|
US4172896A
(en)
|
1978-06-05 |
1979-10-30 |
Dainippon Pharmaceutical Co., Ltd. |
Methane-sulfonamide derivatives, the preparation thereof and composition comprising the same
|
|
US5049578A
(en)
|
1990-03-09 |
1991-09-17 |
E. R. Squibb & Sons, Inc. |
1-aroyl or 1-acyl-2-2pyrrolidinyl-3,5-dihydroxy alkanoic and alkenoic acids, salts, esters and lactones
|
|
GB9217295D0
(en)
|
1992-08-14 |
1992-09-30 |
Wellcome Found |
Controlled released tablets
|
|
US5541231A
(en)
|
1993-07-30 |
1996-07-30 |
Glaxo Wellcome Inc. |
Stabilized Pharmaceutical
|
|
US5358970A
(en)
|
1993-08-12 |
1994-10-25 |
Burroughs Wellcome Co. |
Pharmaceutical composition containing bupropion hydrochloride and a stabilizer
|
|
GB9315856D0
(en)
|
1993-07-30 |
1993-09-15 |
Wellcome Found |
Stabilized pharmaceutical
|
|
WO1999006023A1
(en)
|
1997-07-29 |
1999-02-11 |
Alcon Laboratories, Inc. |
Ophthalmic compositions containing galactomannan polymers and borate
|
|
CA2318920A1
(en)
|
1998-01-29 |
1999-08-05 |
James W. Young |
Pharmaceutical uses of optically pure (-)-bupropion
|
|
ES2196806T3
(es)
|
1998-05-08 |
2003-12-16 |
Smithkline Beecham Plc |
Derivados de fenilurea y de feniltiourea.
|
|
AU2910600A
(en)
|
1999-02-12 |
2000-08-29 |
Smithkline Beecham Plc |
Phenyl urea and phenyl thiourea derivatives
|
|
WO2000047576A1
(en)
|
1999-02-12 |
2000-08-17 |
Smithkline Beecham Plc |
Cinnamide derivatives as orexin-1 receptors antagonists
|
|
EP1150977B1
(en)
|
1999-02-12 |
2004-08-25 |
SmithKline Beecham plc |
Phenyl urea and phenyl thiourea derivatives as orexin receptor antagonists
|
|
CA2374793A1
(en)
|
1999-05-24 |
2000-11-30 |
Penglie Zhang |
Inhibitors of factor xa
|
|
US8889112B2
(en)
|
1999-09-16 |
2014-11-18 |
Ocularis Pharma, Llc |
Ophthalmic formulations including selective alpha 1 antagonists
|
|
AU779266B2
(en)
|
2000-05-11 |
2005-01-13 |
Banyu Pharmaceutical Co., Ltd. |
N-acyltetrahydroisoquinoline derivatives
|
|
EP1289955B1
(en)
|
2000-06-16 |
2005-04-13 |
Smithkline Beecham Plc |
Piperidines for use as orexin receptor antagonists
|
|
EP1353918B1
(en)
|
2000-11-28 |
2005-01-12 |
Smithkline Beecham Plc |
Morpholine derivatives as antagonists of orexin receptors
|
|
WO2002051232A2
(en)
|
2000-12-27 |
2002-07-04 |
Actelion Pharmaceuticals Ltd. |
Novel benzazepines and related heterocyclic derivatives
|
|
MXPA03010129A
(es)
|
2001-05-05 |
2004-03-10 |
Smithkline Beecham Plc |
N-aroilaminas-ciclicas.
