|
US7407955B2
(en)
|
2002-08-21 |
2008-08-05 |
Boehringer Ingelheim Pharma Gmbh & Co., Kg |
8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
|
|
EP1687308B1
(en)
*
|
2003-11-17 |
2019-06-12 |
Merck & Cie |
Process for preparating (6R)-L-erythrotetrahydrobiopterin hydrochloride crystalline form B from other crystalline forms
|
|
CN103030617A
(zh)
*
|
2004-03-16 |
2013-04-10 |
贝林格尔.英格海姆国际有限公司 |
吡喃葡萄糖基取代的苯基衍生物、含该化合物的药物、其用途及其制造方法
|
|
WO2005118586A1
(en)
*
|
2004-06-02 |
2005-12-15 |
Sandoz Ag |
Meropenem intermediate in crystalline form
|
|
DE102004054054A1
(de)
|
2004-11-05 |
2006-05-11 |
Boehringer Ingelheim Pharma Gmbh & Co. Kg |
Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
|
|
DE602005009745D1
(de)
*
|
2004-12-16 |
2008-10-23 |
Boehringer Ingelheim Pharma |
Glucopyranosyl-substituierte benzen-derivate, medikamente mit solchen verbindungen, ihre verwendung und herstellungsverfahren dafür
|
|
JP5264183B2
(ja)
*
|
2005-02-23 |
2013-08-14 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
グルコピラノシル置換((ヘテロ)アリールエチニル−ベンジル)−ベンゼン誘導体及びナトリウム依存性グルコース共輸送体2(sglt2)インヒビターとしてのそれらの使用
|
|
ATE453656T1
(de)
*
|
2005-04-15 |
2010-01-15 |
Boehringer Ingelheim Int |
Glucopyranosyl-substituierte (heteroaryloxy- benzyl)-benzen-derivate als sglt-inhibitoren
|
|
UA91546C2
(uk)
*
|
2005-05-03 |
2010-08-10 |
Бьорінгер Інгельхайм Інтернаціональ Гмбх |
КРИСТАЛІЧНА ФОРМА 1-ХЛОР-4-(β-D-ГЛЮКОПІРАНОЗ-1-ИЛ)-2-[4-((S)-ТЕТРАГІДРОФУРАН-3-ІЛОКСИ)-БЕНЗИЛ]-БЕНЗОЛУ, СПОСІБ ЇЇ ОДЕРЖАННЯ ТА ЇЇ ЗАСТОСУВАННЯ ПРИ ПРИГОТУВАННІ ЛІКАРСЬКИХ ЗАСОБІВ
|
|
US7723309B2
(en)
*
|
2005-05-03 |
2010-05-25 |
Boehringer Ingelheim International Gmbh |
Crystalline forms of 1-chloro-4-(β-D-glucopyranos-1-yl)-2-[4-((R)-tetrahydrofuran-3-yloxy)-benzyl]-benzene, a method for its preparation and the use thereof for preparing medicaments
|
|
US7772191B2
(en)
|
2005-05-10 |
2010-08-10 |
Boehringer Ingelheim International Gmbh |
Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein
|
|
WO2007004230A2
(en)
*
|
2005-07-05 |
2007-01-11 |
Hetero Drugs Limited |
A novel process for the preparation of didanosine using novel intermediates
|
|
AR054871A1
(es)
*
|
2005-07-27 |
2007-07-25 |
Boehringer Ingelheim Int |
Derivados de (hetero)cicloalquiletinil-bencil)-benceno sustituidos con glucopiranosilo, medicamentos que contienen dichos compuestos, sus uso y proceso para su fabricacion
|
|
WO2007025943A2
(en)
*
|
2005-08-30 |
2007-03-08 |
Boehringer Ingelheim International Gmbh |
Glucopyranosyl-substituted benzyl-benzene derivatives, medicaments containing such compounds, their use and process for their manufacture
|
|
AU2006289093A1
(en)
*
|
2005-09-08 |
2007-03-15 |
Boehringer Ingelheim International Gmbh |
Crystalline forms of 1-chloro-4-(beta-D-glucopyranos-1-yl)-2-(4-ethynyl-benzyl)-benzene, methods for its preparation and the use thereof for preparing medicaments
|
|
AR056195A1
(es)
*
|
2005-09-15 |
2007-09-26 |
Boehringer Ingelheim Int |
Procedimientos para preparar derivados de (etinil-bencil)-benceno sustituidos de glucopiranosilo y compuestos intermedios de los mismos
|
|
BRPI0616040A2
(pt)
*
|
2005-09-21 |
2011-06-07 |
Nycomed Gmbh |
cloridrato de sulfonilpirról como inibidor de histona desacetilases
|
|
EP2404911A1
(en)
*
|
2005-10-31 |
2012-01-11 |
