
Prior art keywords
coating layer
polyvinyl alcohol
tablet
coated
coating
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
KR1020067024818A
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English (en)
Korean (ko)
Other versions
KR20070027560A (ko
Inventor
디비아칸트 데사이
빙 브이. 리
Original Assignee
브리스톨-마이어스 스큅 컴퍼니
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34971747&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR101290925(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 브리스톨-마이어스 스큅 컴퍼니 filed Critical 브리스톨-마이어스 스큅 컴퍼니
Publication of KR20070027560A publication Critical patent/KR20070027560A/ko
Application granted granted Critical
Publication of KR101290925B1 publication Critical patent/KR101290925B1/ko
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Expired - Lifetime legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR1020067024818A 2004-05-28 2005-05-26 코팅된 정제 제형 및 방법 Expired - Lifetime KR101290925B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US57531904P 2004-05-28 2004-05-28
US60/575,319 2004-05-28
PCT/US2005/018692 WO2005117841A1 (en) 2004-05-28 2005-05-26 Coated tablet formulation and method

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1020127014475A Division KR20120064141A (ko) 2004-05-28 2005-05-26 코팅된 정제 제형 및 방법

Publications (2)

Publication Number Publication Date
KR20070027560A KR20070027560A (ko) 2007-03-09
KR101290925B1 true KR101290925B1 (ko) 2013-07-29

Family

ID=34971747

Family Applications (2)

Application Number Title Priority Date Filing Date
KR1020067024818A Expired - Lifetime KR101290925B1 (ko) 2004-05-28 2005-05-26 코팅된 정제 제형 및 방법
KR1020127014475A Ceased KR20120064141A (ko) 2004-05-28 2005-05-26 코팅된 정제 제형 및 방법

Family Applications After (1)

Application Number Title Priority Date Filing Date
KR1020127014475A Ceased KR20120064141A (ko) 2004-05-28 2005-05-26 코팅된 정제 제형 및 방법

Country Status (33)

Country Link
US (4) US7951400B2 (enExample)
EP (3) EP2298288B2 (enExample)
JP (1) JP4901727B2 (enExample)
KR (2) KR101290925B1 (enExample)
CN (2) CN1988891B (enExample)
AR (2) AR049062A1 (enExample)
AU (1) AU2005249467B2 (enExample)
BR (1) BRPI0510419B8 (enExample)
CA (1) CA2568391C (enExample)
CY (2) CY1117813T1 (enExample)
DK (2) DK1753406T4 (enExample)
ES (3) ES2582646T5 (enExample)
GE (1) GEP20094639B (enExample)
HR (2) HRP20160880T4 (enExample)
HU (2) HUE029446T2 (enExample)
IL (2) IL179454A (enExample)
LT (1) LT2298288T (enExample)
ME (2) ME02643B (enExample)
MX (1) MXPA06013711A (enExample)
MY (1) MY147639A (enExample)
NO (1) NO343907B1 (enExample)
NZ (1) NZ551591A (enExample)
PE (1) PE20060425A1 (enExample)
PH (1) PH12013500450A1 (enExample)
PL (2) PL2298288T5 (enExample)
PT (2) PT1753406E (enExample)
RS (2) RS54929B2 (enExample)
RU (1) RU2372894C2 (enExample)
SI (3) SI1753406T2 (enExample)
TW (2) TWI415635B (enExample)
UA (1) UA88168C2 (enExample)
WO (1) WO2005117841A1 (enExample)
ZA (1) ZA200609541B (enExample)

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