|
|
EP1435955A2
(en)
|
2001-05-05 |
2004-07-14 |
SmithKline Beecham P.L.C. |
N-aroyl cyclic amine derivatives as orexin receptor antagonists
|
|
GB0115862D0
(en)
|
2001-06-28 |
2001-08-22 |
Smithkline Beecham Plc |
Compounds
|
|
GB0124463D0
(en)
|
2001-10-11 |
2001-12-05 |
Smithkline Beecham Plc |
Compounds
|
|
GB0126292D0
(en)
|
2001-11-01 |
2002-01-02 |
Smithkline Beecham Plc |
Compounds
|
|
GB0127145D0
(en)
|
2001-11-10 |
2002-01-02 |
Smithkline Beecham |
Compounds
|
|
GB0130341D0
(en)
|
2001-12-19 |
2002-02-06 |
Smithkline Beecham Plc |
Compounds
|
|
GB0130335D0
(en)
|
2001-12-19 |
2002-02-06 |
Smithkline Beecham Plc |
Compounds
|
|
GB0130393D0
(en)
|
2001-12-19 |
2002-02-06 |
Smithkline Beecham Plc |
Compounds
|
|
MXPA04002269A
(es)
|
2002-07-09 |
2004-06-29 |
Actelion Pharmaceuticals Ltd |
Derivados de 7,8,9,10-tetrahidro-6h-azepino,6,7,8,9-tetrahidro-pirido y 2,3-dihidro-2h-pirrolo[2,1-b]-quinazolinona.
|
|
ES2273083T3
(es)
|
2002-09-18 |
2007-05-01 |
Glaxo Group Limited |
N-aroilaminas ciclicas como antagonistas de los receptores de orexina.
|
|
US7279578B2
(en)
|
2002-10-11 |
2007-10-09 |
Actelion Pharmaceuticals Ltd. |
Sulfonylamino-acetic acid derivatives
|
|
GB0225938D0
(en)
|
2002-11-06 |
2002-12-11 |
Glaxo Group Ltd |
Novel compounds
|
|
GB0225884D0
(en)
|
2002-11-06 |
2002-12-11 |
Glaxo Group Ltd |
Novel compounds
|
|
GB0225944D0
(en)
|
2002-11-06 |
2002-12-11 |
Glaxo Group Ltd |
Novel compounds
|
|
US6951882B2
(en)
|
2002-12-12 |
2005-10-04 |
Janssen Pharmaceutica N.V. |
Substituted 4-phenyl-[1,3]-dioxanes
|
|
MXPA05010137A
(es)
|
2003-03-26 |
2005-11-16 |
Actelion Pharmaceuticals Ltd |
Derivados de tetrahidroisoquinolil acetamida para usarse como antagonistas del receptor de orexina.
|
|
WO2004096780A1
(en)
|
2003-04-28 |
2004-11-11 |
Actelion Pharmaceuticals Ltd |
Quinoxalinone-3- one derivatives as orexin receptor antagonists
|
|
US6933289B2
(en)
|
2003-07-01 |
2005-08-23 |
Allergan, Inc. |
Inhibition of irritating side effects associated with use of a topical ophthalmic medication
|
|
ATE444732T1
(de)
|
2003-08-07 |
2009-10-15 |
Allergan Inc |
Zusammensetzungen zur abgabe von therapeutika in die augen und verfahren zu ihrer herstellung und verwendung
|
|
US20050059744A1
(en)
|
2003-09-12 |
2005-03-17 |
Allergan, Inc. |
Methods and compositions for the treatment of pain and other alpha 2 adrenergic-mediated conditions
|
|
HUP0304101A3
(en)
|
2003-12-22 |
2008-10-28 |
Sanofi Aventis |
Pyrazole derivatives, process for producing them, their use, pharmaceutical compositions containing them and their intermediates
|
|
HUP0400405A3
(en)
|
2004-02-10 |
2009-03-30 |
Sanofi Synthelabo |
Pyrimidine derivatives, process for producing them, their use, pharmaceutical compositions containing them and their intermediates
|
|
WO2005118548A1
(en)
|
2004-03-01 |
2005-12-15 |
Actelion Pharmaceuticals Ltd |
Substituted 1,2,3,4-tetrahydroisoquinoline derivatives
|
|
WO2006067224A2
(en)
|
2004-12-23 |
2006-06-29 |
Biovitrum Ab (Publ) |
Spiro-benzodioxole and spiro-benzodioxane compounds as orexin receptor antagonists
|
|
US20080262046A1
(en)
|
2005-04-12 |
2008-10-23 |
Coleman Paul J |
Amidopropoxyphenyl Orexin Receptor Antagonists