Janssen Pharmaceutica NV |
Novel processes for the preparation of piperazinyl and diazapanyl benzamide derivatives
|
|
AR059489A1
(es)
*
|
2006-02-15 |
2008-04-09 |
Boehringer Ingelheim Vetmed |
Derivados de benzonitrilo sustituidos con glucopiranosilo, composiciones farmaceuticas que contienen compuestos de este tipo, su uso y procedimiento para su fabricacion
|
|
PE20080697A1
(es)
*
|
2006-05-03 |
2008-08-05 |
Boehringer Ingelheim Int |
Derivados de benzonitrilo sustituidos con glucopiranosilo, composiciones farmaceuticas que contienen compuestos de este tipo, su uso y procedimiento para su fabricacion
|
|
EP2540725A1
(de)
|
2006-05-04 |
2013-01-02 |
Boehringer Ingelheim International GmbH |
Polymorphe von 1-((4-Methyl-chinazolin-2-yl)methyl)-3-methyl-7-(2-butin-1-yl)-8-(3-(R)-amino-piperidin-1-yl)xanthin
|
|
EP1852108A1
(en)
|
2006-05-04 |
2007-11-07 |
Boehringer Ingelheim Pharma GmbH & Co.KG |
DPP IV inhibitor formulations
|
|
PE20080251A1
(es)
|
2006-05-04 |
2008-04-25 |
Boehringer Ingelheim Int |
Usos de inhibidores de dpp iv
|
|
CA2656057C
(en)
*
|
2006-06-16 |
2012-10-02 |
H. Lundbeck A/S |
Crystalline forms of 4-[2-(4-methylphenylsulfanyl)-phenyl]piperidine with combined serotonin and norepinephrine reuptake inhibition for the treatment of neuropathic pain
|
|
WO2008020011A1
(en)
*
|
2006-08-15 |
2008-02-21 |
Boehringer Ingelheim International Gmbh |
Glucopyranosyl-substituted cyclopropylbenzene derivatives, pharmaceutical compositions containing such compounds, their use as sglt inhibitors and process for their manufacture
|
|
WO2008034859A1
(en)
*
|
2006-09-21 |
2008-03-27 |
Boehringer Ingelheim International Gmbh |
Glucopyranosyl-substituted difluorobenzyl-benzene derivatives, medicaments containing such compounds, their use and process for their manufacture
|
|
WO2008049923A1
(en)
*
|
2006-10-27 |
2008-05-02 |
Boehringer Ingelheim International Gmbh |
CRYSTALLINE FORM OF 4-(ß-D-GLUCOPYRANOS-1-YL)-1-METHYL-2-[4-((S)-TETRAHYDROFURAN-3-YLOXY)-BENZYL]-BENZENE, A METHOD FOR ITS PREPARATION AND THE USE THEREOF FOR PREPARING MEDICAMENTS
|
|
CA2667345C
(en)
*
|
2006-10-27 |
2016-03-22 |
Signal Pharmaceuticals, Llc |
Solid forms comprising 4-[9-(tetrahydro-furan-3-yl)-8-(2,4,6-trifluoro-phenylamino)-9h-purin-2-ylamino]-cyclohexan-1-ol, compositions thereof, and uses therewith
|
|
CA2668623A1
(en)
*
|
2006-11-06 |
2008-05-15 |
Boehringer Ingelheim International Gmbh |
Glucopyranosyl-substituted benzyl-benzonitrile derivatives, medicaments containing such compounds, their use and process for their manufacture
|
|
WO2008075736A1
(ja)
|
2006-12-21 |
2008-06-26 |
Astellas Pharma Inc. |
C-グリコシド誘導体の製造方法及びその合成中間体
|
|
WO2008101939A1
(en)
*
|
2007-02-21 |
2008-08-28 |
Boehringer Ingelheim International Gmbh |
Tetrasubstituted glucopyranosylated benzene derivatives, medicaments containing such compounds, their use and process for their manufacture
|
|
CL2008002427A1
(es)
|
2007-08-16 |
2009-09-11 |
Boehringer Ingelheim Int |
Composicion farmaceutica que comprende 1-cloro-4-(b-d-glucopiranos-1-il)-2-[4-((s)-tetrahidrofurano-3-iloxi)bencil]-benceno combinado con 1-[(4-metilquinazolin-2-il)metil]-3-metil-7-(2-butin-1-il)-8-(3-(r)-aminopiperidin-1-il)xantina; y su uso para tratar diabetes mellitus tipo 2.
