JP2013521301A5 - - Google Patents

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Publication number
JP2013521301A5
JP2013521301A5 JP2012556199A JP2012556199A JP2013521301A5 JP 2013521301 A5 JP2013521301 A5 JP 2013521301A5 JP 2012556199 A JP2012556199 A JP 2012556199A JP 2012556199 A JP2012556199 A JP 2012556199A JP 2013521301 A5 JP2013521301 A5 JP 2013521301A5
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JP
Japan
Prior art keywords
salt
trifluoromethyl
isopropoxy
pyrrolo
dihydro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
JP2012556199A
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English (en)
Japanese (ja)
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JP2013521301A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2011/026806 external-priority patent/WO2011109471A1/en
Publication of JP2013521301A publication Critical patent/JP2013521301A/ja
Publication of JP2013521301A5 publication Critical patent/JP2013521301A5/ja
Abandoned legal-status Critical Current

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JP2012556199A 2010-03-03 2011-03-02 Ｓ１ｐ１受容体修飾物質およびその結晶形の調製のためのプロセス Abandoned JP2013521301A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US33936210P 2010-03-03 2010-03-03
US61/339,362 2010-03-03
PCT/US2011/026806 WO2011109471A1 (en) 2010-03-03 2011-03-02 Processes for the preparation of s1p1 receptor modulators and crystalline forms thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2015142650A Division JP2015180706A (ja) 2010-03-03 2015-07-17 Ｓ１ｐ１受容体修飾物質およびその結晶形の調製のためのプロセス

Publications (2)

Publication Number Publication Date
JP2013521301A JP2013521301A (ja) 2013-06-10
JP2013521301A5 true JP2013521301A5 (enExample) 2014-04-17

Family

ID=43838192

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2012556199A Abandoned JP2013521301A (ja) 2010-03-03 2011-03-02 Ｓ１ｐ１受容体修飾物質およびその結晶形の調製のためのプロセス
JP2015142650A Abandoned JP2015180706A (ja) 2010-03-03 2015-07-17 Ｓ１ｐ１受容体修飾物質およびその結晶形の調製のためのプロセス

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2015142650A Abandoned JP2015180706A (ja) 2010-03-03 2015-07-17 Ｓ１ｐ１受容体修飾物質およびその結晶形の調製のためのプロセス

Country Status (8)

Country Link
US (2) US9085581B2 (enExample)
EP (1) EP2542554B1 (enExample)
JP (2) JP2013521301A (enExample)
CN (2) CN105503882B (enExample)
CA (1) CA2789480A1 (enExample)
ES (1) ES2558087T3 (enExample)
SG (2) SG183416A1 (enExample)
WO (1) WO2011109471A1 (enExample)

Families Citing this family (12)

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KR20190004843A (ko) * 2008-07-23 2019-01-14 아레나 파마슈티칼스, 인크. 자가면역성 및 염증성의 장애의 치료에 유용한 치환된 1,2,3,4-테트라히드로시클로펜타[ｂ]인돌-3-일)아세트산 유도체
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CN110545848A (zh) 2017-02-16 2019-12-06 艾尼纳制药公司 用于治疗具有肠外表现的炎症性肠病的化合物和方法
US12156866B2 (en) 2018-06-06 2024-12-03 Arena Pharmaceuticals, Inc. Methods of treating conditions related to the S1P1 receptor
EP3847158A1 (en) 2018-09-06 2021-07-14 Arena Pharmaceuticals, Inc. Compounds useful in the treatment of autoimmune and inflammatory disorders
JP7504880B2 (ja) * 2018-10-26 2024-06-24 ケロス セラピューティクス インコーポレイテッド Ａｌｋ２阻害剤の結晶形

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