|
|
WO2007008276A2
(en)
|
2005-05-03 |
2007-01-18 |
Ensemble Discovery Corporation |
Turnover probes and use thereof for nucleic acid detection
|
|
AU2006251590A1
(en)
|
2005-05-23 |
2006-11-30 |
Merck & Co., Inc. |
Proline bis-amide orexin receptor antagonists
|
|
JP2009503106A
(ja)
|
2005-08-04 |
2009-01-29 |
メルク エンド カムパニー インコーポレーテッド |
アミノエタンスルホンアミドオレキシン受容体アンタゴニスト
|
|
CA2620124A1
(en)
|
2005-08-26 |
2007-03-01 |
Merck And Co., Inc. |
Diazaspirodecane orexin receptor antagonists
|
|
WO2007061763A2
(en)
|
2005-11-22 |
2007-05-31 |
Merck & Co., Inc. |
Indole orexin receptor antagonists
|
|
CN101009515A
(zh)
|
2006-01-24 |
2007-08-01 |
华为技术有限公司 |
通信终端设备管理方法及通信终端
|
|
TW200800020A
(en)
|
2006-01-26 |
2008-01-01 |
Basf Ag |
Methods to use 3-pyridyl derivatives as pesticides
|
|
FR2896798A1
(fr)
|
2006-01-27 |
2007-08-03 |
Sanofi Aventis Sa |
Derives de sulfonamides, leur preparation et leur application en therapeutique
|
|
FR2896799B1
(fr)
|
2006-02-02 |
2008-03-28 |
Sanofi Aventis Sa |
Derives de sulfonamides, leur preparation et leur application en therapeutique
|
|
WO2007126934A2
(en)
|
2006-03-29 |
2007-11-08 |
Merck & Co., Inc. |
Amidoethylthioether orexin receptor antagonists
|
|
WO2007116374A1
(en)
|
2006-04-11 |
2007-10-18 |
Actelion Pharmaceuticals Ltd |
Novel sulfonamide compounds
|
|
CA2647077A1
(en)
|
2006-04-26 |
2007-11-01 |
Actelion Pharmaceuticals Ltd |
Pyrazolo-tetrahydro pyridine derivatives as orexin receptor antagonists
|
|
WO2007143813A1
(en)
|
2006-06-16 |
2007-12-21 |
Husky Injection Molding Systems Ltd. |
Preventative maintenance update system
|
|
PT2049529E
(pt)
|
2006-07-14 |
2010-10-13 |
Merck Sharp & Dohme |
Diazepan substituídos antagonistas do receptor da orexina
|
|
US8618102B2
(en)
|
2006-07-14 |
2013-12-31 |
Merck Sharp & Dohme Corp. |
Bridged diazepan orexin receptor antagonists
|
|
WO2008008551A2
(en)
|
2006-07-14 |
2008-01-17 |
Merck & Co., Inc. |
2-substituted proline bis-amide orexin receptor antagonists
|
|
AU2007285371A1
(en)
|
2006-08-15 |
2008-02-21 |
Actelion Pharmaceuticals Ltd. |
Azetidine compounds as orexin receptor antagonists
|
|
CA2659352A1
(en)
|
2006-08-28 |
2008-03-06 |
Actelion Pharmaceuticals Ltd |
1,4,5,6,7,8-hexahydro-1,2,5-triaza-azulene derivatives as orexin receptor antagonists
|
|
TW200823227A
(en)
|
2006-09-29 |
2008-06-01 |
Actelion Pharmaceuticals Ltd |
3-aza-bicyclo[3.1.0]hexane derivatives
|
|
PE20081229A1
(es)
|
2006-12-01 |
2008-08-28 |
Merck & Co Inc |
Antagonistas de receptor de orexina de diazepam sustituido
|
|
WO2008065626A2
(en)
|
2006-12-01 |
2008-06-05 |
Actelion Pharmaceuticals Ltd |
3-heteroaryl (amino or amido)-1- (biphenyl or phenylthiazolyl) carbonylpiperidine derivativesas orexin receptor inhibitors
|
|
CA2669561A1
(en)
|
2006-12-22 |
2008-07-03 |
Actelion Pharmaceuticals Ltd |
5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine derivatives
|
|
CL2007003827A1
(es)
|
2006-12-28 |
2008-09-26 |
Actelion Pharmaceuticals Ltd |
Compuestos derivados de n-(2-aza-biciclo(3.1.0)hex-3-ilmetil)amida; y su uso para prevenir o tratar la depresion, neurosis, esquizofrenia, ansiedad, adicciones, epilepsia, dolor, enfermedades cardiacas, entre otras.