|
|
NZ583369A
(en)
|
2007-08-23 |
2011-08-26 |
Theracos Inc |
Benzylbenzene derivatives and methods of use
|
|
JP5498392B2
(ja)
*
|
2007-11-30 |
2014-05-21 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
1,5−ジヒドロ−ピラゾロ[3,4−d]ピリミジン−4−オン誘導体及びcns障害の治療のためのpde9aモジュレーターとしてのそれらの使用
|
|
UA101004C2
(en)
|
2007-12-13 |
2013-02-25 |
Теракос, Инк. |
Derivatives of benzylphenylcyclohexane and use thereof
|
|
CL2008003653A1
(es)
|
2008-01-17 |
2010-03-05 |
Mitsubishi Tanabe Pharma Corp |
Uso de un inhibidor de sglt derivado de glucopiranosilo y un inhibidor de dppiv seleccionado para tratar la diabetes; y composicion farmaceutica.
|
|
EP2085397A1
(en)
*
|
2008-01-21 |
2009-08-05 |
Esteve Quimica, S.A. |
Crystalline form of abacavir
|
|
ES2541141T3
(es)
*
|
2008-01-31 |
2015-07-16 |
Astellas Pharma Inc. |
Composición farmacéutica para el tratamiento de las enfermedades del hígado graso
|
|
US7935817B2
(en)
*
|
2008-03-31 |
2011-05-03 |
Apotex Pharmachem Inc. |
Salt form and cocrystals of adefovir dipivoxil and processes for preparation thereof
|
|
UA105362C2
(en)
|
2008-04-02 |
2014-05-12 |
Бьорингер Ингельхайм Интернациональ Гмбх |
1-heterocyclyl-1, 5-dihydro-pyrazolo [3, 4-d] pyrimidin-4-one derivatives and their use as pde9a modulators
|
|
PE20091730A1
(es)
|
2008-04-03 |
2009-12-10 |
Boehringer Ingelheim Int |
Formulaciones que comprenden un inhibidor de dpp4
|
|
AR071318A1
(es)
*
|
2008-04-15 |
2010-06-09 |
Basilea Pharmaceutica Ag |
Benzhidril ester del acido (6r,7r)-7-{2-(5-amino-[1,2,4]tiadiazol-3-il)-2-[(z)-tritiloxiimino]-acetilamino}-3-[(r)-1'-terc-butoxicarbonil-2-oxo-[1,3']bipirrolidinil-(3e)-ilidenometil]-8-oxo-5-tia-1-aza-biciclo[4.2.0]oct-2-eno-2-carboxilico cristalino; su elaboracion y uso
|
|
US8097719B2
(en)
*
|
2008-07-15 |
2012-01-17 |
Genesen Labs |
Meropenem intermediate in novel crystalline form and a method of manufacture of meropenem
|
|
AU2009270936B2
(en)
|
2008-07-15 |
2014-12-18 |
Theracos, Inc. |
Deuterated benzylbenzene derivatives and methods of use
|
|
BRPI0916997A2
(pt)
|
2008-08-06 |
2020-12-15 |
Boehringer Ingelheim International Gmbh |
Inibidor de dpp-4 e seu uso
|
|
CN103910702A
(zh)
*
|
2008-08-22 |
2014-07-09 |
泰拉科斯有限公司 |
制备sglt2抑制剂的方法
|
|
AU2009286380B2
(en)
|
2008-08-28 |
2011-09-15 |
Pfizer Inc. |
Dioxa-bicyclo[3.2.1.]octane-2,3,4-triol derivatives
|
|
KR20110063447A
(ko)
|
2008-09-08 |
2011-06-10 |
베링거 인겔하임 인터내셔날 게엠베하 |
피라졸로피리미딘 및 cns 장애의 치료를 위한 이들의 용도
|
|
US20200155558A1
(en)
|
2018-11-20 |
2020-05-21 |
Boehringer Ingelheim International Gmbh |
Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug
|
|
AU2016213789B2
(en)
*
|
2009-02-13 |
2018-01-18 |
Boehringer Ingelheim International Gmbh |
SGLT-2 inhibitor for treating type 1 diabetes mellitus, type 2 diabetes mellitus, impaired glucose tolerance or hyperglycemia
|
|
AU2014200258B2
(en)
*
|
2009-02-13 |
2016-05-12 |
Boehringer Ingelheim International Gmbh |
SGLT-2 inhibitor for treating type 1 diabetes mellitus, type 2 diabetes mellitus, impaired glucose tolerance or hyperglycemia
|
|
JP5685550B2
(ja)
|
2009-02-13 |
2015-03-18 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
