JPS5753454A - Guanidinobenzoate and anticomplementary agent - Google Patents

Guanidinobenzoate and anticomplementary agent

Info

Publication number
JPS5753454A
JPS5753454A JP12826980A JP12826980A JPS5753454A JP S5753454 A JPS5753454 A JP S5753454A JP 12826980 A JP12826980 A JP 12826980A JP 12826980 A JP12826980 A JP 12826980A JP S5753454 A JPS5753454 A JP S5753454A
Authority
JP
Japan
Prior art keywords
agent
expressed
formula
anticomplementary
remedy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP12826980A
Other languages
English (en)
Japanese (ja)
Other versions
JPS611063B2 (https=
Inventor
Setsuo Fujii
Toshiyuki Okutome
Toyoo Nakayama
Takashi Yaegashi
Masateru Kurumi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Torii Pharmaceutical Co Ltd
Original Assignee
Torii Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Torii Pharmaceutical Co Ltd filed Critical Torii Pharmaceutical Co Ltd
Priority to JP12826980A priority Critical patent/JPS5753454A/ja
Priority to AU75062/81A priority patent/AU527371B2/en
Priority to US06/300,534 priority patent/US4454338A/en
Priority to CA000385570A priority patent/CA1177488A/en
Priority to ZA816363A priority patent/ZA816363B/xx
Priority to ES505460A priority patent/ES8206443A1/es
Priority to CS816809A priority patent/CS228534B2/cs
Priority to PH26206A priority patent/PH18109A/en
Priority to FI812876A priority patent/FI73975C/fi
Priority to HU812665A priority patent/HU185956B/hu
Priority to EP81107274A priority patent/EP0048433B1/en
Priority to DE8181107274T priority patent/DE3174717D1/de
Priority to GB8127837A priority patent/GB2083818B/en
Priority to MX10156181U priority patent/MX6922E/es
Priority to NO813138A priority patent/NO153568C/no
Priority to KR1019810003427A priority patent/KR860000264B1/ko
Priority to AT81107274T priority patent/ATE20051T1/de
Priority to SU813384251A priority patent/SU1176832A3/ru
Priority to DK410681A priority patent/DK155003C/da
Priority to DD81233339A priority patent/DD201779A5/de
Publication of JPS5753454A publication Critical patent/JPS5753454A/ja
Priority to US06/572,269 priority patent/US4532255A/en
Publication of JPS611063B2 publication Critical patent/JPS611063B2/ja
Granted legal-status Critical Current

Links

Landscapes

  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP12826980A 1980-09-16 1980-09-16 Guanidinobenzoate and anticomplementary agent Granted JPS5753454A (en)

Priority Applications (21)

Application Number Priority Date Filing Date Title
JP12826980A JPS5753454A (en) 1980-09-16 1980-09-16 Guanidinobenzoate and anticomplementary agent
AU75062/81A AU527371B2 (en) 1980-09-16 1981-09-08 Amidine
US06/300,534 US4454338A (en) 1980-09-16 1981-09-09 Amidine compound
CA000385570A CA1177488A (en) 1980-09-16 1981-09-10 Amidine compound, process for producing same and anti- complement agent comprising same
ZA816363A ZA816363B (en) 1980-09-16 1981-09-14 Novel amidine compound,process for producing same and anti-complement agent comprising same
ES505460A ES8206443A1 (es) 1980-09-16 1981-09-14 Un procedimiento para preparar un derivado de amidina
DE8181107274T DE3174717D1 (en) 1980-09-16 1981-09-15 Novel amidine compounds, process for producing same and anti-complement agent comprising them
KR1019810003427A KR860000264B1 (ko) 1980-09-16 1981-09-15 아미딘 화합물 및 그 염의 제조방법
FI812876A FI73975C (fi) 1980-09-16 1981-09-15 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara amidinoderivat.
HU812665A HU185956B (en) 1980-09-16 1981-09-15 Process for producing new amidine derivatives and pharmaceutical compositions containing them as active agents
EP81107274A EP0048433B1 (en) 1980-09-16 1981-09-15 Novel amidine compounds, process for producing same and anti-complement agent comprising them
CS816809A CS228534B2 (en) 1980-09-16 1981-09-15 Production method of amidine derivative
GB8127837A GB2083818B (en) 1980-09-16 1981-09-15 Amidine compounds
MX10156181U MX6922E (es) 1980-09-16 1981-09-15 Procedimiento para preparar compuestos de amidina
NO813138A NO153568C (no) 1980-09-16 1981-09-15 Analogifremgangsmaate for fremstilling av fysiologisk aktive amidinderivater.
PH26206A PH18109A (en) 1980-09-16 1981-09-15 Novel amidine compounds and anti-complement pharmaceutical composition comprising same
AT81107274T ATE20051T1 (de) 1980-09-16 1981-09-15 Amidinderivate, verfahren zu ihrer herstellung und diese enthaltende antikomplement-mittel.
SU813384251A SU1176832A3 (ru) 1980-09-16 1981-09-15 Способ получени амидиновых производных
DK410681A DK155003C (da) 1980-09-16 1981-09-15 Analogifremgangsmaade til fremstilling af amidin-derivater eller farmaceutisk acceptable syreadditionssalte deraf
DD81233339A DD201779A5 (de) 1980-09-16 1981-09-16 Verfahren zur herstellung neuer amidinverbindungen
US06/572,269 US4532255A (en) 1980-09-16 1984-01-20 Amidine compounds and anticomplement agent comprising same