|
|
WO2008087611A2
(en)
|
2007-01-19 |
2008-07-24 |
Actelion Pharmaceuticals Ltd |
Pyrrolidine- and piperidine- bis-amide derivatives
|
|
US8410142B2
(en)
|
2007-03-02 |
2013-04-02 |
Merck Sharp & Dohme Corp. |
Bipyridine carboxamide orexin receptor antagonists
|
|
JP5138708B2
(ja)
|
2007-03-05 |
2013-02-06 |
エフ.ホフマン−ラ ロシュ アーゲー |
オレキシンアンタゴニストとしてのアミノアミド
|
|
BRPI0808737A2
(pt)
|
2007-03-15 |
2014-08-12 |
Hoffmann La Roche |
Malonamidas como antagonistas de orexinas.
|
|
CL2008000836A1
(es)
|
2007-03-26 |
2008-11-07 |
Actelion Pharmaceuticals Ltd |
Compuestos derivados de tiazolidina, antagonistas del receptor de orexina; composicion farmaceutica que los comprende; y su uso en el tratamiento de neurosis emocional, depresion grave, trastornos psicoticos, alzheimer, parkinson, dolor, entre otras.
|
|
CA2681163A1
(en)
|
2007-04-04 |
2008-10-16 |
F. Hoffmann-La Roche Ag |
Heterocycles as orexin antagonists
|
|
ATE483707T1
(de)
|
2007-05-14 |
2010-10-15 |
Actelion Pharmaceuticals Ltd |
2-cyclopropylthiazolderivate
|
|
CA2688776A1
(en)
|
2007-05-18 |
2008-11-27 |
Merck & Co., Inc. |
Oxo bridged diazepan orexin receptor antagonists
|
|
EP2150115B1
(en)
|
2007-05-23 |
2013-09-18 |
Merck Sharp & Dohme Corp. |
Cyclopropyl pyrrolidine orexin receptor antagonists
|
|
WO2008147518A1
(en)
|
2007-05-23 |
2008-12-04 |
Merck & Co., Inc. |
Pyridyl piperidine orexin receptor antagonists
|
|
CN101730696B
(zh)
|
2007-07-03 |
2013-01-09 |
埃科特莱茵药品有限公司 |
3-氮杂-二环[3.3.0]辛烷化合物
|
|
CN101790515A
(zh)
|
2007-07-27 |
2010-07-28 |
埃科特莱茵药品有限公司 |
反式-3-氮杂-双环[3.1.0]己烷衍生物
|
|
BRPI0814593A2
(pt)
|
2007-07-27 |
2015-01-20 |
Actelion Pharmaceuticals Ltd |
Composto, composição farmacêutica que o contém e uso do composto.