Sglt2阻害剤、dpp−iv阻害剤、更に必要により抗糖尿病薬を含む医薬組成物及びその使用
|
|
US20110014284A1
(en)
*
|
2009-02-13 |
2011-01-20 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical composition, pharmaceutical dosage form, process for their preparation, methods for treating and uses thereof
|
|
DK2396005T3
(da)
*
|
2009-02-13 |
2026-02-09 |
Boehringer Ingelheim Int |
Sglt2 hæmmer til at forbedre glykæmisk kontrol
|
|
UY32427A
(es)
*
|
2009-02-13 |
2010-09-30 |
Boheringer Ingelheim Internat Gmbh |
Composicion farmaceutica, forma farmaceutica, procedimiento para su preparacion, metodos de tratamiento y usos de la misma
|
|
PT2414363E
(pt)
|
2009-03-31 |
2014-02-26 |
Boehringer Ingelheim Int |
Derivados de 1-heterociclil-1,5-di-hidro-pirazolo[3,4- d]pirimidin-4-ona e sua utilização como moduladores de pde9a
|
|
TW201118099A
(en)
*
|
2009-08-12 |
2011-06-01 |
Boehringer Ingelheim Int |
New compounds for the treatment of CNS disorders
|
|
EA020798B1
(ru)
*
|
2009-09-30 |
2015-01-30 |
Бёрингер Ингельхайм Интернациональ Гмбх |
СПОСОБ ПОЛУЧЕНИЯ КРИСТАЛЛИЧЕСКОЙ ФОРМЫ 1-ХЛОР-4-(β-D-ГЛЮКОПИРАНОЗ-1-ИЛ)-2-[4-((S)-ТЕТРАГИДРОФУРАН-3-ИЛОКСИ)БЕНЗИЛ]БЕНЗОЛА
|
|
PT2486029E
(pt)
|
2009-09-30 |
2015-10-14 |
Boehringer Ingelheim Int |
Processos para a preparação de derivados de benzil-benzeno substituídos com glucopiranosilo
|
|
UY32919A
(es)
*
|
2009-10-02 |
2011-04-29 |
Boehringer Ingelheim Int |
Composición farmacéutica, forma de dosificación farmacéutica, procedimiento para su preparación, mé todos para su tratamiento y sus usos
|
|
US8163704B2
(en)
|
2009-10-20 |
2012-04-24 |
Novartis Ag |
Glycoside derivatives and uses thereof
|
|
RS53827B1
(sr)
|
2009-11-02 |
2015-06-30 |
Pfizer Inc. |
Derivati dioksa-biciklo[3.2.1]oktan-2,3,4-triola
|
|
KR20240090632A
(ko)
|
2009-11-27 |
2024-06-21 |
베링거 인겔하임 인터내셔날 게엠베하 |
리나글립틴과 같은 dpp-iv 억제제를 사용한 유전자형 검사된 당뇨병 환자의 치료
|
|
KR101713453B1
(ko)
|
2010-03-12 |
2017-03-07 |
오메로스 코포레이션 |
Pde10 억제제 및 관련 조성물 및 방법
|
|
EP2552442A1
(en)
*
|
2010-03-30 |
2013-02-06 |
Boehringer Ingelheim International GmbH |
Pharmaceutical composition comprising an sglt2 inhibitor and a ppar- gamma agonist and uses thereof
|
|
CN102946875A
(zh)
|
2010-05-05 |
2013-02-27 |
贝林格尔.英格海姆国际有限公司 |
组合疗法
|
|
WO2011153712A1
(en)
|
2010-06-12 |
2011-12-15 |
Theracos, Inc. |
Crystalline form of benzylbenzene sglt2 inhibitor
|
|
EP2603511B1
(en)
|
2010-08-12 |
2017-03-15 |
Boehringer Ingelheim International GmbH |
6-cycloalkyl-1, 5-dihydro-pyrazolo [3, 4-d] pyrimidin-4-one derivatives and their use as pde9a inhibitors
|
|
JP2013536859A
(ja)
*
|
2010-09-01 |
2013-09-26 |
アリーナ ファーマシューティカルズ, インコーポレイテッド |
5−ht2cアゴニストの非吸湿性塩
|
|
WO2012041898A1
(en)
|
2010-09-29 |
2012-04-05 |
Celon Pharma Sp. Z O.O. |
Combination of sglt2 inhibitor and a sugar compound for the treatment of diabetes
|
|
WO2012059416A1
(en)
|
2010-11-02 |
2012-05-10 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical combinations for the treatment of metabolic disorders
|
|
US20120283169A1
(en)
|
2010-11-08 |
2012-11-08 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical composition, methods for treating and uses thereof
|
|
AR083878A1
(es)
|
2010-11-15 |
2013-03-27 |