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP12826980A JPS5753454A (en) 1980-09-16 1980-09-16 Guanidinobenzoate and anticomplementary agent

Publications (2)

Publication Number Publication Date
JPS5753454A true JPS5753454A (en) 1982-03-30
JPS611063B2 JPS611063B2 (https=) 1986-01-13

Family

ID=14980652

Family Applications (1)

Application Number Title Priority Date Filing Date
JP12826980A Granted JPS5753454A (en) 1980-09-16 1980-09-16 Guanidinobenzoate and anticomplementary agent

Country Status (2)

Country Link
JP (1) JPS5753454A (https=)
ZA (1) ZA816363B (https=)

Cited By (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3004405U (ja) * 1994-05-19 1994-11-15 株式会社エス・ピー・ユー 表裏連続模様を有するｔシャツ
WO1996020917A1 (en) * 1995-01-05 1996-07-11 Torii Pharmaceutical Co., Ltd. Substituted amidinonaphthyl ester derivatives
WO1996020920A1 (en) * 1995-01-05 1996-07-11 Torii Pharmaceutical Co., Ltd. Amidinonaphthyl ester derivative
WO1999051662A1 (en) * 1998-04-01 1999-10-14 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Polyimide compositions
JP2000290179A (ja) * 1999-03-31 2000-10-17 Shimizu Pharmaceutical Co Ltd 安定な６−アミジノ−２−ナフチル４−グアニジノベンゾエート酸付加塩製剤ならびにその製造方法
WO2001094299A1 (en) * 2000-06-08 2001-12-13 Shizuoka Coffein Co., Ltd. Benzene derivatives
WO2006123674A1 (ja) * 2005-05-17 2006-11-23 Santen Pharmaceutical Co., Ltd. アミン誘導体を有効成分として含む血管新生阻害剤
EP2119440A1 (en) 2005-05-17 2009-11-18 Santen Pharmaceutical Co., Ltd. Amidino derivatives for use in the prevention or treatment of retinitis pigmentosa and Leber's disease
JP2012087099A (ja) * 2010-10-21 2012-05-10 Katsura Chemical Co Ltd ナファモスタットメシル酸塩の晶析方法
WO2013039187A1 (ja) 2011-09-15 2013-03-21 アステラス製薬株式会社 グアニジノ安息香酸化合物
WO2014142219A1 (ja) 2013-03-13 2014-09-18 アステラス製薬株式会社 グアニジノ安息香酸エステル化合物
JPWO2014007326A1 (ja) * 2012-07-04 2016-06-02 味の素株式会社 ナファモスタットメシル酸塩の製造方法
US9969705B2 (en) 2014-02-13 2018-05-15 Takeda Pharmaceutical Company Limited Fused heterocyclic compound
US10023544B2 (en) 2014-02-13 2018-07-17 Takeda Pharmaceutical Company Limited Heterocyclic compound
KR102288679B1 (ko) 2021-01-14 2021-08-11 대봉엘에스 주식회사 메실산 나파모스타트의 공결정다형 및 그의 제조방법

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2003246730A (ja) * 2002-02-22 2003-09-02 Torii Yakuhin Kk トリプターゼ阻害剤
WO2005120491A1 (ja) * 2004-06-14 2005-12-22 Torii Pharmaceutical Co., Ltd. 炎症性腸疾患の治療薬又は予防薬