|
|
US20090036422A1
(en)
|
2007-08-02 |
2009-02-05 |
Henner Knust |
Monoamide derivatives as orexin receptor antagonists
|
|
JP2010535769A
(ja)
|
2007-08-09 |
2010-11-25 |
メルク・シャープ・エンド・ドーム・コーポレイション |
ピリジンカルボキサミドオレキシン受容体アンタゴニスト
|
|
BRPI0823262A2
(pt)
|
2007-08-10 |
2013-09-24 |
Cortex Pharma Inc |
mÉtodo de tratamento de depressço respiratària e uso de um composto na fabricaÇço de um medicamento para o tratamento de depressço respiratària
|
|
MX2010001575A
(es)
|
2007-08-15 |
2010-03-15 |
Actelion Pharmaceuticals Ltd |
Derivados de 1,2-diamido-etileno como antagonistas de orexina.
|
|
US8288411B2
(en)
|
2007-09-24 |
2012-10-16 |
Actelion Pharmaceuticals Ltd. |
Pyrrolidines and piperidines as orexin receptor antagonists
|
|
US8362009B2
(en)
|
2007-10-29 |
2013-01-29 |
Merck Sharp & Dohme Corp. |
Substituted diazepan orexin receptor antagonists
|
|
WO2009079637A1
(en)
|
2007-12-18 |
2009-06-25 |
Concert Pharmaceuticals, Inc. |
Tetrahydroisoquinoline derivatives
|
|
EP2234999A1
(en)
|
2007-12-21 |
2010-10-06 |
F. Hoffmann-La Roche AG |
Heteroaryl derivatives as orexin receptor antagonists
|
|
AU2009207750B2
(en)
|
2008-01-21 |
2013-03-14 |
F. Hoffmann-La Roche Ag |
Sulfonamides as orexin antagonists
|
|
ATE517090T1
(de)
|
2008-02-12 |
2011-08-15 |
Hoffmann La Roche |
Piperidinsulfonamidderivate
|
|
CN101965343A
(zh)
|
2008-02-21 |
2011-02-02 |
埃科特莱茵药品有限公司 |
2-氮杂-双环[2.2.1]庚烷衍生物
|
|
GB0806536D0
(en)
|
2008-04-10 |
2008-05-14 |
Glaxo Group Ltd |
Novel compounds
|
|
US20110086889A1
(en)
|
2008-06-11 |
2011-04-14 |
Hamed Aissaoui |
Tetrazole compounds as orexin receptor antagonists
|
|
EP2297102A1
(en)
|
2008-06-16 |
2011-03-23 |
F. Hoffmann-La Roche AG |
Heteroaromatic monoamides as orexinin receptor antagonists
|
|
JP2011525910A
(ja)
|
2008-06-25 |
2011-09-29 |
アクテリオン ファーマシューティカルズ リミテッド |
5,6,7,8−テトラヒドロ−イミダゾ[1,5−a]ピラジン化合物
|
|
CA2729985A1
(en)
|
2008-07-07 |
2010-01-14 |
Actelion Pharmaceuticals Ltd |
Thiazolidine compounds as orexin receptor antagonists
|
|
KR101359852B1
(ko)
|
2008-07-29 |
2014-02-06 |
에프. 호프만-라 로슈 아게 |
오렉신 길항제로서 피롤리딘-3-일메틸-아민
|
|
AR072899A1
(es)
|
2008-08-07 |
2010-09-29 |
Merck Sharp & Dohme |
Derivados de terpiridina-carboxamida antagonistas de receptores de orexina, composiciones farmaceuticas que los contienen y uso de los mismos en el tratamiento del insomnio y la obesidad.