Boehringer Ingelheim Int |
Terapia antidiabetica vasoprotectora y cardioprotectora, linagliptina, metodo de tratamiento
|
|
US20130035281A1
(en)
|
2011-02-09 |
2013-02-07 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical composition, methods for treating and uses thereof
|
|
US8809345B2
(en)
|
2011-02-15 |
2014-08-19 |
Boehringer Ingelheim International Gmbh |
6-cycloalkyl-pyrazolopyrimidinones for the treatment of CNS disorders
|
|
AR085689A1
(es)
|
2011-03-07 |
2013-10-23 |
Boehringer Ingelheim Int |
Composiciones farmaceuticas de metformina, linagliptina y un inhibidor de sglt-2
|
|
BR112013031032A2
(pt)
|
2011-06-03 |
2016-11-29 |
Boehringer Ingelheim Int |
inibidores de sglt-2 para o tratamento de distúrbios metabólicos em pacientes tratados com agentes neurolépticos
|
|
US20130035298A1
(en)
*
|
2011-07-08 |
2013-02-07 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical composition, methods for treating and uses thereof
|
|
EP2760859A1
(en)
*
|
2011-09-30 |
2014-08-06 |
Sunshine Lake Pharma Co., Ltd |
Crystalline forms of azilsartan and preparation and uses thereof
|
|
US9555001B2
(en)
|
2012-03-07 |
2017-01-31 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical composition and uses thereof
|
|
US9192617B2
(en)
|
2012-03-20 |
2015-11-24 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical composition, methods for treating and uses thereof
|
|
WO2013152476A1
(en)
|
2012-04-10 |
2013-10-17 |
Theracos, Inc. |
Process for the preparation of benzylbenzene sglt2 inhibitors
|
|
US20130303446A1
(en)
|
2012-05-09 |
2013-11-14 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical combinations for the treatment of metabolic disorders
|
|
JP6218811B2
(ja)
|
2012-05-14 |
2017-10-25 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
Sirs及び/又は敗血症の治療に用いるdpp−4阻害薬としてのキサンチン誘導体
|
|
JP6224084B2
(ja)
|
2012-05-14 |
2017-11-01 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
糸球体上皮細胞関連障害及び/又はネフローゼ症候群の治療に用いるdpp−4阻害薬としてのキサンチン誘導体
|
|
PT2981269T
(pt)
|
2013-04-04 |
2023-10-10 |
Boehringer Ingelheim Vetmedica Gmbh |
Tratamento de distúrbios metabólicos em animais equinos
|
|
US11813275B2
(en)
*
|
2013-04-05 |
2023-11-14 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical composition, methods for treating and uses thereof
|
|
CA2812016A1
(en)
*
|
2013-04-05 |
2014-10-05 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical composition, methods for treating and uses thereof
|
|
CA2812519A1
(en)
|
2013-04-05 |
2014-10-05 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical composition, methods for treating and uses thereof
|
|
TR201901110T4
(tr)
|
2013-04-05 |
2019-02-21 |
Boehringer Ingelheim Int |
Empagliflozinin terapötik kullanımları.
|
|
HK1213818A1
(zh)
*
|
2013-04-05 |
2016-07-15 |
勃林格殷格翰国际有限公司 |
依帕列净的治疗用途
|
|
US20160000816A1
(en)
*
|
2013-04-05 |
2016-01-07 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical composition, methods for treating and uses thereof
|
|
EP4678242A3
(en)
*
|
2013-04-18 |
2026-03-18 |
Boehringer Ingelheim International GmbH |
Pharmaceutical composition, methods for treating and uses thereof
|
|
CN105611920B
(zh)