Cited By (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3004405U (ja) * 1994-05-19 1994-11-15 株式会社エス・ピー・ユー 表裏連続模様を有するｔシャツ
WO1996020917A1 (en) * 1995-01-05 1996-07-11 Torii Pharmaceutical Co., Ltd. Substituted amidinonaphthyl ester derivatives
WO1996020920A1 (en) * 1995-01-05 1996-07-11 Torii Pharmaceutical Co., Ltd. Amidinonaphthyl ester derivative
AU686104B2 (en) * 1995-01-05 1998-02-05 Torii Pharmaceutical Co., Ltd. Substituted amidinonaphthyl ester derivatives
US5885990A (en) * 1995-01-05 1999-03-23 Torii Pharmaceutical Co., Ltd. Substituted amidinonaphthyl ester derivative
WO1999051662A1 (en) * 1998-04-01 1999-10-14 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Polyimide compositions
US6303742B1 (en) 1998-04-01 2001-10-16 Kanekafuchi Kagaku Kogyo Kabushiki Kaisha Polyimide compositions
US6689899B2 (en) 1998-04-01 2004-02-10 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Diamine and acid anhydride
JP2000290179A (ja) * 1999-03-31 2000-10-17 Shimizu Pharmaceutical Co Ltd 安定な６−アミジノ−２−ナフチル４−グアニジノベンゾエート酸付加塩製剤ならびにその製造方法
WO2001094299A1 (en) * 2000-06-08 2001-12-13 Shizuoka Coffein Co., Ltd. Benzene derivatives
EP2143431A1 (en) 2005-05-17 2010-01-13 Santen Pharmaceutical Co., Ltd. Protective agent for neurocyte comprising amidino derivative as active ingredient
WO2006123674A1 (ja) * 2005-05-17 2006-11-23 Santen Pharmaceutical Co., Ltd. アミン誘導体を有効成分として含む血管新生阻害剤
EP2236136A1 (en) 2005-05-17 2010-10-06 Santen Pharmaceutical Co., Ltd. Angiogenesis inhibitor containing amine derivate as active ingredient
EP2119440A1 (en) 2005-05-17 2009-11-18 Santen Pharmaceutical Co., Ltd. Amidino derivatives for use in the prevention or treatment of retinitis pigmentosa and Leber's disease
JP2012087099A (ja) * 2010-10-21 2012-05-10 Katsura Chemical Co Ltd ナファモスタットメシル酸塩の晶析方法
US9199927B2 (en) 2011-09-15 2015-12-01 Astellas Pharma Inc. Guanidinobenzoic acid compound
WO2013039187A1 (ja) 2011-09-15 2013-03-21 アステラス製薬株式会社 グアニジノ安息香酸化合物
KR20140061515A (ko) 2011-09-15 2014-05-21 아스텔라스세이야쿠 가부시키가이샤 구아니디노벤조산 화합물
JPWO2014007326A1 (ja) * 2012-07-04 2016-06-02 味の素株式会社 ナファモスタットメシル酸塩の製造方法
KR20150130392A (ko) 2013-03-13 2015-11-23 아스텔라스세이야쿠 가부시키가이샤 구아니디노벤조산 에스테르 화합물
WO2014142219A1 (ja) 2013-03-13 2014-09-18 アステラス製薬株式会社 グアニジノ安息香酸エステル化合物
JPWO2014142219A1 (ja) * 2013-03-13 2017-02-16 アステラス製薬株式会社 グアニジノ安息香酸エステル化合物
US9969709B2 (en) 2013-03-13 2018-05-15 Takeda Pharmaceutical Company Limited Guanidinobenzoic acid ester compound
US9969705B2 (en) 2014-02-13 2018-05-15 Takeda Pharmaceutical Company Limited Fused heterocyclic compound
US10023544B2 (en) 2014-02-13 2018-07-17 Takeda Pharmaceutical Company Limited Heterocyclic compound
KR102288679B1 (ko) 2021-01-14 2021-08-11 대봉엘에스 주식회사 메실산 나파모스타트의 공결정다형 및 그의 제조방법

Also Published As

Publication number Publication date
ZA816363B (en) 1982-09-29
JPS611063B2 (https=) 1986-01-13

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