|
|
EP2161266A1
(en)
|
2008-08-22 |
2010-03-10 |
EVOTEC Neurosciences GmbH |
Benzofuran derivatives as orexin receptor antagonists
|
|
WO2010038200A1
(en)
|
2008-10-01 |
2010-04-08 |
Actelion Pharmaceuticals Ltd |
Oxazolidine compounds as orexin receptor antagonists
|
|
KR20110071004A
(ko)
|
2008-10-14 |
2011-06-27 |
액테리온 파마슈티칼 리미티드 |
페네틸아미드 유도체 및 이의 헤테로시클릭 유사체
|
|
EP2348856B1
(en)
|
2008-10-21 |
2013-08-14 |
Merck Sharp & Dohme Corp. |
2,4-disubstituted pyrrolidine orexin receptor antagonists
|
|
WO2010048016A1
(en)
|
2008-10-21 |
2010-04-29 |
Merck Sharp & Dohme Corp. |
2,3-disubstituted piperidine orexin receptor antagonists
|
|
JP2012506376A
(ja)
|
2008-10-21 |
2012-03-15 |
メルク・シャープ・エンド・ドーム・コーポレイション |
2,5−二置換モルホリンオレキシン受容体アンタゴニスト
|
|
CA2739916A1
(en)
|
2008-10-21 |
2010-04-29 |
Merck Sharp & Dohme Corp. |
2,5-disubstituted piperidine orexin receptor antagonists
|
|
AU2009307921A1
(en)
|
2008-10-21 |
2010-04-29 |
Merck Sharp & Dohme Corp. |
Disubstituted azepan orexin receptor antagonists
|
|
JP2012506374A
(ja)
|
2008-10-21 |
2012-03-15 |
メルク・シャープ・エンド・ドーム・コーポレイション |
2,5−二置換ピペリジンオレキシン受容体アンタゴニスト
|
|
AU2009308981A1
(en)
|
2008-10-30 |
2010-05-06 |
Merck Sharp & Dohme Corp. |
2,5-disubstituted phenyl carboxamide orexin receptor antagonists
|
|
AU2009308982A1
(en)
|
2008-10-30 |
2010-05-06 |
Merck Sharp & Dohme Corp. |
Pyridazine carboxamide orexin receptor antagonists
|
|
CA2741644C
(en)
|
2008-10-30 |
2013-05-07 |
Merck Sharp & Dohme Corp. |
Isonicotinamide orexin receptor antagonists
|
|
EP2358712A1
(en)
|
2008-11-26 |
2011-08-24 |
Glaxo Group Limited |
Piperidine derivatives useful as orexin receptor antagonists
|
|
EP2358711A1
(en)
|
2008-11-26 |
2011-08-24 |
Glaxo Group Limited |
Piperidine derivatives useful as orexin receptor antagonists
|
|
WO2010060472A1
(en)
|
2008-11-26 |
2010-06-03 |
Glaxo Group Limited |
Imidazopyridazine derivatives acting as orexin antagonists
|
|
AR074238A1
(es)
|
2008-12-02 |
2010-12-29 |
Glaxo Group Ltd |
Compuesto de n-{[(1r,4s,6r)-3-(2-piridinilcarbonil)-3-azabiciclo[4,1.0]hept-4-il]metil}-2-heteroarilamina, su uso para la preparacion de un medicamento util para el tratamiento de una enfermedad que requiere un antagonista del receptor de orexina humano y composicion farmaceutica que lo comprende
|
|
JP2012510493A
(ja)
|
2008-12-02 |
2012-05-10 |
グラクソ グループ リミテッド |
N−{[(ir、4s、6r)−3−(2−ピリジニルカルボニル)−3−アザビシクロ[4.1.0]ヘプタ−4−イル]メチル}−2−ヘテロアリールアミン誘導体およびその使用
|
|
JP2010155827A
(ja)
|
2008-12-04 |
2010-07-15 |
Takeda Chem Ind Ltd |
スピロ環化合物
|
|
GB0823467D0
(en)
|
2008-12-23 |
2009-01-28 |
Glaxo Group Ltd |
Novel Compounds
|
|
WO2010086366A1
