JP2004513168A5 - - Google Patents

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JP2004513168A5
JP2004513168A5 JP2002541095A JP2002541095A JP2004513168A5 JP 2004513168 A5 JP2004513168 A5 JP 2004513168A5 JP 2002541095 A JP2002541095 A JP 2002541095A JP 2002541095 A JP2002541095 A JP 2002541095A JP 2004513168 A5 JP2004513168 A5 JP 2004513168A5
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JP
Japan
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alkyl
formula
methyl
ring
compound
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JP2002541095A
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English (en)
Japanese (ja)
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JP2004513168A (ja
JP4234426B2 (ja
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Priority claimed from PCT/EP2001/012785 external-priority patent/WO2002038561A1/en
Publication of JP2004513168A publication Critical patent/JP2004513168A/ja
Publication of JP2004513168A5 publication Critical patent/JP2004513168A5/ja
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Publication of JP4234426B2 publication Critical patent/JP4234426B2/ja
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JP2002541095A 2000-11-07 2001-11-05 プロテインキナーゼcインヒビターとしてのインドリルマレイミド誘導体 Expired - Fee Related JP4234426B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24640000P 2000-11-07 2000-11-07
US28370501P 2001-04-13 2001-04-13
PCT/EP2001/012785 WO2002038561A1 (en) 2000-11-07 2001-11-05 Indolylmaleimide derivatives as protein kinase c inhibitors

Publications (3)

Publication Number Publication Date
JP2004513168A JP2004513168A (ja) 2004-04-30
JP2004513168A5 true JP2004513168A5 (https=) 2005-04-21
JP4234426B2 JP4234426B2 (ja) 2009-03-04

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JP2002541095A Expired - Fee Related JP4234426B2 (ja) 2000-11-07 2001-11-05 プロテインキナーゼcインヒビターとしてのインドリルマレイミド誘導体

Country Status (30)

Country Link
EP (2) EP1337527B1 (https=)
JP (1) JP4234426B2 (https=)
KR (3) KR100916613B1 (https=)
CN (1) CN1253449C (https=)
AR (1) AR035211A1 (https=)
AT (1) ATE445613T1 (https=)
AU (3) AU2002221810B2 (https=)
BR (1) BRPI0115193B1 (https=)
CA (1) CA2428133C (https=)
CY (1) CY1110564T1 (https=)
CZ (1) CZ307144B6 (https=)
DE (1) DE60140201D1 (https=)
DK (1) DK1337527T3 (https=)
EC (1) ECSP104578A (https=)
ES (1) ES2332770T3 (https=)
HU (1) HU228999B1 (https=)
IL (3) IL155618A0 (https=)
MX (1) MXPA03004037A (https=)
MY (2) MY139979A (https=)
NO (1) NO327427B1 (https=)
NZ (2) NZ535616A (https=)
PE (1) PE20020544A1 (https=)
PL (1) PL208794B1 (https=)
PT (1) PT1337527E (https=)
RU (2) RU2329263C2 (https=)
SG (1) SG159378A1 (https=)
SI (1) SI1337527T1 (https=)
SK (1) SK287919B6 (https=)
TW (2) TWI290553B (https=)
WO (1) WO2002038561A1 (https=)

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EP2338486A1 (en) 2009-12-18 2011-06-29 Johannes Gutenberg-Universität Mainz 3-(indolyl)- or 3-(azaindolyl)-4-arylmaleimide derivatives for use in the treatment of colon and gastric adenocarcinoma
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EP2474541A1 (en) 2010-12-23 2012-07-11 Johannes- Gutenberg-Universität Mainz Conjugated 3-(indolyl)- and 3-(azaindolyl)-4-arylmaleimide compounds and their use in tumor treatment
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JP2014518256A (ja) 2011-06-27 2014-07-28 ノバルティス アーゲー テトラヒドロ−ピリド−ピリミジン誘導体の固体形態および塩類
GB201111427D0 (en) * 2011-07-05 2011-08-17 Amakem Nv Novel bisindolylmaleimides, pan-pkc inhibitors
KR20140058543A (ko) 2011-07-08 2014-05-14 노파르티스 아게 신규 피롤로 피리미딘 유도체
EP2567959B1 (en) 2011-09-12 2014-04-16 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
US8846712B2 (en) 2011-09-12 2014-09-30 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
EP2760862B1 (en) 2011-09-27 2015-10-21 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
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JP5903499B2 (ja) 2011-12-22 2016-04-13 ノバルティス アーゲー ジヒドロ−ベンゾ−オキサジンおよびジヒドロ−ピリド−オキサジン誘導体
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