JP2008540687A5 - - Google Patents

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Publication number
JP2008540687A5
JP2008540687A5 JP2008512617A JP2008512617A JP2008540687A5 JP 2008540687 A5 JP2008540687 A5 JP 2008540687A5 JP 2008512617 A JP2008512617 A JP 2008512617A JP 2008512617 A JP2008512617 A JP 2008512617A JP 2008540687 A5 JP2008540687 A5 JP 2008540687A5
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JP
Japan
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alkyl
group
aryl
heteroaryl
cycloalkyl
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JP2008512617A
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English (en)
Japanese (ja)
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JP2008540687A (ja
JP5463034B2 (ja
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Priority claimed from PCT/US2006/020970 external-priority patent/WO2006128184A2/en
Publication of JP2008540687A publication Critical patent/JP2008540687A/ja
Publication of JP2008540687A5 publication Critical patent/JP2008540687A5/ja
Application granted granted Critical
Publication of JP5463034B2 publication Critical patent/JP5463034B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2008512617A 2005-05-20 2006-05-22 ピリミジン若しくはトリアジン縮合二環式メタロプロテアーゼ阻害薬 Expired - Fee Related JP5463034B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US68347005P 2005-05-20 2005-05-20
US60/683,470 2005-05-20
US70646505P 2005-08-08 2005-08-08
US60/706,465 2005-08-08
US73499105P 2005-11-09 2005-11-09
US60/734,991 2005-11-09
PCT/US2006/020970 WO2006128184A2 (en) 2005-05-20 2006-05-22 Pyrimidine or triazine fused bicyclic metalloprotease inhibitors

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP2013089076A Division JP5391351B2 (ja) 2005-05-20 2013-04-22 ヘテロ二環式メタロプロテアーゼ阻害薬
JP2013254709A Division JP2014088396A (ja) 2005-05-20 2013-12-10 ヘテロ二環式メタロプロテアーゼ阻害薬

Publications (3)

Publication Number Publication Date
JP2008540687A JP2008540687A (ja) 2008-11-20
JP2008540687A5 true JP2008540687A5 (enExample) 2009-07-30
JP5463034B2 JP5463034B2 (ja) 2014-04-09

Family

ID=37239216

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2008512617A Expired - Fee Related JP5463034B2 (ja) 2005-05-20 2006-05-22 ピリミジン若しくはトリアジン縮合二環式メタロプロテアーゼ阻害薬
JP2013089076A Expired - Fee Related JP5391351B2 (ja) 2005-05-20 2013-04-22 ヘテロ二環式メタロプロテアーゼ阻害薬
JP2013254709A Withdrawn JP2014088396A (ja) 2005-05-20 2013-12-10 ヘテロ二環式メタロプロテアーゼ阻害薬

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2013089076A Expired - Fee Related JP5391351B2 (ja) 2005-05-20 2013-04-22 ヘテロ二環式メタロプロテアーゼ阻害薬
JP2013254709A Withdrawn JP2014088396A (ja) 2005-05-20 2013-12-10 ヘテロ二環式メタロプロテアーゼ阻害薬

Country Status (13)

Country Link
US (2) US20060293345A1 (enExample)
EP (1) EP1910367A2 (enExample)
JP (3) JP5463034B2 (enExample)
KR (1) KR20080087070A (enExample)
CN (1) CN101238127A (enExample)
AU (1) AU2006251989B2 (enExample)
BR (1) BRPI0609802A2 (enExample)
CA (1) CA2608890C (enExample)
CR (1) CR9614A (enExample)
EA (1) EA013525B1 (enExample)
IL (1) IL187495A0 (enExample)
NO (1) NO20076554L (enExample)
WO (1) WO2006128184A2 (enExample)

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HK1207562A1 (en) 2012-01-18 2016-02-05 苏州泰飞尔医药有限公司 High penetration prodrug compositions and pharmaceutical composition thereof for treatment of pulmonary conditions
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