JP6700263B2 - エロビキシバットの結晶変態 - Google Patents
エロビキシバットの結晶変態 Download PDFInfo
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- JP6700263B2 JP6700263B2 JP2017519487A JP2017519487A JP6700263B2 JP 6700263 B2 JP6700263 B2 JP 6700263B2 JP 2017519487 A JP2017519487 A JP 2017519487A JP 2017519487 A JP2017519487 A JP 2017519487A JP 6700263 B2 JP6700263 B2 JP 6700263B2
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
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| EP14190290.8 | 2014-10-24 | ||
| EP14190290.8A EP3012252A1 (en) | 2014-10-24 | 2014-10-24 | Crystal modifications of elobixibat |
| PCT/EP2015/074573 WO2016062848A1 (en) | 2014-10-24 | 2015-10-23 | Crystal modifications of elobixibat |
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| JP2017537061A JP2017537061A (ja) | 2017-12-14 |
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2014
- 2014-10-24 EP EP14190290.8A patent/EP3012252A1/en not_active Withdrawn
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2015
- 2015-10-23 WO PCT/EP2015/074573 patent/WO2016062848A1/en not_active Ceased
- 2015-10-23 RU RU2017114109A patent/RU2017114109A/ru unknown
- 2015-10-23 US US15/519,808 patent/US10183920B2/en active Active
- 2015-10-23 EP EP21167339.7A patent/EP3904344A1/en not_active Withdrawn
- 2015-10-23 AU AU2015334883A patent/AU2015334883B2/en active Active
- 2015-10-23 JP JP2017519487A patent/JP6700263B2/ja active Active
- 2015-10-23 EP EP15784385.5A patent/EP3209649B1/en active Active
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| RU2017114109A3 (enExample) | 2019-04-30 |
| AU2015334883A1 (en) | 2017-03-23 |
| JP2017537061A (ja) | 2017-12-14 |
| EP3209649B1 (en) | 2021-04-21 |
| US20190177286A1 (en) | 2019-06-13 |
| CN107001301A (zh) | 2017-08-01 |
| WO2016062848A1 (en) | 2016-04-28 |
| CA2959760A1 (en) | 2016-04-28 |
| KR20170072908A (ko) | 2017-06-27 |
| CA2959760C (en) | 2023-10-10 |
| ES2874573T3 (es) | 2021-11-05 |
| US20170240516A1 (en) | 2017-08-24 |
| CN112375044A (zh) | 2021-02-19 |
| EP3012252A1 (en) | 2016-04-27 |
| EP3209649A1 (en) | 2017-08-30 |
| US10183920B2 (en) | 2019-01-22 |
| US10519120B2 (en) | 2019-12-31 |
| KR102498539B1 (ko) | 2023-02-09 |
| AU2015334883B2 (en) | 2019-10-24 |
| RU2017114109A (ru) | 2018-11-26 |
| EP3904344A1 (en) | 2021-11-03 |
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