(en)
|
2009-01-30 |
2010-08-05 |
Novartis Ag |
4-aryl-butane-1,3-diamides
|
|
BRPI1013933A2
(pt)
|
2009-04-24 |
2017-06-13 |
Glaxo Group Ltd |
3-azabiciclo [4.1.0] heptanos usados como antagonistas de orexina
|
|
WO2011005636A1
(en)
|
2009-07-09 |
2011-01-13 |
Merck Sharp & Dohme Corp. |
Tetrahydronapthyridine orexin receptor antagonists
|
|
EP2275421A1
(en)
|
2009-07-15 |
2011-01-19 |
Rottapharm S.p.A. |
Spiro amino compounds suitable for the treatment of inter alia sleep disorders and drug addiction
|
|
WO2011016234A1
(en)
|
2009-08-04 |
2011-02-10 |
Raqualia Pharma Inc. |
Picolinamide derivatives as ttx-s blockers
|
|
WO2011023578A1
(en)
|
2009-08-24 |
2011-03-03 |
Glaxo Group Limited |
5-methyl-piperidine derivatives as orexin receptor antagonists for the treatment of sleep disorder
|
|
JP2013502448A
(ja)
|
2009-08-24 |
2013-01-24 |
グラクソ グループ リミテッド |
オレキシンアンタゴニストとして用いられるピペリジン誘導体
|
|
US9062044B2
(en)
|
2009-10-23 |
2015-06-23 |
Janssen Pharmaceutica Nv |
Disubstituted octahydropyrrolo[3,4-c]pyrroles as orexin receptor modulators
|
|
RS54945B1
(sr)
|
2009-10-23 |
2016-11-30 |
Janssen Pharmaceutica Nv |
Disupstituisani oktahidropirolo[3,4-c]piroli kao oreksin receptor modulatori
|
|
WO2011050200A1
(en)
|
2009-10-23 |
2011-04-28 |
Janssen Pharmaceutica Nv |
Fused heterocyclic compounds as orexin receptor modulators
|
|
US20120196901A1
(en)
|
2009-10-29 |
2012-08-02 |
Merck Sharp & Dohme Corp. |
Tertiary amide orexin receptor antagonists
|
|
EP2504316A1
(en)
|
2009-11-23 |
2012-10-03 |
MSD Oss B.V. |
Heterocylic compounds as antagonists of the orexin receptors
|
|
WO2011073316A1
(en)
|
2009-12-18 |
2011-06-23 |
Novartis Ag |
4-aryl-butane-1,3-diamides
|
|
WO2011076744A1
(en)
|
2009-12-21 |
2011-06-30 |
Novartis Ag |
Disubstituted heteroaryl-fused pyridines
|
|
US8530648B2
(en)
|
2009-12-21 |
2013-09-10 |
Novartis Ag |
Diaza-spiro[5.5]undecanes
|
|
WO2011138266A1
(en)
|
2010-05-03 |
2011-11-10 |
Evotec Ag |
Indolizine and imidazopyridine derivatives as orexin receptor antagonists
|
|
WO2011138265A2
(en)
|
2010-05-03 |
2011-11-10 |
Evotec Ag |
Indole and indazole derivatives as orexin receptor antagonists
|
|
CA2821893A1
(en)
|
2010-12-17 |
2012-06-21 |
Taisho Pharmaceutical Co., Ltd. |
Pyrazole derivative
|
|
WO2012085857A1
(en)
|
2010-12-22 |
2012-06-28 |
Actelion Pharmaceuticals Ltd |
3,8-diaza-bicyclo[4.2.0]oct-3-yl amides
|
|
US20120165339A1
(en)
|
2010-12-22 |
2012-06-28 |
Eisai R&D Management Co., Ltd. |
Cyclopropane derivatives
|
|
US20120165331A1
(en)
|
2010-12-22 |
2012-06-28 |
Sangamesh Badiger |
Di/tri-aza-spiro-C9-C11alkanes
|
|