|
2013-10-12 |
2021-07-16 |
泰拉科斯萨普有限责任公司 |
羟基-二苯甲烷衍生物的制备
|
|
ES2969764T3
(es)
|
2013-12-17 |
2024-05-22 |
Boehringer Ingelheim Vetmedica Gmbh |
Un inhibidor de SGLT-2 para usar en el tratamiento de un trastorno metabólico en animales felinos
|
|
US9902751B2
(en)
|
2013-12-30 |
2018-02-27 |
Mylan Laboratories Limited |
Process for the preparation of empagliflozin
|
|
CN115671290A
(zh)
*
|
2014-01-23 |
2023-02-03 |
勃林格殷格翰动物保健有限公司 |
犬科动物中代谢紊乱的治疗
|
|
WO2015150299A2
(en)
|
2014-04-01 |
2015-10-08 |
Boehringer Ingelheim Vetmedica Gmbh |
Treatment of metabolic disorders in equine animals
|
|
NZ630803A
(en)
|
2014-04-28 |
2016-03-31 |
Omeros Corp |
Optically active pde10 inhibitor
|
|
NZ716494A
(en)
|
2014-04-28 |
2017-07-28 |
Omeros Corp |
Processes and intermediates for the preparation of a pde10 inhibitor
|
|
CN105384730A
(zh)
*
|
2014-09-03 |
2016-03-09 |
杭州普晒医药科技有限公司 |
依帕列净的晶型及其制备方法、药物组合物和用途
|
|
CN105481843A
(zh)
*
|
2014-09-19 |
2016-04-13 |
重庆医药工业研究院有限责任公司 |
一种恩格列净无定型物及其制备方法
|
|
WO2016046150A1
(en)
|
2014-09-25 |
2016-03-31 |
Boehringer Ingelheim Vetmedica Gmbh |
Combination treatment of sglt2 inhibitors and dopamine agonists for preventing metabolic disorders in equine animals
|
|
WO2016051368A1
(en)
|
2014-10-01 |
2016-04-07 |
Mylan Laboratories Ltd |
Complex of amorphous empagliflozin and a cyclodextrin
|
|
CZ2015110A3
(cs)
|
2015-02-18 |
2016-08-31 |
Zentiva, K.S. |
Pevné formy empagliflozinu
|
|
EA201791982A1
(ru)
|
2015-03-09 |
2020-02-17 |
Интекрин Терапьютикс, Инк. |
Способы лечения неалкогольной жировой болезни печени и/или липодистрофии
|
|
CZ2015279A3
(cs)
|
2015-04-24 |
2016-11-02 |
Zentiva, K.S. |
Pevné formy amorfního empagliflozinu
|
|
KR20170139074A
(ko)
|
2015-04-24 |
2017-12-18 |
오메로스 코포레이션 |
Pde10 억제제 및 관련 조성물 및 방법
|
|
CN104788438B
(zh)
*
|
2015-05-04 |
2018-02-02 |
南京华威医药科技集团有限公司 |
恩格列净b晶型及其制备
|
|
CN106317035A
(zh)
*
|
2015-06-23 |
2017-01-11 |
中美华世通生物医药科技(武汉)有限公司 |
恩格列净单晶及其制备方法和用途
|
|
KR102659761B1
(ko)
|
2015-08-27 |
2024-04-24 |
베링거잉겔하임베트메디카게엠베하 |
Sglt-2 억제제를 포함하는 액상 약제학적 조성물
|
|
EP3362055B1
(en)
|
2015-10-15 |
2023-01-18 |
Boehringer Ingelheim International GmbH |
Sglt-2 inhibitor for use in the treatment of a metabolic myopathy
|
|
WO2017079678A1
(en)
|
2015-11-04 |
2017-05-11 |
Omeros Corporation |
Solid state forms of a pde10 inhibitor
|
|
WO2017141202A1
(en)
*
|
2016-02-17 |
2017-08-24 |
Lupin Limited |
Complex of sglt2 inhibitor and process for preparation thereof
|
|
BR112018016001A2
(en)
*
|
2016-03-16 |
2018-12-18 |
Boehringer Ingelheim International Gmbh |
pharmaceutical composition, treatment methods and uses thereof
|
|
WO2017203457A1
(en)
*
|
2016-05-26 |
2017-11-30 |
Dr. Reddy's Laboratories Limited |
Solid state forms of empagliflozin
|
|
CN109310697A
(zh)
|
2016-06-10 |
2019-02-05 |
勃林格殷格翰国际有限公司 |
利格列汀和二甲双胍的组合
|
|
JP2019530722A
(ja)
|
2016-10-13 |
2019-10-24 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
グルコピラノシル置換ベンジル−ベンゼン誘導体を調製するための方法
|
|
US20210212968A1
(en)
|
2016-10-19 |
2021-07-15 |
Boehringer Ingelheim International Gmbh |
Combinations comprising an ssao/vap-1 inhibitor and a sglt2 inhibitor, uses thereof
|
|
KR20190084096A
