JP5399262B2 - Ｌｘｒおよびｆｘｒのモジュレーター - Google Patents
Ｌｘｒおよびｆｘｒのモジュレーター Download PDFInfo
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- JP5399262B2 JP5399262B2 JP2009540497A JP2009540497A JP5399262B2 JP 5399262 B2 JP5399262 B2 JP 5399262B2 JP 2009540497 A JP2009540497 A JP 2009540497A JP 2009540497 A JP2009540497 A JP 2009540497A JP 5399262 B2 JP5399262 B2 JP 5399262B2
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- alkyl
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- haloalkyl
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
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| US86919806P | 2006-12-08 | 2006-12-08 | |
| US60/869,198 | 2006-12-08 | ||
| PCT/US2007/086787 WO2008073825A1 (en) | 2006-12-08 | 2007-12-07 | Lxr and fxr modulators |
Publications (3)
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| JP2010512342A JP2010512342A (ja) | 2010-04-22 |
| JP2010512342A5 JP2010512342A5 (https=) | 2012-01-26 |
| JP5399262B2 true JP5399262B2 (ja) | 2014-01-29 |
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| US (1) | US7998995B2 (https=) |
| EP (1) | EP2121621B1 (https=) |
| JP (1) | JP5399262B2 (https=) |
| KR (1) | KR20090094125A (https=) |
| CN (1) | CN101679297B (https=) |
| AU (1) | AU2007333194A1 (https=) |
| NO (1) | NO20092587L (https=) |
| WO (1) | WO2008073825A1 (https=) |
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| US11214536B2 (en) | 2017-11-21 | 2022-01-04 | Inspirna, Inc. | Polymorphs and uses thereof |
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2007
- 2007-12-07 KR KR1020097013701A patent/KR20090094125A/ko not_active Withdrawn
- 2007-12-07 EP EP07865385.4A patent/EP2121621B1/en active Active
- 2007-12-07 JP JP2009540497A patent/JP5399262B2/ja not_active Expired - Fee Related
- 2007-12-07 WO PCT/US2007/086787 patent/WO2008073825A1/en not_active Ceased
- 2007-12-07 CN CN2007800511486A patent/CN101679297B/zh not_active Expired - Fee Related
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- 2007-12-07 US US12/517,800 patent/US7998995B2/en active Active
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| Publication number | Priority date | Publication date | Assignee | Title |
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| US11214536B2 (en) | 2017-11-21 | 2022-01-04 | Inspirna, Inc. | Polymorphs and uses thereof |
| US11174220B2 (en) | 2019-12-13 | 2021-11-16 | Inspirna, Inc. | Metal salts and uses thereof |
| US11459292B2 (en) | 2019-12-13 | 2022-10-04 | Inspirna, Inc. | Metal salts and uses thereof |
| US11878956B2 (en) | 2019-12-13 | 2024-01-23 | Inspirna, Inc. | Metal salts and uses thereof |
| US12258303B2 (en) | 2019-12-13 | 2025-03-25 | Inspirna, Inc. | Metal salts and uses thereof |
Also Published As
| Publication number | Publication date |
|---|---|
| JP2010512342A (ja) | 2010-04-22 |
| WO2008073825A1 (en) | 2008-06-19 |
| KR20090094125A (ko) | 2009-09-03 |
| CN101679297B (zh) | 2012-01-11 |
| CN101679297A (zh) | 2010-03-24 |
| AU2007333194A1 (en) | 2008-06-19 |
| NO20092587L (no) | 2009-08-31 |
| US7998995B2 (en) | 2011-08-16 |
| US20100069367A1 (en) | 2010-03-18 |
| EP2121621B1 (en) | 2014-05-07 |
| EP2121621A1 (en) | 2009-11-25 |
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