WO2012089606A1
(en)
|
2010-12-28 |
2012-07-05 |
Glaxo Group Limited |
Azabicyclo [4.1.0] hept - 4 - yl derivatives as human orexin receptor antagonists
|
|
WO2012089607A1
(en)
|
2010-12-28 |
2012-07-05 |
Glaxo Group Limited |
Novel compounds with a 3a-azabicyclo [4.1.0] heptane core acting on orexin receptors
|
|
ES2541531T3
(es)
|
2011-02-18 |
2015-07-21 |
Actelion Pharmaceuticals Ltd. |
Nuevos derivados de pirazol e imidazol útiles como antagonistas de orexina
|
|
WO2012114252A1
(en)
|
2011-02-21 |
2012-08-30 |
Actelion Pharmaceuticals Ltd |
Novel indole and pyrrolopyridine amides
|
|
WO2012145581A1
(en)
|
2011-04-20 |
2012-10-26 |
Janssen Pharmaceutica Nv |
Disubstituted octahy-dropyrrolo [3,4-c] pyrroles as orexin receptor modulators
|
|
WO2012153729A1
(ja)
|
2011-05-10 |
2012-11-15 |
大正製薬株式会社 |
ヘテロ芳香環誘導体
|
|
WO2013005755A1
(ja)
|
2011-07-05 |
2013-01-10 |
大正製薬株式会社 |
メチルピペリジン誘導体
|
|
WO2013050938A1
(en)
|
2011-10-04 |
2013-04-11 |
Actelion Pharmaceuticals Ltd |
3,7-diazabicyclo[3.3.1]nonane and 9-oxa-3,7-diazabicyclo[3.3.1]nonane derivatives
|
|
AR088352A1
(es)
|
2011-10-19 |
2014-05-28 |
Merck Sharp & Dohme |
Antagonistas del receptor de 2-piridiloxi-4-nitrilo orexina
|
|
EP2768305A4
(en)
|
2011-10-21 |
2015-04-29 |
Merck Sharp & Dohme |
2,5-DISUBSTITUTED THIOMORPHOLIN OREXINE RECEPTOR ANTAGONISTS
|
|
WO2013062858A1
(en)
|
2011-10-25 |
2013-05-02 |
Merck Sharp & Dohme Corp. |
Isoxazolopyridine orexin receptor antagonists
|
|
WO2013062857A1
(en)
|
2011-10-25 |
2013-05-02 |
Merck Sharp & Dohme Corp. |
Piperidinyl alkyne orexin receptor antagonists
|
|
SI2776430T1
(sl)
|
2011-11-08 |
2016-06-30 |
Actelion Pharmaceuticals Ltd. |
2-(1,2,3-triazol-2-il)benzamidni in 3-(1,2,3-triazol-2-il)pikolinamidni derivati kot antagonisti oreksinskega receptorja
|
|
ITMI20112329A1
(it)
|
2011-12-21 |
2013-06-22 |
Rottapharm Spa |
Nuovi derivati spiro amminici
|
|
HK1204955A1
(zh)
|
2012-02-07 |
2015-12-11 |
Eolas Therapeutics Inc. |
取代的脯氨酸/哌啶用作食慾素受體拮抗劑
|
|
US9440982B2
(en)
|
2012-02-07 |
2016-09-13 |
Eolas Therapeutics, Inc. |
Substituted prolines/piperidines as orexin receptor antagonists
|
|
ES2733750T3
(es)
|
2012-02-17 |
2019-12-02 |
Eisai R&D Man Co Ltd |
Métodos y compuestos útiles en la síntesis de antagonistas del receptor de orexina-2
|
|
ITMI20120322A1
(it)
|
2012-03-01 |
2013-09-02 |
Rottapharm Spa |
Composti di 4,4-difluoro piperidina
|
|
ITMI20120424A1
(it)
|
2012-03-19 |
2013-09-20 |
Rottapharm Spa |
Composti chimici
|
|
WO2015123355A1
(en)
|
2014-02-12 |
2015-08-20 |
Eolas Therapeutics, Inc. |
Substituted prolines / piperidines as orexin receptor antagonists
|