(ko)
|
2016-11-10 |
2019-07-15 |
베링거 인겔하임 인터내셔날 게엠베하 |
약제학적 조성물, 치료 방법 및 이의 용도
|
|
US20200017483A1
(en)
*
|
2017-03-10 |
2020-01-16 |
Msn Laboratories Private Limited, R&D Center |
A process for the preparation of d-glucitol, 1,5-anhydro-1-c-[4-chloro-3-[[4- [[(3s)-tetrahydro-3-furanyl]oxy]phenyl]methyl]phenyl]-, ( 1 s)
|
|
JP2020515639A
(ja)
|
2017-04-03 |
2020-05-28 |
コヒラス・バイオサイエンシズ・インコーポレイテッド |
進行性核上性麻痺の処置のためのPPARγアゴニスト
|
|
CN111989103A
(zh)
|
2018-04-17 |
2020-11-24 |
勃林格殷格翰国际有限公司 |
药物组合物、其治疗方法和用途
|
|
CZ2018188A3
(cs)
|
2018-04-18 |
2019-10-30 |
Zentiva, K.S. |
Částice s obsahem amorfního empagliflozinu, způsob jejich přípravy a farmaceutický přípravek
|
|
KR102204439B1
(ko)
|
2018-05-14 |
2021-01-18 |
에이치케이이노엔 주식회사 |
Sglt-2 억제제 및 dpp-iv 억제제를 포함하는 약제학적 조성물
|
|
JP2021532191A
(ja)
|
2018-07-25 |
2021-11-25 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
アルポート症候群の治療に使用するためのエンパグリフロジン
|
|
WO2020039394A1
(en)
|
2018-08-24 |
2020-02-27 |
Novartis Ag |
New drug combinations
|
|
WO2020058095A1
(en)
|
2018-09-19 |
2020-03-26 |
Galenicum Health S.L.U. |
Pharmaceutical compositions of empagliflozin
|
|
US20210393621A1
(en)
|
2018-10-26 |
2021-12-23 |
The Research Foundation For The State University Of New York |
Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia
|
|
US12213970B2
(en)
|
2018-10-29 |
2025-02-04 |
Boehringer Ingelheim International Gmbh |
Pyridinyl sulfonamide derivatives, pharmaceutical compositions and uses thereof
|
|
KR102812426B1
(ko)
|
2018-10-29 |
2025-05-26 |
베링거 인겔하임 인터내셔날 게엠베하 |
피리디닐 설폰아미드 유도체, 약제학적 조성물 및 이의 용도
|
|
EP4064854A1
(en)
|
2019-11-28 |
2022-10-05 |
Boehringer Ingelheim Vetmedica GmbH |
Use of sglt-2 inhibitors in the drying-off of non-human mammals
|
|
WO2021123165A1
(en)
|
2019-12-19 |
2021-06-24 |
Krka, D.D., Novo Mesto |
Dosage form comprising amorphous solid solution of empagliflozin with polymer
|
|
KR102111248B1
(ko)
|
2019-12-30 |
2020-05-14 |
유니셀랩 주식회사 |
새로운 엠파글리플로진의 공결정
|
|
AU2021222297B2
(en)
|
2020-02-17 |
2026-01-22 |
Boehringer Ingelheim Vetmedica Gmbh |
Use of SGLT-2 inhibitors for the prevention and/or treatment of cardiac diseases in felines
|
|
IL296035A
(en)
|
2020-03-06 |
2022-10-01 |
Vertex Pharma |
Methods of treating apol-1 dependent focal segmental glomerulosclerosis
|
|
CN111303230B
(zh)
*
|
2020-03-09 |
2021-07-13 |
中国食品药品检定研究院 |
一种黄体酮共晶物及其制备方法和用途
|
|
KR102207319B1
(ko)
|
2020-03-23 |
2021-01-25 |
유니셀랩 주식회사 |
새로운 엠파글리플로진의 공결정
|
|
KR102150825B1
(ko)
|
2020-04-06 |
2020-09-03 |
유니셀랩 주식회사 |
새로운 sglt-2 억제제의 신규한 공결정
|
|
US20230110193A1
(en)
|
2020-04-07 |
2023-04-13 |
Boehringer Ingelheim International Gmbh |
Methods for the treatment of headache disorders
|
|
CA3180674A1
(en)
|
2020-04-22 |
2021-10-28 |
Bayer Aktiengesellschaft |
Combination of finerenone and a sglt2 inhibitor for the treatment and/or prevention of cardiovascular and/or renal diseases
|
|
WO2021250565A1
(en)
*
|
2020-06-10 |
2021-12-16 |
Hikal Limited |
An improved process for preparation of empagliflozin and its crystalline polymorph
|
|
WO2022051316A1
(en)
|
2020-09-03 |
2022-03-10 |
Coherus Biosciences, Inc. |
Fixed dose combinations of chs-131 and a sglt-2 inhibitor
