JP2012521406A5 - - Google Patents

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Publication number
JP2012521406A5
JP2012521406A5 JP2012501412A JP2012501412A JP2012521406A5 JP 2012521406 A5 JP2012521406 A5 JP 2012521406A5 JP 2012501412 A JP2012501412 A JP 2012501412A JP 2012501412 A JP2012501412 A JP 2012501412A JP 2012521406 A5 JP2012521406 A5 JP 2012521406A5
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JP
Japan
Prior art keywords
dioxo
acetamide
pyrimidin
tetrahydrofuro
thiazol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2012501412A
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English (en)
Japanese (ja)
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JP2012521406A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2010/000840 external-priority patent/WO2010109329A1/en
Publication of JP2012521406A publication Critical patent/JP2012521406A/ja
Publication of JP2012521406A5 publication Critical patent/JP2012521406A5/ja
Pending legal-status Critical Current

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JP2012501412A 2009-03-23 2010-03-22 Ｔｒｐａ１調節因子としてのフロピリミジンジオン誘導体 Pending JP2012521406A (ja)

Applications Claiming Priority (13)

Application Number Priority Date Filing Date Title
IN665/MUM/2009 2009-03-23
IN665MU2009 2009-03-23
US17135509P 2009-04-21 2009-04-21
US61/171,355 2009-04-21
IN2213MU2009 2009-09-23
IN2213/MUM/2009 2009-09-23
US25199409P 2009-10-15 2009-10-15
US61/251,994 2009-10-15
IN2906/MUM/2009 2009-12-16
IN2906MU2009 2009-12-16
US29447010P 2010-01-12 2010-01-12
US61/294,470 2010-01-12
PCT/IB2010/000840 WO2010109329A1 (en) 2009-03-23 2010-03-22 Furopyrimidinedione derivatives as trpa1 modulators

Publications (2)

Publication Number Publication Date
JP2012521406A JP2012521406A (ja) 2012-09-13
JP2012521406A5 true JP2012521406A5 (enExample) 2013-05-02

Family

ID=42780205

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2012501412A Pending JP2012521406A (ja) 2009-03-23 2010-03-22 Ｔｒｐａ１調節因子としてのフロピリミジンジオン誘導体
JP2012501414A Expired - Fee Related JP5612070B2 (ja) 2009-03-23 2010-03-23 Ｔｒｐａ１調節因子としてのチエノピリミジンジオン誘導体

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2012501414A Expired - Fee Related JP5612070B2 (ja) 2009-03-23 2010-03-23 Ｔｒｐａ１調節因子としてのチエノピリミジンジオン誘導体

Country Status (22)

Country Link
US (4) US20120178766A1 (enExample)
EP (3) EP2411395B1 (enExample)
JP (2) JP2012521406A (enExample)
KR (2) KR20110128898A (enExample)
CN (3) CN102361874A (enExample)
AP (1) AP2948A (enExample)
AU (2) AU2010227225A1 (enExample)
BR (2) BRPI1013705A2 (enExample)
CA (2) CA2756535A1 (enExample)
DK (3) DK2411395T3 (enExample)
EA (2) EA201190138A1 (enExample)
ES (3) ES2424341T3 (enExample)
HU (1) HUE024538T2 (enExample)
IL (2) IL215177A (enExample)
MX (1) MX2011009822A (enExample)
PE (2) PE20120834A1 (enExample)
PL (3) PL2411395T3 (enExample)
PT (3) PT2411395E (enExample)
SG (4) SG184767A1 (enExample)
SI (3) SI2411395T1 (enExample)
WO (2) WO2010109329A1 (enExample)
ZA (2) ZA201107650B (enExample)

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WO2018162607A1 (en) * 2017-03-07 2018-09-13 F. Hoffmann-La Roche Ag Oxadiazole transient receptor potential channel inhibitors
CN109422749B (zh) * 2017-08-21 2023-01-24 重庆医药工业研究院有限责任公司 一种抑制单羧酸转运蛋白的嘧啶二酮衍生物
CN114555601B (zh) 2019-10-15 2024-04-02 勃林格殷格翰国际有限公司 新颖的四唑类
CA3193607A1 (en) * 2020-10-14 2022-04-21 Boehringer Ingelheim International Gmbh Tetrazole derivatives as trpa1 inhibitors
US11661427B2 (en) * 2020-10-14 2023-05-30 Boehringer Ingelheim International Gmbh Tetrazole derivatives as TRPA1 inhibitors
WO2022179469A1 (zh) * 2021-02-23 2022-09-01 南京明德新药研发有限公司 噻吩并嘧啶二酮类化合物及其应用
JP7565457B2 (ja) 2021-04-14 2024-10-10 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ＴＲＰＡ１阻害剤としての３Ｈ，４Ｈ－チエノ－［２，３－ｄ］ピリミジン－４－オン誘導体
CN114656480B (zh) * 2022-04-27 2024-01-26 成都施贝康生物医药科技有限公司 噻吩并嘧啶类化合物、异构体或盐及其制备方法和用途
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