IS4822A - Afleiður af setinni 4-hýdroxýfenýlalkanósýru með gerandefnisvirkni á PPAR-gamma, lyfjaefnablöndur sem innihalda þær, notkun þeirra og aðferð til framleiðslu þeirra - Google Patents

Afleiður af setinni 4-hýdroxýfenýlalkanósýru með gerandefnisvirkni á PPAR-gamma, lyfjaefnablöndur sem innihalda þær, notkun þeirra og aðferð til framleiðslu þeirra

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Publication number
IS4822A
IS4822A IS4822A IS4822A IS4822A IS 4822 A IS4822 A IS 4822A IS 4822 A IS4822 A IS 4822A IS 4822 A IS4822 A IS 4822A IS 4822 A IS4822 A IS 4822A
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derivatives
substituted
production
pharmaceutical preparations
agonist activity
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IS4822A
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English (en)
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IS1869B (is
Inventor
Mark Willson Timothy
Anthony Mook Jrth Robert
Kaldor Istvan
Richard Henke Brad
Norman Deaton David
Edmond Cobb Jeffrey
Jude Sharp Matthew
Alan Erickson Greg
Evan Boswell Grady
Loren Collins Jon
Brackeen Markus
Mark O'callaghan John
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Glaxo Group Limited
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Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Publication of IS4822A publication Critical patent/IS4822A/is
Publication of IS1869B publication Critical patent/IS1869B/is

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
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    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
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    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
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IS4822A 1996-02-28 1998-08-12 Afleiður af setinni 4-hýdroxýfenýlalkanósýru með gerandefnisvirkni á PPAR-gamma, lyfjaefnablöndur sem innihalda þær, notkun þeirra og aðferð til framleiðslu þeirra IS1869B (is)

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