|
|
KR102218323B1
(ko)
|
2020-09-09 |
2021-02-22 |
유니셀랩 주식회사 |
효율적이고 상전이가 되지 않는 엠파글리플로진 무정형의 제조방법
|
|
KR20220080880A
(ko)
|
2020-12-08 |
2022-06-15 |
주식회사 종근당 |
엠파글리플로진 공결정을 함유하는 약제학적 조성물
|
|
US20240269105A1
(en)
|
2021-07-28 |
2024-08-15 |
Boehringer Ingelheim Vetmedica Gmbh |
Use of sglt-2 inhibitors for the prevention and/or treatment of hypertension in non-human mammals
|
|
JP2024525981A
(ja)
|
2021-07-28 |
2024-07-12 |
ベーリンガー インゲルハイム フェトメディカ ゲーエムベーハー |
ヒト以外の哺乳動物における腎疾患の予防及び/又は治療のためのsglt-2阻害剤の使用
|
|
JP2024527434A
(ja)
|
2021-07-28 |
2024-07-24 |
ベーリンガー インゲルハイム フェトメディカ ゲーエムベーハー |
ネコ科動物を除く非ヒト哺乳動物、特にイヌ科動物における心臓疾患の予防及び/又は治療のためのsglt-2阻害剤の使用
|
|
US20250170128A1
(en)
|
2021-12-30 |
2025-05-29 |
NEWAMSTERDAM PHARMA B.V. (Dutch Chamber of Commerce No. 5597 1946) |
Obicetrapib and SGLT2 Inhibitor Combination
|
|
AU2023277704A1
(en)
|
2022-05-25 |
2024-12-05 |
Boehringer Ingelheim Vetmedica Gmbh |
Aqueous pharmaceutical compositions comprising sglt-2 inhibitors
|
|
EP4299055A1
(en)
|
2022-06-29 |
2024-01-03 |
Sanovel Ilac Sanayi Ve Ticaret A.S. |
Oral dosage formulations comprising empagliflozin
|
|
EP4342459A1
(en)
|
2022-09-20 |
2024-03-27 |
Galenicum Health S.L.U. |
Pharmaceutical compositions of empagliflozin
|
|
EP4378455A1
(en)
|
2022-11-29 |
2024-06-05 |
Sanovel Ilac Sanayi Ve Ticaret A.S. |
A pharmaceutical formulation comprising empagliflozin
|
|
EP4420658A1
(en)
|
2023-02-24 |
2024-08-28 |
Sanovel Ilac Sanayi Ve Ticaret A.S. |
A film coated tablet comprising empagliflozin
|
|
EP4676494A1
(en)
|
2023-03-06 |
2026-01-14 |
Boehringer Ingelheim Vetmedica GmbH |
Systems for delivery of liquid pharmaceutical compositions in particular comprising one or more sglt-2 inhibitor(s)
|
|
EP4442254A1
(en)
|
2023-04-04 |
2024-10-09 |
Sanovel Ilac Sanayi Ve Ticaret A.S. |
Film coated tablets comprising empagliflozin
|
|
EP4442253A1
(en)
|
2023-04-04 |
2024-10-09 |
Sanovel Ilac Sanayi Ve Ticaret A.S. |
A film coated tablet comprising empagliflozin and surfactant
|
|
EP4442252A1
(en)
|
2023-04-04 |
2024-10-09 |
Sanovel Ilac Sanayi Ve Ticaret A.S. |
A tablet formulation of a solid dispersion comprising empagliflozin
|
|
TW202446389A
(zh)
|
2023-04-24 |
2024-12-01 |
荷蘭商新阿姆斯特丹製藥公司 |
非晶形奧比特拉(obicetrapib)與sglt2抑制劑之組合
|
|
KR20260019532A
(ko)
|
2023-05-24 |
2026-02-10 |
베링거잉겔하임베트메디카게엠베하 |
하나 이상의 sglt-2 억제제와 텔미사르탄을 포함하는 비인간 포유류의 신장 질환 및/또는 고혈압의 병용 치료 및/또는 예방
|
|
US20240390317A1
(en)
|
2023-05-24 |
2024-11-28 |
Boehringer Ingelheim Vetmedica Gmbh |
Combination treatment and/or prevention of cardiac diseases in non-human mammals comprising one or more sglt-2 inhibitors and pimobendan and/or telmisartan
|
|
KR20250007816A
(ko)
|
2023-07-06 |
2025-01-14 |
주식회사 경보제약 |
엠파글리플로진 2l프롤린의 신규 결정형 및 이의 제조방법
|
|
KR20250038170A
(ko)
|
2023-09-11 |
2025-03-19 |
동광제약 주식회사 |
엠파글리플로진의 무정형 안정화 방법
|
|
TW202543596A
(zh)
|
2024-03-15 |
2025-11-16 |
法商因文帝華公司 |
預防接受過氧化物酶體增生劑活化受體(ppar)促效劑治療患者之血液病症
|
|
WO2025224069A1
(en)
|
2024-04-23 |
2025-10-30 |
Bayer Aktiengesellschaft |
Co-crystals of finerenone, pecavaptan, and sglt2 inhibitors
|
|
CN119735586A
(zh)
*
|
2025-02-25 |
2025-04-01 |
济南大学 |
一种恩格列净晶型iii及其制备方法
|